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Title
Comprehensive analysis of kinase inhibitor selectivity
Authors
Keywords
-
Journal
NATURE BIOTECHNOLOGY
Volume 29, Issue 11, Pages 1046-1051
Publisher
Springer Nature
Online
2011-10-31
DOI
10.1038/nbt.1990
References
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Related references
Note: Only part of the references are listed.- High-Throughput Kinase Profiling: A More Efficient Approach toward the Discovery of New Kinase Inhibitors
- (2011) Chandrasekhar V. Miduturu et al. CHEMISTRY & BIOLOGY
- Navigating the kinome
- (2011) James T Metz et al. Nature Chemical Biology
- Characterization of a selective inhibitor of the Parkinson's disease kinase LRRK2
- (2011) Xianming Deng et al. Nature Chemical Biology
- Activation State-Dependent Binding of Small Molecule Kinase Inhibitors: Structural Insights from Biochemistry
- (2010) Lisa M. Wodicka et al. CHEMISTRY & BIOLOGY
- Kinase inhibition-related adverse events predicted from in vitro kinome and clinical trial data
- (2010) Xinan Yang et al. JOURNAL OF BIOMEDICAL INFORMATICS
- Trends in Kinase Selectivity: Insights for Target Class-Focused Library Screening
- (2010) Shana L. Posy et al. JOURNAL OF MEDICINAL CHEMISTRY
- Fluorophore Labeling of the Glycine-Rich Loop as a Method of Identifying Inhibitors That Bind to Active and Inactive Kinase Conformations†
- (2010) Jeffrey R. Simard et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Small-molecule kinase inhibitors provide insight into Mps1 cell cycle function
- (2010) Nicholas Kwiatkowski et al. Nature Chemical Biology
- The lack of target specificity of small molecule anticancer kinase inhibitors is correlated with their ability to damage myocytes in vitro
- (2010) Brian B. Hasinoff et al. TOXICOLOGY AND APPLIED PHARMACOLOGY
- Kinase selectivity potential for inhibitors targeting the ATP binding site: a network analysis
- (2009) Danzhi Huang et al. BIOINFORMATICS
- AC220 is a uniquely potent and selective inhibitor of FLT3 for the treatment of acute myeloid leukemia (AML)
- (2009) P. P. Zarrinkar et al. BLOOD
- SGX523 is an exquisitely selective, ATP-competitive inhibitor of the MET receptor tyrosine kinase with antitumor activity in vivo
- (2009) S. G. Buchanan et al. MOLECULAR CANCER THERAPEUTICS
- Identification of a Kinase Profile that Predicts Chromosome Damage Induced by Small Molecule Kinase Inhibitors
- (2009) Andrew J. Olaharski et al. PLoS Computational Biology
- Assessment of Chemical Coverage of Kinome Space and Its Implications for Kinase Drug Discovery
- (2008) Paul Bamborough et al. JOURNAL OF MEDICINAL CHEMISTRY
- Global target profile of the kinase inhibitor bosutinib in primary chronic myeloid leukemia cells
- (2008) L L Remsing Rix et al. LEUKEMIA
- A quantitative analysis of kinase inhibitor selectivity
- (2008) Mazen W Karaman et al. NATURE BIOTECHNOLOGY
- High-throughput kinase profiling as a platform for drug discovery
- (2008) David M. Goldstein et al. NATURE REVIEWS DRUG DISCOVERY
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