Detection of recombinant and endogenous mouse melatonin receptors by monoclonal antibodies targeting the C-terminal domain

The orphan GPR50 receptor promotes constitutive TGFβ receptor signaling and protects against cancer development

(2018) Stefanie Wojciech et al.   Nature Communications

Cannabidiol skews biased agonism at cannabinoid CB1 and CB2 receptors with smaller effect in CB1-CB2 heteroreceptor complexes

(2018) Gemma Navarro et al.   BIOCHEMICAL PHARMACOLOGY

Melatonin receptors limit dopamine reuptake by regulating dopamine transporter cell-surface exposure

(2018) Abla Benleulmi-Chaachoua et al.   CELLULAR AND MOLECULAR LIFE SCIENCES

Orexin A/Hypocretin Modulates Leptin Receptor-Mediated Signaling by Allosteric Modulations Mediated by the Ghrelin GHS-R1A Receptor in Hypothalamic Neurons

(2017) Mireia Medrano et al.   MOLECULAR NEUROBIOLOGY

Targeting Melatonin MT2 Receptors: A Novel Pharmacological Avenue for Inflammatory and Neuropathic Pain

(2017) Luca Posa et al.   CURRENT MEDICINAL CHEMISTRY

Update on melatonin receptors: IUPHAR Review 20

(2016) Ralf Jockers et al.   BRITISH JOURNAL OF PHARMACOLOGY

The Difficult Journey from Genome-wide Association Studies to Pathophysiology: The Melatonin Receptor 1B (MT2) Paradigm

(2016) Amélie Bonnefond et al.   Cell Metabolism

Amyloid β peptide directly impairs pineal gland melatonin synthesis and melatonin receptor signaling through the ERK pathway

(2015) Erika Cecon et al.   FASEB JOURNAL

Convergence of Melatonin and Serotonin (5-HT) Signaling at MT2/5-HT2CReceptor Heteromers

(2015) Maud Kamal et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Anatomical and cellular localization of melatonin MT1and MT2receptors in the adult rat brain

(2015) Baptiste Lacoste et al.   JOURNAL OF PINEAL RESEARCH

Generic GPCR residue numbers – aligning topology maps while minding the gaps

(2015) Vignir Isberg et al.   TRENDS IN PHARMACOLOGICAL SCIENCES

Understanding melatonin receptor pharmacology: Latest insights from mouse models, and their relevance to human disease

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Alterations of melatonin receptors MT1 and MT2 in the hypothalamic suprachiasmatic nucleus during depression

(2013) Ying-Hui Wu et al.   JOURNAL OF AFFECTIVE DISORDERS

Distribution of MT1 Melatonin Receptor Promoter-Driven RFP Expression in the Brains of BAC C3H/HeN Transgenic Mice

(2013) EB Adamah-Biassi et al.   JOURNAL OF HISTOCHEMISTRY & CYTOCHEMISTRY

MT1 and MT2 Melatonin Receptors: Ligands, Models, Oligomers, and Therapeutic Potential

(2013) Darius. P. Zlotos et al.   JOURNAL OF MEDICINAL CHEMISTRY

Heteromeric MT1/MT2 Melatonin Receptors Modulate Photoreceptor Function

(2013) K. Baba et al.   Science Signaling

Molecular pharmacology of the mouse melatonin receptors MT1 and MT2

(2011) Séverine Devavry et al.   EUROPEAN JOURNAL OF PHARMACOLOGY

Localization of Melatonin Receptor 1 in Mouse Retina and Its Role in the Circadian Regulation of the Electroretinogram and Dopamine Levels

(2011) Anamika Sengupta et al.   PLoS One

Molecular organization and dynamics of the melatonin MT1 receptor/RGS20/Gi protein complex reveal asymmetry of receptor dimers for RGS and Gi coupling

(2010) Pascal Maurice et al.   EMBO JOURNAL

Expression of the orphan GPR50 protein in rodent and human dorsomedial hypothalamus, tanycytes and median eminence

(2010) Anissa Sidibe et al.   JOURNAL OF PINEAL RESEARCH

International Union of Basic and Clinical Pharmacology. LXXV. Nomenclature, Classification, and Pharmacology of G Protein-Coupled Melatonin Receptors

(2010) M. L. Dubocovich et al.   PHARMACOLOGICAL REVIEWS

Molecular cloning and pharmacological characterization of rat melatonin MT1 and MT2 receptors

(2008) Valérie Audinot et al.   BIOCHEMICAL PHARMACOLOGY

GPR50 is the mammalian ortholog of Mel1c: Evidence of rapid evolution in mammals

(2008) Laurence Dufourny et al.   BMC EVOLUTIONARY BIOLOGY

The PDZ Protein Mupp1 Promotes GiCoupling and Signaling of the Mt1Melatonin Receptor

(2008) Jean-Luc Guillaume et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Function and expression of melatonin receptors on human pancreatic islets

(2008) Reshma D. Ramracheya et al.   JOURNAL OF PINEAL RESEARCH