Organocatalytic synthesis of optically active heteroaromatic compounds

Optically Active Thiophenes via an Organocatalytic One-Pot Methodology

(2012) Lars Krogager Ransborg et al.   ORGANIC LETTERS

The Diarylprolinol Silyl Ether System: A General Organocatalyst

(2011) Kim L. Jensen et al.   ACCOUNTS OF CHEMICAL RESEARCH

One-Pot Reactions Accelerate the Synthesis of Active Pharmaceutical Ingredients

(2011) Carine Vaxelaire et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Taming the Friedel-Crafts Reaction: Organocatalytic Approach to Optically Active 2,3-Dihydrobenzofurans

(2011) Łukasz Albrecht et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Simple Recipe for Sophisticated Cocktails: Organocatalytic One-Pot Reactions-Concept, Nomenclature, and Future Perspectives

(2011) Łukasz Albrecht et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Organocatalytic Cyclization and Cycloaddition Reactions

(2011) Albert Moyano et al.   CHEMICAL REVIEWS

Organocatalytic Strategies for the Construction of Optically Active Imidazoles, Oxazoles, and Thiazoles

(2011) Łukasz Albrecht et al.   CHEMISTRY-A EUROPEAN JOURNAL

Catalytic Asymmetric Aziridination of α,β-Unsaturated Aldehydes

(2011) Luca Deiana et al.   CHEMISTRY-A EUROPEAN JOURNAL

Enantioselective α-Arylation of Aldehydes via the Productive Merger of Iodonium Salts and Organocatalysis

(2011) Anna E. Allen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Novel one-pot process for the synthesis of 1,3-thiazoles via organocatalysed epoxidation of nitro-olefins

(2011) Katharina M. Weiß et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Asymmetric organocatalytic [3 + 2]-annulation strategy for the synthesis of N-fused heteroaromatic compounds

(2011) Łukasz Albrecht et al.   Chemical Science

Strategies for the synthesis of 2,3-dihydrobenzofurans

(2011) Tom D. Sheppard   JOURNAL OF CHEMICAL RESEARCH

Asymmetric Synthesis with Silicon-Based Bulky Amino Organocatalysts

(2010) Li-Wen Xu et al.   ADVANCED SYNTHESIS & CATALYSIS

Enantioselective epoxidation of electron-deficient olefins: an organocatalytic approach

(2010) Katharina M. Weiß et al.   CHEMICAL RECORD

Immunosuppressive effects of 2-acetyl-4-tetrahydroxybutyl imidazole (THI) in the rat

(2010) S. J. P. GOBIN et al.   CLINICAL AND EXPERIMENTAL IMMUNOLOGY

Enantioselective Friedel-Crafts Alkylation of Thiophenes with Ethyl Glyoxylate: Easy Access to Chiral Secondary Alcohols

(2010) Zhong Huang et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Organocatalyzed Asymmetric Friedel-Crafts Reactions

(2010) Vincent Terrasson et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis, Chiral High Performance Liquid Chromatographic Resolution and Enantiospecific Activity of a Potent New Geranylgeranyl Transferase Inhibitor, 2-Hydroxy-3-imidazo[1,2-a]pyridin-3-yl-2-phosphonopropionic Acid

(2010) Charles E. McKenna et al.   JOURNAL OF MEDICINAL CHEMISTRY

Inhibition of Sphingosine 1-Phosphate Lyase for the Treatment of Rheumatoid Arthritis: Discovery of (E)-1-(4-((1R,2S,3R)-1,2,3,4-Tetrahydroxybutyl)-1H-imidazol-2-yl)ethanone Oxime (LX2931) and (1R,2S,3R)-1-(2-(Isoxazol-3-yl)-1H-imidazol-4-yl)butane-1,2,3,4-tetraol (LX2932)

(2010) Jeffrey T. Bagdanoff et al.   JOURNAL OF MEDICINAL CHEMISTRY

An Organocatalytic Approach to 2-Hydroxyalkyl- and 2-Aminoalkyl Furanes

(2010) Łukasz Albrecht et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Asymmetric Formaltrans-Dihydroxylation andtrans-Aminohydroxylation of α,β-Unsaturated Aldehydes via an Organocatalytic Reaction Cascade

(2010) Łukasz Albrecht et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

The Gewald multicomponent reaction

(2010) Yijun Huang et al.   MOLECULAR DIVERSITY

Organocatalytic cascade reactions as a new tool in total synthesis

(2010) Christoph Grondal et al.   Nature Chemistry

New development of synthesis and reactivity of seleno- and tellurophenes

(2010) Cristiano R. B. Rhoden et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Direct Preparation of Heteroaromatic Compounds from Alkenes

(2010) Timothy Donohoe et al.   SYNLETT

Synthetic studies towards oxygenated and unsaturated furanocembranoid macrocycles. Precursors to plumarellide, rameswaralide and mandapamates

(2010) Gerald Pattenden et al.   TETRAHEDRON LETTERS

Exploration of a proposed biomimetic synthetic route to plumarellide. Development of a facile transannular Diels–Alder reaction from a macrocyclic enedione leading to a new 5,6,7-tricyclic ring system

(2010) Yi Li et al.   TETRAHEDRON LETTERS

Achieving Molecular Complexity by Organocatalytic One-Pot Strategies-A Fast Entry for Synthesis of Sphingoids, Amino Sugars, and Polyhydroxylated α-Amino Acids

(2009) Hao Jiang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Brønsted Acid Catalyzed Enantioselective Three-Component Reaction Involving the α Addition of Isocyanides to Imines

(2009) Tao Yue et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Anodic Oxidation and Organocatalysis: Direct Regio- and Stereoselective Access to meta-Substituted Anilines by α-Arylation of Aldehydes

(2009) Kim L. Jensen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chiral Brønsted acid catalyzed Friedel–Crafts alkylation reactions

(2009) Shu-Li You et al.   CHEMICAL SOCIETY REVIEWS

Synthesis and cytotoxic activity of 2-methylimidazo[1,2-a]pyridine- and quinoline-substituted 2-aminopyrimidine derivatives

(2009) Miguel Angel Vilchis-Reyes et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Duloxetine in the treatment of generalized anxiety disorder

(2009) Susan G Kornstein et al.   Expert Review of Neurotherapeutics

Inhibition of Sphingosine-1-Phosphate Lyase for the Treatment of Autoimmune Disorders

(2009) Jeffrey T. Bagdanoff et al.   JOURNAL OF MEDICINAL CHEMISTRY

Practical Catalytic Asymmetric Synthesis of Diaryl-, Aryl Heteroaryl-, and Diheteroarylmethanols

(2009) Luca Salvi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective Intramolecular Friedel−Crafts-Type α-Arylation of Aldehydes

(2009) K. C. Nicolaou et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective α-Arylation of Aldehydes via Organo-SOMO Catalysis. An Ortho-Selective Arylation Reaction Based on an Open-Shell Pathway

(2009) Jay C. Conrad et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of dihydrodehydrodiconiferyl alcohol: the revised structure of lawsonicin

(2009) Junxiu Meng et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Highly Enantioselective Friedel−Crafts Reaction of Thiophenes with Glyoxylates: Formal Synthesis of Duloxetine

(2009) Jakub Majer et al.   ORGANIC LETTERS

Recent Progress in the Synthesis of 2,3-Dihydrobenzofurans

(2009) Ferruccio Bertolini et al.   ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL

Kilogram-Scale Synthesis of the CXCR4 Antagonist GSK812397

(2009) Sharon Boggs et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Asymmetric Hydrogenation of Heteroaromatic Ketones and Cyclic and Acyclic Enones Mediated by Cu(I)-Chiral Diphosphine Catalysts

(2009) Hideo Shimizu et al.   SYNLETT

An intramolecular [4+3]-cycloaddition approach to rameswaralide inspired by biosynthesis speculation

(2009) Gerald Pattenden et al.   TETRAHEDRON LETTERS

Enantioselective aziridination reaction of α,β-unsaturated aldehydes using an organocatalyst and tert-butyl N-arenesulfonyloxycarbamates

(2009) Hiromi Arai et al.   TETRAHEDRON LETTERS

Asymmetric Aminocatalysis-Gold Rush in Organic Chemistry

(2008) Paolo Melchiorre et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Influence of 6- or 8-substitution on the antiviral activity of 3-arylalkylthiomethylimidazo[1,2-a]pyridine against human cytomegalovirus (CMV) and varicella-zoster virus (VZV): Part II

(2008) Jean-Baptiste Véron et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Catalytic Asymmetric Friedel−Crafts Alkylation ReactionsCopper Showed the Way

(2008) Thomas B. Poulsen et al.   CHEMICAL REVIEWS

Furanocembranoids from the Soft CoralsSinularia asterolobataandLitophyton arboreum

(2008) Daniela Grote et al.   CHEMISTRY & BIODIVERSITY

Emerging approaches for the syntheses of bicyclic imidazo[1,2-x]-heterocycles

(2008) Christopher Hulme et al.   MOLECULAR DIVERSITY

Lamellarins and Related Pyrrole-Derived Alkaloids from Marine Organisms

(2007) Hui Fan et al.   CHEMICAL REVIEWS