High Constitutive Activity Is an Intrinsic Feature of Ghrelin Receptor Protein

Amphipols From A to Z*

(2011) J.-L. Popot et al.   Annual Review of Biophysics

Structural insights into agonist-induced activation of G-protein-coupled receptors

(2011) Xavier Deupi et al.   CURRENT OPINION IN STRUCTURAL BIOLOGY

G Protein Activation by Serotonin Type 4 Receptor Dimers

(2011) Lucie P. Pellissier et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

G protein-coupled receptors: mutations and endocrine diseases

(2011) Gilbert Vassart et al.   Nature Reviews Endocrinology

New advances in production and functional folding of G-protein-coupled receptors

(2011) Jean-Louis Banères et al.   TRENDS IN BIOTECHNOLOGY

Homogeneous time-resolved fluorescence-based assay to screen for ligands targeting the growth hormone secretagogue receptor type 1a

(2010) Jean-Philippe Leyris et al.   ANALYTICAL BIOCHEMISTRY

Monomeric Rhodopsin Is Sufficient for Normal Rhodopsin Kinase (GRK1) Phosphorylation and Arrestin-1 Binding

(2010) Timothy H. Bayburt et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Monomeric Rhodopsin Is the Minimal Functional Unit Required for Arrestin Binding

(2010) Hisao Tsukamoto et al.   JOURNAL OF MOLECULAR BIOLOGY

Energy Landscapes as a Tool to Integrate GPCR Structure, Dynamics, and Function

(2010) Xavier Deupi et al.   PHYSIOLOGY

Amphipol-Assisted in Vitro Folding of G Protein-Coupled Receptors

(2009) Tassadite Dahmane et al.   BIOCHEMISTRY

G protein-coupled receptor hetero-dimerization: contribution to pharmacology and function

(2009) Graeme Milligan   BRITISH JOURNAL OF PHARMACOLOGY

In VivoCharacterization of High Basal Signaling from the Ghrelin Receptor

(2009) Pia Steen Petersen et al.   ENDOCRINOLOGY

Membrane protein assembly into Nanodiscs

(2009) Timothy H. Bayburt et al.   FEBS LETTERS

Leukotriene BLT2 Receptor Monomers Activate the Gi2GTP-binding Protein More Efficiently than Dimers

(2009) Laure Arcemisbéhère et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

A Conserved Aromatic Lock for the Tryptophan Rotameric Switch in TM-VI of Seven-transmembrane Receptors

(2009) Birgitte Holst et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Purification and Functional Reconstitution of Monomeric μ-Opioid Receptors

(2009) Adam J. Kuszak et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Activation of the Ghrelin Receptor is Described by a Privileged Collective Motion: A Model for Constitutive and Agonist-induced Activation of a Sub-class A G-Protein Coupled Receptor (GPCR)

(2009) Nicolas Floquet et al.   JOURNAL OF MOLECULAR BIOLOGY

Growth Hormone Secretagogues and Growth Hormone Releasing Peptides Act As Orthosteric Super-Agonists but Not Allosteric Regulators for Activation of the G Protein G o1 by the Ghrelin Receptor

(2009) K. A. Bennett et al.   MOLECULAR PHARMACOLOGY

The effect of ligand efficacy on the formation and stability of a GPCR-G protein complex

(2009) X. J. Yao et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

The apparent cooperativity of some GPCRs does not necessarily imply dimerization

(2009) Marc Chabre et al.   TRENDS IN PHARMACOLOGICAL SCIENCES

New Trisubstituted 1,2,4-Triazole Derivatives as Potent Ghrelin Receptor Antagonists. 3. Synthesis and Pharmacological in Vitro and in Vivo Evaluations

(2008) Aline Moulin et al.   JOURNAL OF MEDICINAL CHEMISTRY

Rapid Incorporation of Functional Rhodopsin into Nanoscale Apolipoprotein Bound Bilayer (NABB) Particles

(2008) Sourabh Banerjee et al.   JOURNAL OF MOLECULAR BIOLOGY

The constitutive activity of the ghrelin receptor attenuates apoptosis via a protein kinase C-dependent pathway

(2008) Pui Ngan Lau et al.   MOLECULAR AND CELLULAR ENDOCRINOLOGY