Original access to 5-aryluracils from 5-iodo-2′-deoxyuridine via a microwave assisted Suzuki-Miyaura cross-coupling/deglycosylation sequence in pure water

Palladium-Catalyzed Direct Arylation of 5-Halouracils and 5-Halouracil Nucleosides with Arenes and Heteroarenes Promoted by TBAF

(2014) Yong Liang et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-catalyzed Suzuki reaction in aqueous solvents applied to unprotected nucleosides and nucleotides

(2014) Gwénaëlle Hervé et al.   RSC Advances

Improved microwave-assisted ligand-free Suzuki–Miyaura cross-coupling of 5-iodo-2′-deoxyuridine in pure water

(2013) Shawn Gallagher-Duval et al.   NEW JOURNAL OF CHEMISTRY

New, Efficient Approach for the Ligand-Free Suzuki–Miyaura Reaction of 5-Iodo-2′-deoxyuridine in Water

(2013) Christophe Len et al.   SYNTHESIS-STUTTGART

Synthesis of 6-aryluridines via Suzuki–Miyaura cross-coupling reaction at room temperature under aerobic ligand-free conditions in neat water

(2013) Gérald Enderlin et al.   TETRAHEDRON LETTERS

Highly Effective Synthesis of C-5-Substituted 2′-Deoxyuridine Using Suzuki-Miyaura Cross-Coupling in Water

(2012) Christophe Len et al.   SYNTHESIS-STUTTGART

Regioselective Direct C–H Arylations of Protected Uracils. Synthesis of 5- and 6-Aryluracil Bases

(2011) Miroslava Čerňová et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-catalyzed direct 5-arylation of 1,3-dimethyluracil with aryl bromides: an electrophilic metalation–deprotonation with electrophilic arylpalladium intermediate

(2011) Ko Hoon Kim et al.   TETRAHEDRON LETTERS

Switching the Regioselectivity of Direct C-H Arylation of 1,3-Dimethyluracil

(2009) Miroslava Čerňová et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Modeling the Dissociative Hydrolysis of the Natural DNA Nucleosides

(2009) Jennifer L. Przybylski et al.   JOURNAL OF PHYSICAL CHEMISTRY B

Use of Pd-catalyzed Suzuki–Miyaura coupling reaction in the rapid synthesis of 5-aryl-6-(phosphonomethoxy)uracils and evaluation of their inhibitory effect towards human thymidine phosphorylase

(2009) Karel Pomeisl et al.   TETRAHEDRON

Palladium-catalyzed intramolecular arylation of pyrimidines: a novel and expedient avenue to benzannulated pyridopyrimidines

(2009) K.C. Majumdar et al.   TETRAHEDRON

Zwitterionic uracil derivatives as potent GnRH receptor antagonists with improved pharmaceutical properties

(2008) Colin F. Regan et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Potent and orally bioavailable zwitterion GnRH antagonists with low CYP3A4 inhibitory activity

(2008) Chen Chen et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Intramolecular cyclization reaction — Palladium(0)-catalyzed cyclization is more effective than tin hydride mediated reaction

(2008) Krishna C Majumdar et al.   CANADIAN JOURNAL OF CHEMISTRY

Discovery of SodiumR-(+)-4-{2-[5-(2-Fluoro-3-methoxyphenyl)-3-(2-fluoro-6-[trifluoromethyl]benzyl)-4-methyl-2,6-dioxo-3,6-dihydro-2H-pyrimidin-1-yl]-1-phenylethylamino}butyrate (Elagolix), a Potent and Orally Available Nonpeptide Antagonist of the Human Gonadotropin-Releasing Hormone Receptor

(2008) Chen Chen et al.   JOURNAL OF MEDICINAL CHEMISTRY

Regio- and chemoselective magnesiation of protected uracils and thiouracils using TMPMgCl·LiCl and TMP2Mg·2LiCl

(2008) Marc Mosrin et al.   ORGANIC & BIOMOLECULAR CHEMISTRY