TsOH·H2O-mediated N-amidation of quinoline N-oxides: facile and regioselective synthesis of N-(quinolin-2-yl)amides
Published 2018 View Full Article
- Home
- Publications
- Publication Search
- Publication Details
Title
TsOH·H2O-mediated N-amidation of quinoline N-oxides: facile and regioselective synthesis of N-(quinolin-2-yl)amides
Authors
Keywords
-
Journal
ORGANIC & BIOMOLECULAR CHEMISTRY
Volume 16, Issue 34, Pages 6202-6205
Publisher
Royal Society of Chemistry (RSC)
Online
2018-08-13
DOI
10.1039/c8ob00862k
References
Ask authors/readers for more resources
Related references
Note: Only part of the references are listed.- Selectfluor-mediated regioselective nucleophilic functionalization of N-heterocycles under metal- and base-free conditions
- (2018) Long-Yong Xie et al. GREEN CHEMISTRY
- Quinoline hybrids and their antiplasmodial and antimalarial activities
- (2017) Yuan-Qiang Hu et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- A base-free, ultrasound accelerated one-pot synthesis of 2-sulfonylquinolines in water
- (2017) Long-Yong Xie et al. GREEN CHEMISTRY
- Discovery and Optimization of Isoquinoline Ethyl Ureas as Antibacterial Agents
- (2017) Philippe Panchaud et al. JOURNAL OF MEDICINAL CHEMISTRY
- Hydrophilic, Potent, and Selective 7-Substituted 2-Aminoquinolines as Improved Human Neuronal Nitric Oxide Synthase Inhibitors
- (2017) Anthony V. Pensa et al. JOURNAL OF MEDICINAL CHEMISTRY
- Lewis Acid Catalyzed Dehydrogenative Coupling of Tertiary Propargylic Alcohols with Quinoline N-Oxides
- (2017) Ya-Ping Han et al. JOURNAL OF ORGANIC CHEMISTRY
- Local epigenetic reprogramming induced by G-quadruplex ligands
- (2017) Guillaume Guilbaud et al. Nature Chemistry
- Nitrilium ions – synthesis and applications
- (2017) Tom van Dijk et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Strategic Approach to 8-Azacoumarins
- (2017) Dong Wang et al. ORGANIC LETTERS
- Iodine-Catalyzed Direct C–H Alkenylation of Azaheterocycle N-Oxides with Alkenes
- (2017) Zhenhao Zhang et al. ORGANIC LETTERS
- Fast, Base-Free and Aqueous Synthesis of Quinolin-2(1H)-ones under Ambient Conditions
- (2017) Long-Yong Xie et al. ACS Sustainable Chemistry & Engineering
- A direct metal-free C2–H functionalization of quinoline N-oxides: a highly selective amination and alkylation strategy towards 2-substituted quinolines
- (2017) Wen-Zhu Bi et al. Organic Chemistry Frontiers
- Transition-Metal-Free Regioselective Alkylation of Pyridine N -Oxides Using 1,1-Diborylalkanes as Alkylating Reagents
- (2016) Woohyun Jo et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Synthesis of 1H-pyrrolo[3,2-h]quinoline-8-amine derivatives that target CTG trinucleotide repeats
- (2016) Jun Matsumoto et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Nonclassical Routes for Amide Bond Formation
- (2016) Renata Marcia de Figueiredo et al. CHEMICAL REVIEWS
- In Situ Generated HypoIodite Activator for the C2 Sulfonylation of Heteroaromatic N-oxides
- (2016) Yuan Su et al. JOURNAL OF ORGANIC CHEMISTRY
- Recent Developments in Amide Synthesis Using Nonactivated Starting Materials
- (2016) Andrea Ojeda-Porras et al. JOURNAL OF ORGANIC CHEMISTRY
- Catalyst and solvent-free alkylation of quinoline N-oxides with olefins: A direct access to quinoline-substituted α-hydroxy carboxylic derivatives
- (2016) Rakesh Kumar et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- C2-Alkenylation of N-heteroaromatic compounds via Brønsted acid catalysis
- (2016) Giacomo E. M. Crisenza et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Cu-Catalyzed Deoxygenative C2-Sulfonylation Reaction of Quinoline N-Oxides with Sodium Sulfinate
- (2016) Bingnan Du et al. ORGANIC LETTERS
- Acid-Free Silver-Catalyzed Cross-Dehydrogenative Carbamoylation of Pyridines with Formamides
- (2016) Wei Han et al. SYNLETT
- A review on anticancer potential of bioactive heterocycle quinoline
- (2015) Obaid Afzal et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Phenyl Ether- and Aniline-Containing 2-Aminoquinolines as Potent and Selective Inhibitors of Neuronal Nitric Oxide Synthase
- (2015) Maris A. Cinelli et al. JOURNAL OF MEDICINAL CHEMISTRY
- Oxidative cross-coupling of pyridine N-oxides and ethers between C(sp2)–H/C(sp3)–H bonds under transition-metal-free conditions
- (2015) Wei Sun et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Metal-free methylation of a pyridine N-oxide C–H bond by using peroxides
- (2015) Gang Li et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Copper(ii)-catalyzed electrophilic amination of quinoline N-oxides with O-benzoyl hydroxylamines
- (2015) Gang Li et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Gold-catalyzed α-furanylations of quinoline N-oxides with alkenyldiazo carbonyl species
- (2015) Vinayak Vishnu Pagar et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Synthesis of Benzofuro[3,2-b]pyridines via Palladium-Catalyzed Dual C–H Activation of 3-Phenoxypyridine 1-Oxides
- (2015) Wei Sun et al. ORGANIC LETTERS
- Base-Promoted Cross-Dehydrogenative Coupling of Quinoline N-Oxides with 1,3-Azoles
- (2015) Xiaopei Chen et al. ORGANIC LETTERS
- Regioselective Metal-Free Cross-Coupling of Quinoline N-Oxides with Boronic Acids
- (2015) Luis Bering et al. ORGANIC LETTERS
- The development of carbene-stabilized N–O radical coupling strategy in metal-free regioselective C–H azidation of quinoline N-oxides
- (2015) Pan Li et al. Organic Chemistry Frontiers
- Copper-catalyzed direct C–H arylation of pyridine N-oxides with arylboronic esters: one-pot synthesis of 2-arylpyridines
- (2014) Yan Shen et al. CHEMICAL COMMUNICATIONS
- Practical preparation of challenging amides from non-nucleophilic amines and esters under flow conditions
- (2014) Johannes L. Vrijdag et al. CHEMICAL COMMUNICATIONS
- Direct regioselective phosphonation of heteroaryl N-oxides with H-phosphonates under metal and external oxidant free conditions
- (2014) Hui Wang et al. CHEMICAL COMMUNICATIONS
- Conversion of Pyridine N-Oxides to Tetrazolopyridines
- (2014) Shanshan Liu et al. JOURNAL OF ORGANIC CHEMISTRY
- 2-Aminopyridines via Reaction of Pyridine N-Oxides and Activated Isocyanides
- (2014) Mitchell Vamos et al. JOURNAL OF ORGANIC CHEMISTRY
- Direct, Catalytic, and Regioselective Synthesis of 2-Alkyl-, Aryl-, and Alkenyl-Substituted N-Heterocycles from N-Oxides
- (2014) Oleg V. Larionov et al. ORGANIC LETTERS
- Light-mediated in cell downregulation of G-quadruplex-containing genes using a photo-caged ligand
- (2013) Pierre Murat et al. CHEMICAL COMMUNICATIONS
- Copper-catalysed amidation of 2-chloro-pyridines
- (2013) Lionel Nicolas et al. RSC Advances
- The Medicinal Chemist’s Toolbox: An Analysis of Reactions Used in the Pursuit of Drug Candidates
- (2011) Stephen D. Roughley et al. JOURNAL OF MEDICINAL CHEMISTRY
- Direct DehydrativeN-Pyridinylation of Amides
- (2009) Jonathan William Medley et al. JOURNAL OF ORGANIC CHEMISTRY
- Palladium-Catalyzed Alkenylation of Quinoline-N-oxides via C−H Activation under External-Oxidant-Free Conditions
- (2009) Junliang Wu et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- A Novel Small Molecule That Alters Shelterin Integrity and Triggers a DNA-Damage Response at Telomeres
- (2008) Raphaël Rodriguez et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
Find Funding. Review Successful Grants.
Explore over 25,000 new funding opportunities and over 6,000,000 successful grants.
ExploreDiscover Peeref hubs
Discuss science. Find collaborators. Network.
Join a conversation