Remarkable Enhancement in Boron Uptake Within Glioblastoma Cells With Carboranyl-Indole Carboxamides

Recent developments with boron as a platform for novel drug design

(2016) Zbigniew J. Leśnikowski   Expert Opinion on Drug Discovery

Synthesis and evaluation of boron folates for Boron-Neutron-Capture-Therapy (BNCT)

(2015) Kathrin Kettenbach et al.   RADIOCHIMICA ACTA

Preparation and evaluation of carborane-derived inhibitors of prostate specific membrane antigen (PSMA)

(2014) Mohamed E. El-Zaria et al.   DALTON TRANSACTIONS

[18F]DPA-C5yne, a novel fluorine-18-labelled analogue of DPA-714: radiosynthesis and preliminary evaluation as a radiotracer for imaging neuroinflammation with PET

(2014) Vincent Médran-Navarrete et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

Synthesis of a carborane-containing cholesterol derivative and evaluation as a potential dual agent for MRI/BNCT applications

(2014) Diego Alberti et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Structure of the Mitochondrial Translocator Protein in Complex with a Diagnostic Ligand

(2014)  ukasz Jaremko et al.   SCIENCE

The translocator protein (TSPO): A novel target for cancer chemotherapy

(2013) Christopher J.D. Austin et al.   INTERNATIONAL JOURNAL OF BIOCHEMISTRY & CELL BIOLOGY

Synthesis and cellular uptake of boron-rich pyrazolopyrimidines: exploitation of the translocator protein for the efficient delivery of boron into human glioma cells

(2011) Ellen L. Crossley et al.   CHEMICAL COMMUNICATIONS

Carbaboranes as Pharmacophores: Properties, Synthesis, and Application Strategies

(2011) Matthias Scholz et al.   CHEMICAL REVIEWS

Boron in Drug Discovery: Carboranes as Unique Pharmacophores in Biologically Active Compounds

(2011) Fatiah Issa et al.   CHEMICAL REVIEWS

Oral cancer, cigarette smoke and mitochondrial 18kDa translocator protein (TSPO) — In vitro, in vivo, salivary analysis

(2010) Rafael Nagler et al.   BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR BASIS OF DISEASE

Carborane-Conjugated 2-Quinolinecarboxamide Ligands of the Translocator Protein for Boron Neutron Capture Therapy

(2010) Andrea Cappelli et al.   BIOCONJUGATE CHEMISTRY

Boronated phosphonium salts containing arylboronic acid, closo-carborane, or nido-carborane: synthesis, X-ray diffraction, in vitro cytotoxicity, and cellular uptake

(2010) Daniel E. Morrison et al.   JOURNAL OF BIOLOGICAL INORGANIC CHEMISTRY

Translocator Protein Blockade Reduces Prostate Tumor Growth

(2009) A. Fafalios et al.   CLINICAL CANCER RESEARCH

The Translocator Protein (18 kDa): Central Nervous System Disease and Drug Design

(2009) Alana M. Scarf et al.   JOURNAL OF MEDICINAL CHEMISTRY

Translocator protein 18 kDa (TSPO): Molecular sensor of brain injury and repair

(2008) Ming-Kai Chen et al.   PHARMACOLOGY & THERAPEUTICS