The Ugi four-component reaction enables expedient synthesis and comparison of photoaffinity probes

1,3,5-Trisubstituted benzenes as fluorescent photoaffinity probes for human carbonic anhydrase II capture

(2013) Partha Sarathi Addy et al.   CHEMICAL COMMUNICATIONS

5-Carboxy-8-hydroxyquinoline is a broad spectrum 2-oxoglutarate oxygenase inhibitor which causes iron translocation

(2013) Richard J. Hopkinson et al.   Chemical Science

Tandem photoaffinity labeling–bioorthogonal conjugation in medicinal chemistry

(2012) David J. Lapinsky   BIOORGANIC & MEDICINAL CHEMISTRY

Ugi reaction-assisted rapid assembly of affinity-based probes against potential protein tyrosine phosphatases

(2012) Jingyan Ge et al.   CHEMICAL COMMUNICATIONS

Reporter Ligand NMR Screening Method for 2-Oxoglutarate Oxygenase Inhibitors

(2012) Ivanhoe K. H. Leung et al.   JOURNAL OF MEDICINAL CHEMISTRY

Affinity-Based Probes Based on Type II Kinase Inhibitors

(2012) Pratistha Ranjitkar et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Diazirine based photoaffinity labeling

(2011) Luba Dubinsky et al.   BIOORGANIC & MEDICINAL CHEMISTRY

A Photoreactive Small-Molecule Probe for 2-Oxoglutarate Oxygenases

(2011) Dante Rotili et al.   CHEMISTRY & BIOLOGY

Probing small molecule–protein interactions: A new perspective for functional proteomics

(2011) Thomas Lenz et al.   Journal of Proteomics

Fast and efficient MCR-based synthesis of clickable rhodamine tags for protein profiling

(2011) Sebastian Brauch et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Readily Accessible Bicyclononynes for Bioorthogonal Labeling and Three-Dimensional Imaging of Living Cells

(2010) Jan Dommerholt et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of S-Adenosyl-L-homocysteine Capture Compounds for Selective Photoinduced Isolation of Methyltransferases

(2010) Christian Dalhoff et al.   CHEMBIOCHEM

Photoactivable peptides for identifying enzyme–substrate and protein–protein interactions

(2010) Dante Rotili et al.   CHEMICAL COMMUNICATIONS

Quantitative High-Throughput Screening Identifies 8-Hydroxyquinolines as Cell-Active Histone Demethylase Inhibitors

(2010) Oliver N. F. King et al.   PLoS One

Functional Profiling, Identification, and Inhibition of Plasmepsins in Intraerythrocytic Malaria Parasites

(2009) Kai Liu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Monoacylglycerol Lipase Regulates a Fatty Acid Network that Promotes Cancer Pathogenesis

(2009) Daniel K. Nomura et al.   CELL

Application of a Proteolysis/Mass Spectrometry Method for Investigating the Effects of Inhibitors on Hydroxylase Structure

(2009) Christopher J. Stubbs et al.   JOURNAL OF MEDICINAL CHEMISTRY

Structural Basis for Binding of Hypoxia-Inducible Factor to the Oxygen-Sensing Prolyl Hydroxylases

(2009) Rasheduzzaman Chowdhury et al.   STRUCTURE