Optimizing Solubility and Permeability of a Biopharmaceutics Classification System (BCS) Class 4 Antibiotic Drug Using Lipophilic Fragments Disturbing the Crystal Lattice

Title
Optimizing Solubility and Permeability of a Biopharmaceutics Classification System (BCS) Class 4 Antibiotic Drug Using Lipophilic Fragments Disturbing the Crystal Lattice
Authors
Keywords
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Journal
JOURNAL OF MEDICINAL CHEMISTRY
Volume 56, Issue 6, Pages 2690-2694
Publisher
American Chemical Society (ACS)
Online
2013-02-25
DOI
10.1021/jm301721e

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