A review of the influence of functional group modifications to the core scaffold of synthetic cathinones on drug pharmacokinetics

MDPV in forensic routine cases: Psychotic and aggressive behavior in relation to plasma concentrations

(2018) Marco Diestelmann et al.   FORENSIC SCIENCE INTERNATIONAL

Mephedrone (4-Methylmethcathinone): Acute Behavioral Effects, Hyperthermic, and Pharmacokinetic Profile in Rats

(2018) Klára Šíchová et al.   Frontiers in Psychiatry

The pharmacokinetic profile of synthetic cathinones in a pregnancy model

(2017) Lauren G. Strange et al.   NEUROTOXICOLOGY AND TERATOLOGY

Impact of common clandestine structural modifications on synthetic cathinone “bath salt” pharmacokinetics

(2017) Gregory G. Grecco et al.   TOXICOLOGY AND APPLIED PHARMACOLOGY

Pharmacokinetic, Ambulatory, and Hyperthermic Effects of 3,4-Methylenedioxy-N-Methylcathinone (Methylone) in Rats

(2017) Kristýna Štefková et al.   Frontiers in Psychiatry

Phase I metabolites of mephedrone display biological activity as substrates at monoamine transporters

(2016) F P Mayer et al.   BRITISH JOURNAL OF PHARMACOLOGY

Human Pharmacology of Mephedrone in Comparison with MDMA

(2016) Esther Papaseit et al.   NEUROPSYCHOPHARMACOLOGY

Pharmacokinetic Profiles and Pharmacodynamic Effects for Methylone and Its Metabolites in Rats

(2016) Joshua S Elmore et al.   NEUROPSYCHOPHARMACOLOGY

Increasing use of ‘party drugs’ in people living with HIV on antiretrovirals

(2015) Margherita Bracchi et al.   AIDS

Synthetic Cathinones: A New Public Health Problem

(2015) Laurent Karila et al.   Current Neuropharmacology

3-Methyl-methcathinone: Pharmacokinetic profile evaluation in pigs in relation to pharmacodynamics

(2015) Jakob A Shimshoni et al.   JOURNAL OF PSYCHOPHARMACOLOGY

Concentrations of MDPV in rat striatum correlate with the psychostimulant effect

(2015) Judith Novellas et al.   JOURNAL OF PSYCHOPHARMACOLOGY

Linear pharmacokinetics of 3,4-methylenedioxypyrovalerone (MDPV) and its metabolites in the rat: relationship to pharmacodynamic effects

(2014) Sebastien Anizan et al.   ADDICTION BIOLOGY

In vitro cytochrome P450 inhibition potential of methylenedioxy-derived designer drugs studied with a two-cocktail approach

(2014) Julia Dinger et al.   ARCHIVES OF TOXICOLOGY

The preclinical pharmacology of mephedrone; not just MDMA by another name

(2014) A R Green et al.   BRITISH JOURNAL OF PHARMACOLOGY

Synthetic Cathinones (“Bath Salts”)

(2014) Matthew L. Banks et al.   JOURNAL OF EMERGENCY MEDICINE

Sudden Cardiac Death Associated With Methylone Use

(2013) Peter N. Carbone et al.   AMERICAN JOURNAL OF FORENSIC MEDICINE AND PATHOLOGY

Monoamine transporter and receptor interaction profiles of a new series of designer cathinones

(2013) L.D. Simmler et al.   NEUROPHARMACOLOGY

An integrated pharmacokinetic and pharmacodynamic study of a new drug of abuse, methylone, a synthetic cathinone sold as “bath salts”

(2013) Raúl López-Arnau et al.   PROGRESS IN NEURO-PSYCHOPHARMACOLOGY & BIOLOGICAL PSYCHIATRY

Mephedrone pharmacokinetics after intravenous and oral administration in rats: relation to pharmacodynamics

(2013) J. Martínez-Clemente et al.   PSYCHOPHARMACOLOGY

Pharmacogenetics of cytochrome P450 2B6 (CYP2B6): advances on polymorphisms, mechanisms, and clinical relevance

(2013) Ulrich M. Zanger et al.   Frontiers in Genetics

Generation of metabolites by an automated online metabolism method using human liver microsomes with subsequent identification by LC-MS(n), and metabolism of 11 cathinones

(2012) Daniel M. Mueller et al.   ANALYTICAL AND BIOANALYTICAL CHEMISTRY

Pharmacological characterization of designer cathinonesin vitro

(2012) LD Simmler et al.   BRITISH JOURNAL OF PHARMACOLOGY

2011 Annual Report of the American Association of Poison Control Centers’ National Poison Data System (NPDS): 29th Annual Report

(2012) Alvin C. Bronstein et al.   CLINICAL TOXICOLOGY

In vitrometabolism studies on mephedrone and analysis of forensic cases

(2012) Anders Just Pedersen et al.   Drug Testing and Analysis

Three Fatal Intoxications Due to Methylone

(2012) J. M. Pearson et al.   JOURNAL OF ANALYTICAL TOXICOLOGY

The Designer Methcathinone Analogs, Mephedrone and Methylone, are Substrates for Monoamine Transporters in Brain Tissue

(2011) Michael H Baumann et al.   NEUROPSYCHOPHARMACOLOGY

Beta-keto amphetamines: studies on the metabolism of the designer drug mephedrone and toxicological detection of mephedrone, butylone, and methylone in urine using gas chromatography–mass spectrometry

(2010) Markus R. Meyer et al.   ANALYTICAL AND BIOANALYTICAL CHEMISTRY

Studies on the metabolism of the α-pyrrolidinophenone designer drug methylenedioxy-pyrovalerone (MDPV) in rat and human urine and human liver microsomes using GC-MS and LC-high-resolution MS and its detectability in urine by GC-MS

(2010) Markus R. Meyer et al.   JOURNAL OF MASS SPECTROMETRY

Toxicological determination and in vitro metabolism of the designer drug methylenedioxypyrovalerone (MPDV) by gas chromatography/mass spectrometry and liquid chromatography/quadrupole time-of-flight mass spectrometry

(2010) Sabina Strano-Rossi et al.   RAPID COMMUNICATIONS IN MASS SPECTROMETRY

Determination of the metabolites of the new designer drugs bk-MBDB and bk-MDEA in human urine

(2009) Kei Zaitsu et al.   FORENSIC SCIENCE INTERNATIONAL

Population Pharmacokinetics of 3,4-Methylenedioxymethamphetamine and Main Metabolites in Rats

(2009) Déborah Hirt et al.   TOXICOLOGICAL SCIENCES

Sprague–Dawley rats display sex-linked differences in the pharmacokinetics of 3,4-methylenedioxymethamphetamine (MDMA) and its metabolite 3,4-methylenedioxyamphetamine (MDA)

(2009) Julien Fonsart et al.   TOXICOLOGY AND APPLIED PHARMACOLOGY

Mechanism-Based Inactivation of Human Cytochromes P450s: Experimental Characterization, Reactive Intermediates, and Clinical Implications

(2007) Paul F. Hollenberg et al.   CHEMICAL RESEARCH IN TOXICOLOGY