Metal free sulfenylation and bis-sulfenylation of indoles: persulfate mediated synthesis

Iodine-Catalyzed Regioselective Sulfenylation of Indoles with Sulfonyl Hydrazides

(2013) Fu-Lai Yang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Transition-Metal-Free Synthesis of Unsymmetrical Diaryl Chalcogenides from Arenes and Diaryl Dichalcogenides

(2013) Ch Durga Prasad et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis and antioxidant activity of new C-3 sulfenyl indoles

(2013) Claudio C. Silveira et al.   TETRAHEDRON LETTERS

A Metal-Free Sulfenylation and Bromosulfenylation of Indoles: Controllable Synthesis of 3-Arylthioindoles and 2-Bromo-3-arylthioindoles

(2012) Dayun Huang et al.   ADVANCED SYNTHESIS & CATALYSIS

Transition metal-free direct C–H bond thiolation of 1,3,4-oxadiazoles and related heteroarenes

(2012) Liang-Hua Zou et al.   CHEMICAL COMMUNICATIONS

Visible light-induced 3-sulfenylation of N-methylindoles with arylsulfonyl chlorides

(2012) Min Chen et al.   CHEMICAL COMMUNICATIONS

An Efficient Catalytic Method for Regioselective Sulfenylation of Electron-Rich Aza-Aromatics at Room Temperature

(2012) Enrico Marcantoni et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Iodine-catalyzed oxidative system for 3-sulfenylation of indoles with disulfides using DMSO as oxidant under ambient conditions in dimethyl carbonate

(2012) Wenlei Ge et al.   GREEN CHEMISTRY

Toward Highly Potent Cancer Agents by Modulating the C-2 Group of the Arylthioindole Class of Tubulin Polymerization Inhibitors

(2012) Giuseppe La Regina et al.   JOURNAL OF MEDICINAL CHEMISTRY

KOtBu Mediated Synthesis of Phenanthridinones and Dibenzoazepinones

(2012) Bhagat Singh Bhakuni et al.   ORGANIC LETTERS

Copper(I) Iodide Catalyzed 3-Sulfenylation of Indoles with Unsymmetric Benzothiazolyl-Containing Disulfides at Room Temperature

(2012) Yunyang Wei et al.   SYNTHESIS-STUTTGART

Efficient synthesis of 3-selanyl- and 3-sulfanylindoles employing trichloroisocyanuric acid and dichalcogenides

(2012) Claudio C. Silveira et al.   TETRAHEDRON

An efficient copper mediated synthetic methodology for benzo[d]isothiazol-3(2H)-ones and related sulfur–nitrogen heterocycles

(2012) Bhagat Singh Bhakuni et al.   TETRAHEDRON LETTERS

Venting-while-Heating Microwave-Assisted Synthesis of 3-Arylthioindoles

(2012) Giuseppe La Regina et al.   ACS Combinatorial Science

Synthesis of di(hetero)aryl sulfides by directly using arylsulfonyl chlorides as a sulfur source

(2011) Qian Wu et al.   CHEMICAL COMMUNICATIONS

Catalytic asymmetric cleavage of sp3C–N bonds for access to highly enantioenriched N-benzylic sulfonamides

(2011) Xue-Song Wu et al.   CHEMICAL COMMUNICATIONS

Indolylarylsulfones as HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: New Cyclic Substituents at Indole-2-carboxamide

(2011) Giuseppe La Regina et al.   JOURNAL OF MEDICINAL CHEMISTRY

Design and Synthesis of 2-Heterocyclyl-3-arylthio-1H-indoles as Potent Tubulin Polymerization and Cell Growth Inhibitors with Improved Metabolic Stability

(2011) Giuseppe La Regina et al.   JOURNAL OF MEDICINAL CHEMISTRY

An efficient and clean CuI-catalyzed chalcogenylation of aromatic azaheterocycles with dichalcogenides

(2011) Zhen Li et al.   TETRAHEDRON

Copper catalyzed/mediated synthetic methodology for ebselen and related isoselenazolones

(2011) Shah Jaimin Balkrishna et al.   TETRAHEDRON

Copper-catalyzed chalcogenoamination of 2-alkynylanilines with dichalcogenides for one-step synthesis of 3-sulfenylindoles and 3-selenylindoles

(2011) Zhen Li et al.   TETRAHEDRON LETTERS

Cu-Catalyzed Efficient Synthetic Methodology for Ebselen and Related Se−N Heterocycles

(2010) Shah Jaimin Balkrishna et al.   ORGANIC LETTERS

The use of anhydrous CeCl3 as a catalyst for the synthesis of 3-sulfenyl indoles

(2010) Claudio C. Silveira et al.   TETRAHEDRON LETTERS

Palladium-Catalyzed Annulation of 2-(1-Alkynyl)benzenamines with Disulfides: Synthesis of 3-Sulfenylindoles

(2009) Yan-Jin Guo et al.   ADVANCED SYNTHESIS & CATALYSIS

Indolylarylsulfones Bearing Natural and Unnatural Amino Acids. Discovery of Potent Inhibitors of HIV-1 Non-Nucleoside Wild Type and Resistant Mutant Strains Reverse Transcriptase and Coxsackie B4 Virus

(2009) Francesco Piscitelli et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of 3-Sulfenyl- and 3-Selenylindoles by the Pd/Cu-Catalyzed Coupling ofN,N-Dialkyl-2-iodoanilines and Terminal Alkynes, Followed byn-Bu4NI-Induced Electrophilic Cyclization

(2009) Yu Chen et al.   JOURNAL OF ORGANIC CHEMISTRY

Iron(III) Chloride: A Versatile Catalyst for the Practical Synthesis of 3-Sulfenylindoles

(2009) Jhillu Yadav et al.   SYNTHESIS-STUTTGART

Copper-catalyzed direct thiolation of benzoxazole with diaryl disulfides and aryl thiols

(2009) Shin-ichi Fukuzawa et al.   TETRAHEDRON LETTERS

A Novel Synthetic Route to 3-Sulfenyl- and 3-Selenylindoles byn-Bu4NI-Induced Electrophilic Cyclization

(2008) Yu Chen et al.   ORGANIC LETTERS

Oxone‐Mediated Oxidative 3‐Arylthio Substitution of Indoles

(2008) Guaili Wu et al.   SYNTHETIC COMMUNICATIONS