Heterocyclic electrophiles as new MurA inhibitors

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Irreversible inhibitors of the 3C protease of Coxsackie virus through templated assembly of protein-binding fragments

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Covalent protein modification: the current landscape of residue-specific electrophiles

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Inhibitors of the peptidoglycan biosynthesis enzymes MurA-F

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Chemical and Computational Methods for the Characterization of Covalent Reactive Groups for the Prospective Design of Irreversible Inhibitors

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A Fragment-Based Method to Discover Irreversible Covalent Inhibitors of Cysteine Proteases

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Electrophilic Fragment-Based Design of Reversible Covalent Kinase Inhibitors

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The nature ofStaphylococcus aureusMurA and MurZ and approaches for detection of peptidoglycan biosynthesis inhibitors

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