Aurora Kinase Inhibitors Based on the Imidazo[1,2-a]pyrazine Core: Fluorine and Deuterium Incorporation Improve Oral Absorption and Exposure

Title
Aurora Kinase Inhibitors Based on the Imidazo[1,2-a]pyrazine Core: Fluorine and Deuterium Incorporation Improve Oral Absorption and Exposure
Authors
Keywords
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Journal
JOURNAL OF MEDICINAL CHEMISTRY
Volume 54, Issue 1, Pages 201-210
Publisher
American Chemical Society (ACS)
Online
2010-12-04
DOI
10.1021/jm1010995

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