Highly regioselective C–H bond functionalization: palladium-catalyzed arylation of substituted imidazo[1,2-a]pyridine with aryl chlorides

Oxidative Biaryl Coupling of Thiophenes and Thiazoles with Arylboronic Acids through Palladium Catalysis: Otherwise Difficult C4-Selective CH Arylation Enabled by Boronic Acids

(2011) Sylvia Kirchberg et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Nickel-catalyzed sp2 C–H bonds arylation of N-aromatic heterocycles with Grignard reagents at room temperature

(2011) Gui-Rong Qu et al.   CHEMICAL COMMUNICATIONS

Palladium-catalyzed desulfitative C-arylation of a benzo[d]oxazole C–H bond with arene sulfonyl chlorides

(2011) Manli Zhang et al.   CHEMICAL COMMUNICATIONS

C-H Bond Functionalization of Arylpyrimidines Catalyzed by an in situ Generated Ruthenium(II) Carboxylate System and the Construction of Tris(heteroaryl)-Substituted Benzenes

(2011) Bogdan Štefane et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

C–H bond functionalisation with [RuH(codyl)2]BF4 catalyst precursor

(2011) Wenbo Li et al.   GREEN CHEMISTRY

Systematic Structure Modifications of Imidazo[1,2-a]pyrimidine to Reduce Metabolism Mediated by Aldehyde Oxidase (AO)

(2011) Angelica Linton et al.   JOURNAL OF MEDICINAL CHEMISTRY

Base-Mediated Intermolecular sp2C−H Bond Arylation via Benzyne Intermediates

(2011) Thanh Truong et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A General Method for Copper-Catalyzed Arene Cross-Dimerization

(2011) Hien-Quang Do et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Catalyzed Arylation of 1H-Perfluoroalkanes

(2011) Ilya Popov et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Silver-Mediated Palladium-Catalyzed Direct C−H Arylation of 3-Bromoisothiazole-4-carbonitrile

(2011) Heraklidia A. Ioannidou et al.   ORGANIC LETTERS

Ligand-Free Copper-Catalyzed Regioselective C-2 Arylation of Imidazo[2,1-b]thiazoles

(2011) Guoli Huang et al.   ORGANIC LETTERS

A Base Promoted Cyclization ofN-Propargylaminopyridines. Synthesis of Imidazo[1,2-a]pyridine Derivatives

(2011) Suren Husinec et al.   ORGANIC LETTERS

Direct C5-Arylation Reaction between Imidazoles and Aryl Chlorides Catalyzed by Palladium Complexes with Phosphines and N-Heterocyclic Carbenes

(2011) P. Vijaya Kumar et al.   ORGANOMETALLICS

Chelation-assisted palladium-catalyzed high regioselective heck diarylation reaction of 9-allyl-9H-purine: synthesis of 9-(3,3-diaryl-allyl)-9H-purines

(2011) Hai-Ming Guo et al.   RSC Advances

A General Catalyst for the β-Selective C-H Bond Arylation of Thiophenes with Iodoarenes

(2010) Kirika Ueda et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Nickel-Catalyzed Direct CH Arylation and Alkenylation of Heteroarenes with Organosilicon Reagents

(2010) Hitoshi Hachiya et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

General and Efficient Copper-Catalyzed Three-Component Coupling Reaction towards Imidazoheterocycles: One-Pot Synthesis of Alpidem and Zolpidem

(2010) Natalia Chernyak et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Transition Metal-Catalyzed Direct Arylation of Substrates with Activated sp3-Hybridized C−H Bonds and Some of Their Synthetic Equivalents with Aryl Halides or Pseudohalides

(2010) Fabio Bellina et al.   CHEMICAL REVIEWS

Palladium-Catalyzed C−H Functionalization of Heteroarenes with Aryl Bromides and Chlorides

(2010) Shunsuke Tamba et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed Indole, Pyrrole, and Furan Arylation by Aryl Chlorides

(2010) Enrico T. Nadres et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium- and Copper-Catalyzed Arylation of Carbon−Hydrogen Bonds

(2009) Olafs Daugulis et al.   ACCOUNTS OF CHEMICAL RESEARCH

Transition-Metal-Catalyzed Direct Arylation of (Hetero)Arenes by CH Bond Cleavage

(2009) Lutz Ackermann et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium(II)-Catalyzed CH Activation/CC Cross-Coupling Reactions: Versatility and Practicality

(2009) Xiao Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Diethyl carbonate as a solvent for ruthenium catalysed C–H bond functionalisation

(2009) Percia Arockiam et al.   GREEN CHEMISTRY

Copper-Mediated Direct Arylation of 1,3,4-Oxadiazoles and 1,2,4-Triazoles with Aryl Iodides

(2009) Tsuyoshi Kawano et al.   ORGANIC LETTERS

Nickel-Catalyzed Direct Arylation of Azoles with Aryl Bromides

(2009) Hitoshi Hachiya et al.   ORGANIC LETTERS

Direct Functionalization of Nitrogen Heterocycles via Rh-Catalyzed C−H Bond Activation

(2008) Jared C. Lewis et al.   ACCOUNTS OF CHEMICAL RESEARCH

Structural Requirements for Eszopiclone and Zolpidem Binding to the γ-Aminobutyric Acid Type-A (GABAA) Receptor Are Different

(2008) Susan M. Hanson et al.   JOURNAL OF MEDICINAL CHEMISTRY

Rh(I)-Catalyzed Arylation of Heterocycles via C−H Bond Activation:  Expanded Scope through Mechanistic Insight

(2008) Jared C. Lewis et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Direct Arylation of Arene C−H Bonds by Cooperative Action of NHCarbene−Ruthenium(II) Catalyst and Carbonate via Proton Abstraction Mechanism

(2008) Ismail Özdemir et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rh(I)-Catalyzed Direct Arylation of Pyridines and Quinolines

(2008) Ashley M. Berman et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed Direct Arylation of Nitro-Substituted Aromatics with Aryl Halides

(2008) Laurence Caron et al.   ORGANIC LETTERS

Assisted Ruthenium-Catalyzed C−H Bond Activation: Carboxylic Acids as Cocatalysts for Generally Applicable Direct Arylations in Apolar Solvents

(2008) Lutz Ackermann et al.   ORGANIC LETTERS