The Synthesis of Aromatic Heterocycles from Propargylic Compounds

Synthesis of Trisubstituted Isoxazoles by Palladium(II)-Catalyzed Cascade Cyclization–Alkenylation of 2-Alkyn-1-one O-Methyl Oximes

(2012) Zhigang She et al.   JOURNAL OF ORGANIC CHEMISTRY

Au(I)-Catalyzed Intramolecular Hydroamination of the Fluorinated N′-Aryl-N-Propargyl Amidines: Mild Conditions for the Synthesis of 2-Fluoroalkyl Imidazole Derivatives

(2012) Shan Li et al.   ORGANIC LETTERS

From 2000 to Mid-2010: A Fruitful Decade for the Synthesis of Pyrazoles

(2011) Santos Fustero et al.   CHEMICAL REVIEWS

Recent progress in synthesis and bioactivity studies of indolizines

(2011) Girija S. Singh et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Microwave-Assisted Cerium(III)-Promoted Cyclization of Propargyl Amides to Polysubstituted Oxazole Derivatives

(2011) Giuseppe Bartoli et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Substituted 1,4,5,6-Tetrahydrocyclopenta[b]pyrroles by Platinum-Catalyzed Cascade Cyclization/Ring Expansion of 2-Alkynyl-1-azaspiro[2.3]hexanes

(2011) Masahiro Yoshida et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Pyrazoles via Electrophilic Cyclization

(2011) Metin Zora et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Substituted Acetylenic Epoxides Followed by Indium-Catalyzed Rearrangement to 2,3,5-Trisubstituted Furans

(2011) Jun Yong Kang et al.   JOURNAL OF ORGANIC CHEMISTRY

A DFT study on the mechanism of gold(iii)-catalyzed synthesis of highly substituted furans via [3, 3]-sigmatropic rearrangements and/or [1, 2]-acyloxy migration based on propargyl ketones

(2011) Ran Fang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Recent advances in indole syntheses: New routes for a classic target

(2011) Rubén Vicente   ORGANIC & BIOMOLECULAR CHEMISTRY

Microwave-Assisted Domino Access to C2-Chain Functionalized Furans from Tertiary Propargyl Vinyl Ethers

(2011) David Tejedor et al.   ORGANIC LETTERS

Transition-Metal-Catalyzed Uninterrupted Four-Step Sequence to Access Trisubstituted Isoxazoles

(2011) Eric Gayon et al.   ORGANIC LETTERS

Palladium-Catalyzed Cyclization of Propargylic Compounds

(2010) Li-Na Guo et al.   ACCOUNTS OF CHEMICAL RESEARCH

Regioselective Functionalization of the Imidazole Ring via Transition Metal-Catalyzed CN and CC Bond Forming Reactions

(2010) Fabio Bellina et al.   ADVANCED SYNTHESIS & CATALYSIS

Gold-Catalyzed Cycloisomerization Reactions of 2-Tosylaminophenylprop-1-yn-3-ols as a Versatile Approach for Indole Synthesis

(2010) Prasath Kothandaraman et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Regioselective Rhodium(II)-Catalyzed Hydroaminations of Propargylguanidines

(2010) Morgan J. Gainer et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Marine Indole Alkaloids: Potential New Drug Leads for the Control of Depression and Anxiety

(2010) Anna J. Kochanowska-Karamyan et al.   CHEMICAL REVIEWS

Multicomponent reactions for the synthesis of pyrroles

(2010) Verónica Estévez et al.   CHEMICAL SOCIETY REVIEWS

Diverse Methyl Sulfone-Containing Benzo[b]thiophene Library via Iodocyclization and Palladium-Catalyzed Coupling

(2010) Chul-Hee Cho et al.   JOURNAL OF COMBINATORIAL CHEMISTRY

Synthesis of Polysubstituted Furans Based on a Stepwise Sonogashira Coupling of (Z)-3-Iodoalk-2-en-1-ols with Terminal Propargylic Alcohols and Subsequent Au(I)- or Pd(II)-Catalyzed Cyclization−Aromatization via Elimination of H2O

(2010) Xiaobing Zhang et al.   JOURNAL OF ORGANIC CHEMISTRY

Brønsted Acid Catalyzed Cyclization of Propargylic Alcohols with Thioamides. Facile Synthesis of Di- and Trisubstituted Thiazoles

(2010) Xiaoxiang Zhang et al.   JOURNAL OF ORGANIC CHEMISTRY

Iron-Catalyzed Domino Process for the Synthesis of α-Carbonyl Furan Derivatives via One-Pot Cyclization Reaction

(2010) Huanfeng Jiang et al.   JOURNAL OF ORGANIC CHEMISTRY

An Atom-Economic Synthesis of Nitrogen Heterocycles from Alkynes

(2010) Barry M. Trost et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Facile one-pot synthesis of three different substituted thiazoles from propargylic alcohols

(2010) Xun Gao et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

One-pot highly efficient synthesis of substituted pyrroles and N-bridgehead pyrroles by zinc-catalyzed multicomponent reaction

(2010) Xiao-tao Liu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Reagent-Controlled Oxidative Aromatization in Iodocyclization: Switchable Access to Dihydropyrazoles and Pyrazoles

(2010) Takashi Okitsu et al.   ORGANIC LETTERS

Two-Component Approach Toward a Fully Substituted N-Fused Pyrrole Ring

(2010) Dmitri Chernyak et al.   ORGANIC LETTERS

Silver-Catalyzed One-Pot Cyclization Reaction of Electron- Deficient Alkynes and 2-Yn-1-ols: An Efficient Domino Process to Polysubstituted Furans

(2009) Hua Cao et al.   ADVANCED SYNTHESIS & CATALYSIS

Addition-Hydroamination Reactions of Propargyl Cyanamides: Rapid Access to Highly Substituted 2-Aminoimidazoles

(2009) Robert L. Giles et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Niacin: a re-emerging pharmaceutical for the treatment of dyslipidaemia

(2009) Helen Vosper   BRITISH JOURNAL OF PHARMACOLOGY

Cyclization of Propargylic Amides: Mild Access to Oxazole Derivatives

(2009) Jan P. Weyrauch et al.   CHEMISTRY-A EUROPEAN JOURNAL

Recent Advances in the Synthesis of Indole and Quinoline Derivatives through Cascade Reactions

(2009) José Barluenga et al.   Chemistry-An Asian Journal

Catalyzed Propargylic Substitution

(2009) Remko J. Detz et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Rhodium(I)-Catalyzed Synthesis of Indoles: Amino-Claisen Rearrangement ofN-Propargylanilines

(2009) Akio Saito et al.   JOURNAL OF ORGANIC CHEMISTRY

Flexible Synthesis of Pyrimidines with Chiral Monofluorinated and Difluoromethyl Side Chains

(2009) Pierre Bannwarth et al.   JOURNAL OF ORGANIC CHEMISTRY

Brønsted Acid-Catalyzed Propargylation/Cycloisomerization Tandem Reaction: One-Pot Synthesis of Substituted Oxazoles from Propargylic Alcohols and Amides

(2009) Ying-ming Pan et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Isoquinoline Derivatives via Ag- Catalyzed Cyclization of 2-Alkynyl Benzyl Azides

(2009) Yan-Ning Niu et al.   JOURNAL OF ORGANIC CHEMISTRY

Gold-Catalyzed Cyclization of Alkynylaziridines as an Efficient Approach toward FunctionalizedN-Phth Pyrroles

(2009) Xiangwei Du et al.   JOURNAL OF ORGANIC CHEMISTRY

Muscarine, imidazole, oxazole and thiazole alkaloids

(2009) Zhong Jin   NATURAL PRODUCT REPORTS

The Meyer–Schuster rearrangement for the synthesis of α,β-unsaturated carbonyl compounds

(2009) Douglas A. Engel et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Sulfur-Assisted Five-Cascade Sequential Reactions for the Convenient and Efficient Synthesis of Allyl Thiophen-2-yl Acetates, Propionates, and Ketones

(2009) Hongwei Zhou et al.   ORGANIC LETTERS

α-Sulfanyl and α-Selanyl Propadienyl Cations: Regioselective Generations and Cycloadditions with Thioamides and Selemides Controlled by MeNO2−H2O System

(2009) Mitsuhiro Yoshimatsu et al.   ORGANIC LETTERS

Au(I)-Catalyzed Rearrangement Reaction of Propargylic Aziridine: Synthesis of Trisubstituted and Cycloalkene-Fused Pyrroles

(2009) Xiong Zhao et al.   ORGANIC LETTERS

Counterion Effects in a Gold-Catalyzed Synthesis of Pyrroles from Alkynyl Aziridines

(2009) Paul W. Davies et al.   ORGANIC LETTERS

Copper-Catalyzed Domino Rearrangement/Dehydrogenation Oxidation/Carbene Oxidation for One-Pot Regiospecific Synthesis of Highly Functionalized Polysubstituted Furans

(2009) Hua Cao et al.   ORGANIC LETTERS

Synthesis of Pyrroles by Gold(I)-Catalyzed Amino−Claisen Rearrangement ofN-Propargyl Enaminone Derivatives

(2009) Akio Saito et al.   ORGANIC LETTERS

An Efficient Domino Approach for the Synthesis of Multisubstituted Pyrroles via Gold/Silver-Catalyzed Amination/Cycloisomerization of (Z)-2-En-4-yn-1-ols

(2008) Yuhua Lu et al.   ADVANCED SYNTHESIS & CATALYSIS

Indium(III) Chloride-Catalyzed Propargylation/Amination/Cycloisomerization Tandem Reaction: One-Pot Synthesis of Highly Substituted Pyrroles from Propargylic Alcohols, 1,3-Dicarbonyl Compounds and Primary Amines

(2008) Xiao-tao Liu et al.   ADVANCED SYNTHESIS & CATALYSIS

Catalytic Synthesis of Indoles from Alkynes

(2008) Karolin Krüger (née Alex) et al.   ADVANCED SYNTHESIS & CATALYSIS

Ruthenium-Catalyzed Cycloaddition of Nitrile Oxides and Alkynes: Practical Synthesis of Isoxazoles

(2008) Scott Grecian et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

One-Pot Synthesis of Substituted Furans Using Cu(OTf)2-Catalyzed Propargylation/Cycloisomerization Tandem Reaction

(2008) Ying-ming Pan et al.   JOURNAL OF COMBINATORIAL CHEMISTRY

Silver(I)-Catalyzed Facile Synthesis of Pyrazoles From PropargylN-Sulfonylhydrazones

(2008) Young Tak Lee et al.   JOURNAL OF ORGANIC CHEMISTRY

Intramolecular Pd(II)-Catalyzed Cyclization of Propargylamides: Straightforward Synthesis of 5-Oxazolecarbaldehydes

(2008) Egle M. Beccalli et al.   JOURNAL OF ORGANIC CHEMISTRY

Iodine-Mediated Electrophilic Cyclization of 2-Alkynyl-1-methylene Azide Aromatics Leading to Highly Substituted Isoquinolines and Its Application to the Synthesis of Norchelerythrine

(2008) Dirk Fischer et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

N-Propargylic β-Enaminones: Common Intermediates for the Synthesis of Polysubstituted Pyrroles and Pyridines

(2008) Sandro Cacchi et al.   ORGANIC LETTERS

Ruthenium-Catalyzed Intramolecular Cyclization of 3-Butyne-1,2-diols into Furans

(2008) Yukito Yada et al.   ORGANOMETALLICS

Efficient Synthesis of Substituted 3-Iodofurans by Electrophilic Cyclization of Propargylic Oxirane Derivatives

(2007) Yong-Xin Xie et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY