Recombinant Human Melatonin Receptor MT1 Isolated in Mixed Detergents Shows Pharmacology Similar to That in Mammalian Cell Membranes

Large scale expression and purification of the mouse 5-HT3 receptor

(2013) Ghérici Hassaine et al.   BIOCHIMICA ET BIOPHYSICA ACTA-BIOMEMBRANES

Melatonin MT1and MT2receptors display different molecular pharmacologies only in the G-protein coupled state

(2013) Céline Legros et al.   BRITISH JOURNAL OF PHARMACOLOGY

New perspectives in melatonin uses

(2012) A. Carpentieri et al.   PHARMACOLOGICAL RESEARCH

Stabilization of Functional Recombinant Cannabinoid Receptor CB2 in Detergent Micelles and Lipid Bilayers

(2012) Krishna Vukoti et al.   PLoS One

Distinct roles of metabotropic glutamate receptor dimerization in agonist activation and G-protein coupling

(2012) D. El Moustaine et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

The Morphology and Composition of Cholesterol-Rich Micellar Nanostructures Determine Transmembrane Protein (GPCR) Activity

(2011) Michelle A. O'Malley et al.   BIOPHYSICAL JOURNAL

Nanobody stabilization of G protein-coupled receptor conformational states

(2011) Jan Steyaert et al.   CURRENT OPINION IN STRUCTURAL BIOLOGY

Uncovering the intimate relationship between lipids, cholesterol and GPCR activation

(2011) Joanne Oates et al.   CURRENT OPINION IN STRUCTURAL BIOLOGY

Molecular pharmacology of the mouse melatonin receptors MT1 and MT2

(2011) Séverine Devavry et al.   EUROPEAN JOURNAL OF PHARMACOLOGY

High Constitutive Activity Is an Intrinsic Feature of Ghrelin Receptor Protein

(2011) Marjorie Damian et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Description of the constitutive activity of cloned human melatonin receptors hMT1 and hMT2 and discovery of inverse agonists

(2011) Séverine Devavry et al.   JOURNAL OF PINEAL RESEARCH

GPCR stabilization using the bicelle-like architecture of mixed sterol-detergent micelles

(2011) Aaron A. Thompson et al.   METHODS

Structure of the human histamine H1 receptor complex with doxepin

(2011) Tatsuro Shimamura et al.   NATURE

Production of a Bioengineered G-Protein Coupled Receptor of Human Formyl Peptide Receptor 3

(2011) Xiaoqiang Wang et al.   PLoS One

Evaluation of subjective efficacy and safety of ramelteon in Japanese subjects with chronic insomnia

(2011) Makoto Uchiyama et al.   SLEEP MEDICINE

Erratum: Agomelatine, the first melatonergic antidepressant: discovery, characterization and development

(2010) Christian de Bodinat et al.   NATURE REVIEWS DRUG DISCOVERY

Study of Bioengineered Zebra Fish Olfactory Receptor 131-2: Receptor Purification and Secondary Structure Analysis

(2010) Kwong-Joo Leck et al.   PLoS One

High-throughput screening assay for new ligands at human melatonin receptors

(2009) Jian-hua Yan et al.   ACTA PHARMACOLOGICA SINICA

The end of a myth: cloning and characterization of the ovine melatonin MT2 receptor

(2009) F Cogé et al.   BRITISH JOURNAL OF PHARMACOLOGY

Solubilization and characterization of the anthrax toxin pore in detergent micelles

(2009) Gregory Vernier et al.   PROTEIN SCIENCE

Molecular cloning and pharmacological characterization of rat melatonin MT1 and MT2 receptors

(2008) Valérie Audinot et al.   BIOCHEMICAL PHARMACOLOGY

Melatonin receptors, heterodimerization, signal transduction and binding sites: what's new?

(2008) R Jockers et al.   BRITISH JOURNAL OF PHARMACOLOGY

Over-Expression, Solubilization, and Purification of G Protein-Coupled Receptors for Structural Biology

(2008) Mark Chiu et al.   COMBINATORIAL CHEMISTRY & HIGH THROUGHPUT SCREENING

Structural insights into G-protein-coupled receptor activation

(2008) William I Weis et al.   CURRENT OPINION IN STRUCTURAL BIOLOGY

Determination of the molecular mass and dimensions of membrane proteins by size exclusion chromatography

(2008) Edmund R.S. Kunji et al.   METHODS

A Specific Cholesterol Binding Site Is Established by the 2.8 Å Structure of the Human β2-Adrenergic Receptor

(2008) Michael A. Hanson et al.   STRUCTURE