Cinnamoyl-Oxaborole Amides: Synthesis and Their in Vitro Biological Activity

New thiazolidine-2,4-dione derivatives combined with organometallic ferrocene: Synthesis, structure and antiparasitic activity

(2018) Ogunyemi O. Oderinlo et al.   APPLIED ORGANOMETALLIC CHEMISTRY

Novel lead compounds in pre-clinical development against African sleeping sickness

(2017) Michael Berninger et al.   MedChemComm

Antitrypanosomal Activities and Mechanisms of Action of Novel Tetracyclic Iridoids from Morinda lucida Benth.

(2016) Kofi D. Kwofie et al.   ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

The animal trypanosomiases and their chemotherapy: a review

(2016) FEDERICA GIORDANI et al.   PARASITOLOGY

One-pot synthesis of amides from carboxylic acids activated using thionyl chloride

(2016) A. Leggio et al.   RSC Advances

Discovery of an orally bioavailable isoxazoline benzoxaborole ( AN8030 ) as a long acting animal ectoparasiticide

(2015) Yong-Kang Zhang et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Recent Developments in the Chemistry and Biological Applications of Benzoxaboroles

(2015) Agnieszka Adamczyk-Woźniak et al.   CHEMICAL REVIEWS

Anti-Trypanosomal Activity of Nigerian Plants and Their Constituents

(2015) Ngozi Nwodo et al.   MOLECULES

An analysis of the attrition of drug candidates from four major pharmaceutical companies

(2015) Michael J. Waring et al.   NATURE REVIEWS DRUG DISCOVERY

A mild and efficient amide formation reaction mediated by P(OEt)3 and iodine

(2015) Pei-Jiang Chen et al.   RSC Advances

Computer-Aided Drug Discovery Approaches against the Tropical Infectious Diseases Malaria, Tuberculosis, Trypanosomiasis, and Leishmaniasis

(2015) Peter M. Njogu et al.   ACS Infectious Diseases

Neglected Parasitic Infections in the United States: Trichomoniasis

(2014) W. Evan Secor et al.   AMERICAN JOURNAL OF TROPICAL MEDICINE AND HYGIENE

The unique chemistry of benzoxaboroles: Current and emerging applications in biotechnology and therapeutic treatments

(2014) C. Tony Liu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Recent Approaches to Chemical Discovery and Development Against Malaria and the Neglected Tropical Diseases Human African Trypanosomiasis and Schistosomiasis

(2014) Mathew Njoroge et al.   CHEMICAL REVIEWS

Natural Cinnamic Acids, Synthetic Derivatives and Hybrids with Antimicrobial Activity

(2014) Juan Guzman   MOLECULES

A Palladium on Carbon Catalyzed One-Pot Synthesis of Substituted Benzimidazoles

(2014) Soumen Joardar et al.   SYNTHESIS-STUTTGART

The role of modern drug discovery in the fight against neglected and tropical diseases

(2014) Jeremy N. Burrows et al.   MedChemComm

Co-infection of tuberculosis and parasitic diseases in humans: a systematic review

(2013) Xin-Xu Li et al.   Parasites & Vectors

A Dual Read-Out Assay to Evaluate the Potency of Compounds Active against Mycobacterium tuberculosis

(2013) Juliane Ollinger et al.   PLoS One

The synthesis of benzoxaboroles and their applications in medicinal chemistry

(2013) Jiong Zhang et al.   Science China-Chemistry

A current analysis of chemotherapy strategies for the treatment of human African trypanosomiasis

(2013) Peter Babokhov et al.   Pathogens and Global Health

Pathway-Selective Sensitization of Mycobacterium tuberculosis for Target-Based Whole-Cell Screening

(2012) Garth L. Abrahams et al.   CHEMISTRY & BIOLOGY

Design, Synthesis and Biological Evaluation of Potent Azadipeptide Nitrile Inhibitors and Activity-Based Probes as Promising Anti-Trypanosoma bruceiAgents

(2012) Peng-Yu Yang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Cinnamic Acid/Chloroquinoline Conjugates as Potent Agents against Chloroquine-Resistant Plasmodium falciparum

(2012) Bianca Pérez et al.   ChemMedChem

Cinnamic Acid Derivatives in Tuberculosis, Malaria and Cardiovascular Diseases - A Review

(2012) Prithwiraj De et al.   CURRENT ORGANIC CHEMISTRY

Comprehensive analysis of methods used for the evaluation of compounds against Mycobacterium tuberculosis

(2012) Scott G. Franzblau et al.   TUBERCULOSIS

Antitrypanosomal Activity of Fexinidazole, a New Oral Nitroimidazole Drug Candidate for Treatment of Sleeping Sickness

(2011) Marcel Kaiser et al.   ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

Design, synthesis and antimycobacterial activity of cinnamide derivatives: A molecular hybridization approach

(2011) Manoj D. Kakwani et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Boron-containing inhibitors of synthetases

(2011) Stephen J. Baker et al.   CHEMICAL SOCIETY REVIEWS

Boron-based drugs as antiprotozoals

(2011) Robert T. Jacobs et al.   CURRENT OPINION IN INFECTIOUS DISEASES

Development of novel drugs for human African trypanosomiasis

(2011) Reto Brun et al.   Future Microbiology

Design, Synthesis, and Biological Evaluation of New Cinnamic Derivatives as Antituberculosis Agents

(2011) Prithwiraj De et al.   JOURNAL OF MEDICINAL CHEMISTRY

Putting sleeping sickness to bed

(2011) Cassandra Willyard   NATURE MEDICINE

Innovative Partnerships for Drug Discovery against Neglected Diseases

(2011) Palle H. Jakobsen et al.   PLoS Neglected Tropical Diseases

SCYX-7158, an Orally-Active Benzoxaborole for the Treatment of Stage 2 Human African Trypanosomiasis

(2011) Robert T. Jacobs et al.   PLoS Neglected Tropical Diseases

Synthesis and biological evaluations of P4-benzoxaborole-substituted macrocyclic inhibitors of HCV NS3 protease

(2010) Charles Z. Ding et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Influence of the Substituents on the Structure and Properties of Benzoxaboroles

(2010) Agnieszka Adamczyk-Woźniak et al.   JOURNAL OF PHYSICAL CHEMISTRY A

Benzoxaboroles – Old compounds with new applications

(2009) Agnieszka Adamczyk-Woźniak et al.   JOURNAL OF ORGANOMETALLIC CHEMISTRY

Design and Synthesis of Novel 2-Phenylaminopyrimidine (PAP) Derivatives and Their Antiproliferative Effects in Human Chronic Myeloid Leukemia Cells

(2009) Sheng Chang et al.   MOLECULES

Effectiveness of melarsoprol and eflornithine as first-line regimens for gambiense sleeping sickness in nine Médecins Sans Frontières programmes

(2008) Manica Balasegaram et al.   TRANSACTIONS OF THE ROYAL SOCIETY OF TROPICAL MEDICINE AND HYGIENE

Synthesis and antimycobacterial evaluation of new trans-cinnamic acid hydrazide derivatives

(2007) Samir A. Carvalho et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS