Design and synthesis of tryptophan containing dipeptide derivatives as formyl peptide receptor 1 antagonist

A non-peptide receptor inhibitor with selectivity for one of the neutrophil formyl peptide receptors, FPR 1

(2012) Hülya Çevik-Aras et al.   BIOCHEMICAL PHARMACOLOGY

Antioxidant and antimicrobial activities of ethyl acetate extract, fractions and compounds from stem bark of Albizia adianthifolia (Mimosoideae)

(2012) Jean de Dieu Tamokou et al.   BMC Complementary and Alternative Medicine

Structure-Based Rationale Design and Synthesis of Aurantiamide Acetate Analogues - Towards a New Class of Potent Analgesic and Anti-inflammatory Agents

(2012) Ramesh Suhas et al.   Chemical Biology & Drug Design

G protein-coupled receptor FPR1 as a pharmacologic target in inflammation and human glioblastoma

(2012) Mingyong Liu et al.   INTERNATIONAL IMMUNOPHARMACOLOGY

Chemical Constituents from Stem Bark and Roots of Clausena anisata

(2012) Jules Songue et al.   MOLECULES

Synthesis and biological evaluation of Matijing-Su derivatives as potent anti-HBV agents

(2011) Jingying Qiu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Discovery of pyrazoles as novel FPR1 antagonists

(2011) Andrew D. Morley et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Neutrophil elastase inhibitors

(2011) William C Groutas et al.   EXPERT OPINION ON THERAPEUTIC PATENTS

2-(2-Fluorobenzamido)benzoate ethyl ester (EFB-1) inhibits superoxide production by human neutrophils and attenuates hemorrhagic shock-induced organ dysfunction in rats

(2011) Huang-Ping Yu et al.   FREE RADICAL BIOLOGY AND MEDICINE

Anthranilic acid-based inhibitors of phosphodiesterase: Design, synthesis, and bioactive evaluation

(2011) Yih-Dih Cheng et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Cytotoxic N-(fluorenyl-9-methoxycarbonyl) (Fmoc)-dipeptides: Structure–activity relationships and synergistic studies

(2010) Chiao-Ting Yen et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and evaluation of benzoxazinone derivatives on activity of human neutrophil elastase and on hemorrhagic shock-induced lung injury in rats

(2010) Pei-Wen Hsieh et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

The Annexin I Sequence Gln9-Ala10-Trp11-Phe12Is a Core Structure for Interaction with the Formyl Peptide Receptor 1

(2010) Charlotta Movitz et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Intramolecular Hydrogen Bonding in Medicinal Chemistry

(2010) Bernd Kuhn et al.   JOURNAL OF MEDICINAL CHEMISTRY

AmideCis−TransIsomerization in Aqueous Solutions of MethylN-Formyl-d-glucosaminides and MethylN-Acetyl-d-glucosaminides: Chemical Equilibria and Exchange Kinetics

(2010) Xiaosong Hu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis and anti-hepatitis B virus activities of Matijing-Su derivatives

(2009) Bixue Xu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Respiratory burst function of ovine neutrophils

(2009) John-Paul Tung et al.   BMC IMMUNOLOGY

Chemical constituents from the radix of Curcuma wenyujin

(2009) Zhong-Jun Ma et al.   FITOTERAPIA

Phagocytic leukocytes and reactive oxygen species

(2009) John M. Robinson   HISTOCHEMISTRY AND CELL BIOLOGY

Identification of Novel Small-Molecule Agonists for Human Formyl Peptide Receptors and Pharmacophore Models of Their Recognition

(2009) L. N. Kirpotina et al.   MOLECULAR PHARMACOLOGY

International Union of Basic and Clinical Pharmacology. LXXIII. Nomenclature for the Formyl Peptide Receptor (FPR) Family

(2009) R. D. Ye et al.   PHARMACOLOGICAL REVIEWS

The Role of Neutrophils in the Pathogenesis of Transfusion-Related Acute Lung Injury

(2009) Yoke Lin Fung et al.   TRANSFUSION MEDICINE REVIEWS

Design and synthesis of new N-(fluorenyl-9-methoxycarbonyl) (Fmoc)-dipeptides as anti-inflammatory agents

(2008) Chiao-Ting Yen et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Cyclopeptides with Anti-inflammatory Activity from Seeds ofAnnona montana

(2008) Pei-Hsuan Chuang et al.   JOURNAL OF NATURAL PRODUCTS

Identification of Novel Formyl Peptide Receptor-Like 1 Agonists That Induce Macrophage Tumor Necrosis Factor   Production

(2008) I. A. Schepetkin et al.   MOLECULAR PHARMACOLOGY