[18 F]FPyZIDE: A versatile prosthetic reagent for the fluorine-18 radiolabeling of biologics via copper-catalyzed or strain-promoted alkyne-azide cycloadditions

Synthesis and Biologic Evaluation of a Novel18F-Labeled Adnectin as a PET Radioligand for Imaging PD-L1 Expression

(2017) David J. Donnelly et al.   JOURNAL OF NUCLEAR MEDICINE

[18F]Fluoroalkyl azides for rapid radiolabeling and (Re)investigation of their potential towards in vivo click chemistry

(2017) Christoph Denk et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Clinical Applications of Radiolabeled Peptides for PET

(2017) Isaac M. Jackson et al.   SEMINARS IN NUCLEAR MEDICINE

Copper Catalysis in Living Systems and In Situ Drug Synthesis

(2016) Jessica Clavadetscher et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Click Chemistry and Radiochemistry: The First 10 Years

(2016) Jan-Philip Meyer et al.   BIOCONJUGATE CHEMISTRY

Extent of the Oxidative Side Reactions to Peptides and Proteins During the CuAAC Reaction

(2016) Siheng Li et al.   BIOCONJUGATE CHEMISTRY

Pretargeted PET Imaging Using a Site-Specifically Labeled Immunoconjugate

(2016) Brendon E. Cook et al.   BIOCONJUGATE CHEMISTRY

18F-Containing Positron Emission Tomography Probe Conjugation Methodology for Biologics as Specific Binders for Tumors

(2016) Kenji Arimitsu et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

Efficient synthesis of [18F]FPyME: A new approach for the preparation of maleimide-containing prosthetic groups for the conjugation with thiols

(2016) Melanie Cavani et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

Development and Applications of the Copper-Catalyzed Azide-Alkyne Cycloaddition (CuAAC) as a Bioorthogonal Reaction

(2016) Li Li et al.   MOLECULES

Synthesis, radiolabeling with fluorine-18 and preliminary in vivo evaluation of a heparan sulphate mimetic as potent angiogenesis and heparanase inhibitor for cancer applications

(2016) B. Kuhnast et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Development of 6-[18F]fluoro-carbohydrate-based prosthetic groups and their conjugation to peptides via click chemistry

(2015) Charlotte Collet et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

Synthesis of68Ga-labeled NOTA-RGD-GE11 heterodimeric peptide for dual integrin and epidermal growth factor receptor-targeted tumor imaging

(2015) Hung-Man Yu et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

Radiopeptides for Imaging and Therapy: A Radiant Future

(2015) K. L. S. Chatalic et al.   JOURNAL OF NUCLEAR MEDICINE

Radiofluorination of PSMA-HBED via Al18F2+ Chelation and Biological Evaluations In Vitro

(2015) Noeen Malik et al.   MOLECULAR IMAGING AND BIOLOGY

18F-Trifluoroborate Derivatives of [Des-Arg10]Kallidin for Imaging Bradykinin B1 Receptor Expression with Positron Emission Tomography

(2015) Zhibo Liu et al.   MOLECULAR PHARMACEUTICS

Bioorthogonal Reactions for Labeling Proteins

(2014) Kathrin Lang et al.   ACS Chemical Biology

Synthesis and in Vitro and in Vivo Evaluation of SiFA-Tagged Bombesin and RGD Peptides as Tumor Imaging Probes for Positron Emission Tomography

(2014) Simon Lindner et al.   BIOCONJUGATE CHEMISTRY

Click Chemistry in Complex Mixtures: Bioorthogonal Bioconjugation

(2014) Craig S. McKay et al.   CHEMISTRY & BIOLOGY

Prospective of 68Ga-Radiopharmaceutical Development

(2014) Irina Velikyan   Theranostics

18F-Labeling Using Click Cycloadditions

(2014) Kathrin Kettenbach et al.   Biomed Research International

Dual isotope labeling: Conjugation of 32P-oligonucleotides with 18F-aryltrifluoroborate via copper(I) catalyzed cycloaddition

(2013) Ying Li et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

2-Fluoropyridine prosthetic compounds for the 18F labeling of bombesin analogues

(2013) James Inkster et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Recent Trends in Bioorthogonal Click-Radiolabeling Reactions Using Fluorine-18

(2013) Marc Pretze et al.   MOLECULES

Rearrangements and addition reactions of biarylazacyclooctynones and the implications to copper-free click chemistry

(2013) Mariya Chigrinova et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Optimization of acetonitrile co-solvent and copper stoichiometry for pseudo-ligandless click chemistry with nucleic acids

(2012) Eduardo Paredes et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Labeling Strategies of Peptides with 18F for Positron Emission Tomography

(2012) D. E. Olberg et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

64Cu-NO2A-RGD-Glu-6-Ahx-BBN(7-14)NH2: a heterodimeric targeting vector for positron emission tomography imaging of prostate cancer

(2012) Andrew B. Jackson et al.   NUCLEAR MEDICINE AND BIOLOGY

Evaluation of an integrin αvβ6-specific peptide labeled with [18F]fluorine by copper-free, strain-promoted click chemistry

(2012) Sven H. Hausner et al.   NUCLEAR MEDICINE AND BIOLOGY

[18F]Si-RiboRGD: From Design and Synthesis to the Imaging of αvβ3 Integrins in Melanoma Tumors

(2012) Eric Amigues et al.   ChemPlusChem

From Mechanism to Mouse: A Tale of Two Bioorthogonal Reactions

(2011) Ellen M. Sletten et al.   ACCOUNTS OF CHEMICAL RESEARCH

Cu-free click cycloaddition reactions in chemical biology

(2010) John C. Jewett et al.   CHEMICAL SOCIETY REVIEWS

In vitro reactive oxygen species production by histatins and copper(I,II)

(2008) Eric A. Houghton et al.   JOURNAL OF BIOLOGICAL INORGANIC CHEMISTRY

[18F]FPyKYNE, a fluoropyridine-based alkyne reagent designed for the fluorine-18 labelling of macromolecules using click chemistry

(2008) Bertrand Kuhnast et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

Radiosynthesis and bioconjugation of [18F]FPy5yne, a prosthetic group for the18F labeling of bioactive peptides

(2008) James A. H. Inkster et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS