Ready synthesis of free N-H 2-arylindoles via the copper-catalyzed amination of 2-bromo-arylacetylenes with aqueous ammonia and sequential intramolecular cyclization

A P,N-Ligand for Palladium-Catalyzed Ammonia Arylation: Coupling of Deactivated Aryl Chlorides, Chemoselective Arylations, and Room Temperature Reactions

(2010) Rylan J. Lundgren et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Organometallic Reactions of Ammonia

(2010) Jessica L. Klinkenberg et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A general and mild domino approach to substituted 1-aminoindoles

(2010) Nis Halland et al.   CHEMICAL COMMUNICATIONS

Direct amination of aryl halides with ammonia

(2010) Yoann Aubin et al.   CHEMICAL SOCIETY REVIEWS

A Simple and Efficient Catalytic System for Coupling Aryl Halides with Aqueous Ammonia in Water

(2010) Zhiqing Wu et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Copper catalysis in the construction of indole and benzo[b]furan rings

(2010) Sandro Cacchi et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper-CatalyzedN-Arylation/Hydroamin(d)ation Domino Synthesis of Indoles and its Application to the Preparation of a Chek1/KDR Kinase Inhibitor Pharmacophore

(2009) Lutz Ackermann et al.   ADVANCED SYNTHESIS & CATALYSIS

An Efficient Copper-Catalyzed Amination of Aryl Halides by Aqueous Ammonia

(2009) Deping Wang et al.   ADVANCED SYNTHESIS & CATALYSIS

A General and Mild Palladium-Catalyzed Domino Reaction for the Synthesis of 2H-Indazoles

(2009) Nis Halland et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Efficient copper-catalyzed coupling of aryl chlorides, bromides and iodides with aqueous ammonia

(2009) Hanhui Xu et al.   CHEMICAL COMMUNICATIONS

CuI/4-Hydro-l-proline as a More Effective Catalytic System for Coupling of Aryl Bromides withN-Boc Hydrazine and Aqueous Ammonia

(2009) Liqin Jiang et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed Coupling of Ammonia with Aryl Chlorides, Bromides, Iodides, and Sulfonates: A General Method for the Preparation of Primary Arylamines

(2009) Giang D. Vo et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

One-pot Synthesis of Benzo[b]thiophenes and Benzo[b]selenophenes fromo-Halo-Substituted Ethynylbenzenes: Convenient Approach to Mono-, Bis-, and Tris-Chalcogenophene-Annulated Benzenes

(2009) Tomoya Kashiki et al.   ORGANIC LETTERS

Sonogashira Cross-Coupling Reactions and Construction of the Indole Ring System Using a Robust, Silica-Supported Palladium Catalyst

(2009) Elizabeth Tyrrell et al.   SYNTHESIS-STUTTGART

Palladium-free zinc-mediated hydroamination of alkynes: efficient synthesis of indoles from 2-akynylaniline derivatives

(2009) Kentaro Okuma et al.   TETRAHEDRON LETTERS

One-Pot/Four-Step/Palladium-Catalyzed Synthesis of Indole Derivatives: The Combination of Heterogeneous and Homogeneous Systems

(2008) Hayato Sakai et al.   ADVANCED SYNTHESIS & CATALYSIS

Palladium-Catalyzed Direct Arylation of (Hetero)Arenes with Aryl Boronic Acids

(2008) Shang-Dong Yang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Very Simple Copper-Catalyzed Synthesis of Anilines by Employing Aqueous Ammonia

(2008) Ning Xia et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Ammonium salts as an inexpensive and convenient nitrogen source in the Cu-catalyzed amination of aryl halides at room temperature

(2008) Jinho Kim et al.   CHEMICAL COMMUNICATIONS

Copper-Mediated Coupling Reactions and Their Applications in Natural Products and Designed Biomolecules Synthesis

(2008) Gwilherm Evano et al.   CHEMICAL REVIEWS

InBr3-Promoted Divergent Approach to Polysubstituted Indoles and Quinolines from 2-Ethynylanilines: Switch from an Intramolecular Cyclization to an Intermolecular Dimerization by a Type of Terminal Substituent Group

(2008) Norio Sakai et al.   JOURNAL OF ORGANIC CHEMISTRY

Tandem copper-catalysed aryl and alkenyl amination reactions: the synthesis of N-functionalised indoles

(2008) Roy C. Hodgkinson et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Indium-HI-mediated one-pot reaction of 1-(2-arylethynyl)-2-nitroarenes to 2-arylindoles

(2008) Ji Sook Kim et al.   TETRAHEDRON LETTERS

Palladium-Catalyzed Aryl Amination–Heck Cyclization Cascade: A One-Flask Approach to 3-Substituted Indoles

(2007) Thomas Jensen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION