Rapid, one-step, high yielding18F-labeling of an aryltrifluoroborate bioconjugate by isotope exchange at very high specific activity

A historical perspective on the specific activity of radiopharmaceuticals: what have we learned in the 35 years of the ISRC?

(2012) Suzanne E. Lapi et al.   NUCLEAR MEDICINE AND BIOLOGY

Harvesting 18F-fluoride ions in water via direct 18F–19F isotopic exchange: radiofluorination of zwitterionic aryltrifluoroborates and in vivo stability studies

(2012) Zibo Li et al.   MedChemComm

Biomedical Applications of Tetrazine Cycloadditions

(2011) Neal K. Devaraj et al.   ACCOUNTS OF CHEMICAL RESEARCH

Rapid and Simple One-Step F-18 Labeling of Peptides

(2011) Orit Jacobson et al.   BIOCONJUGATE CHEMISTRY

High-Yielding Aqueous18F-Labeling of Peptides via Al18F Chelation

(2011) Christopher A. D’Souza et al.   BIOCONJUGATE CHEMISTRY

New F-18 Prosthetic Group via Oxime Coupling

(2011) Patrick Carberry et al.   BIOCONJUGATE CHEMISTRY

Oxalic Acid Supported Si–18F-Radiofluorination: One-Step Radiosynthesis of N-Succinimidyl 3-(Di-tert-butyl[18F]fluorosilyl)benzoate ([18F]SiFB) for Protein Labeling

(2011) Alexey P. Kostikov et al.   BIOCONJUGATE CHEMISTRY

Inorganic approaches for radiolabelling biomolecules with fluorine-18 for imaging with Positron Emission Tomography

(2011) Gareth E. Smith et al.   DALTON TRANSACTIONS

Chelating Agents and their Use in Radiopharmaceutical Sciences

(2011) B. Wangler et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

Anthranilamide: A Simple, Removableortho-Directing Modifier for Arylboronic Acids Serving also as a Protecting Group in Cross-Coupling Reactions

(2011) Hideki Ihara et al.   ORGANIC LETTERS

A Fluoride-Derived Electrophilic Late-Stage Fluorination Reagent for PET Imaging

(2011) E. Lee et al.   SCIENCE

SiFA Azide: A New Building Block for PET Imaging Using Click Chemistry

(2011) Lutz Tietze et al.   SYNLETT

Towards kit-like 18F-labeling of marimastat, a noncovalent inhibitor drug for in vivo PET imaging cancer associated matrix metalloproteases

(2011) Ying Li et al.   MedChemComm

Aryl Trifluoroborates in Suzuki-Miyaura Coupling: The Roles of Endogenous Aryl Boronic Acid and Fluoride

(2010) Mike Butters et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Matrix Metalloproteinase 9 Targeting Peptides: Syntheses,68Ga-labeling, and Preliminary Evaluation in a Rat Melanoma Xenograft Model

(2010) Tiina Ujula et al.   BIOCONJUGATE CHEMISTRY

Radiosynthesis and Biodistribution of a Prosthetic Group (18F-FENMA) Conjugated to Cyclic RGD Peptides

(2010) Dag Erlend Olberg et al.   BIOCONJUGATE CHEMISTRY

Fast18F Labeling of a Near-Infrared Fluorophore Enables Positron Emission Tomography and Optical Imaging of Sentinel Lymph Nodes

(2010) Richard Ting et al.   BIOCONJUGATE CHEMISTRY

Novel Matrix Metalloproteinase Inhibitor [18F]Marimastat-Aryltrifluoroborate as a Probe for In vivo Positron Emission Tomography Imaging in Cancer

(2010) U. auf dem Keller et al.   CANCER RESEARCH

Substitution of hydroxide by fluoride at the boron center of a BODIPY dye

(2010) Todd W. Hudnall et al.   JOURNAL OF FLUORINE CHEMISTRY

68Ga-Labeled Inhibitors of Prostate-Specific Membrane Antigen (PSMA) for Imaging Prostate Cancer

(2010) Sangeeta Ray Banerjee et al.   JOURNAL OF MEDICINAL CHEMISTRY

A Novel Facile Method of Labeling Octreotide with 18F-Fluorine

(2010) P. Laverman et al.   JOURNAL OF NUCLEAR MEDICINE

Direct One-Step18F-Labeling of Peptides via Nucleophilic Aromatic Substitution

(2009) Jessica Becaud et al.   BIOCONJUGATE CHEMISTRY

New Strategy for the Preparation of Clickable Peptides and Labeling with 1-(Azidomethyl)-4-[18F]-fluorobenzene for PET

(2009) David Thonon et al.   BIOCONJUGATE CHEMISTRY

Single-Step High-Yield Radiosynthesis and Evaluation of a Sensitive18F-Labeled Ligand for Imaging Brain Peripheral Benzodiazepine Receptors with PET

(2009) Emmanuelle Briard et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and Application of [18F]FDG-Maleimidehexyloxime ([18F]FDG-MHO): A [18F]FDG-Based Prosthetic Group for the Chemoselective18F-Labeling of Peptides and Proteins†

(2008) Frank Wuest et al.   BIOCONJUGATE CHEMISTRY

Chemistry with [18F]Fluoride Ion

(2008) Lisheng Cai et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Capturing aqueous [18F]-fluoride with an arylboronic ester for PET: Synthesis and aqueous stability of a fluorescent [18F]-labeled aryltrifluoroborate

(2008) Richard Ting et al.   JOURNAL OF FLUORINE CHEMISTRY

In Vivo Positron Emission Tomography (PET) Imaging with an αvβ6Specific Peptide Radiolabeled using18F-“Click” Chemistry: Evaluation and Comparison with the Corresponding 4-[18F]Fluorobenzoyl- and 2-[18F]Fluoropropionyl-Peptides

(2008) Sven H. Hausner et al.   JOURNAL OF MEDICINAL CHEMISTRY

Radiohalogenated Prostate-Specific Membrane Antigen (PSMA)-Based Ureas as Imaging Agents for Prostate Cancer

(2008) Ying Chen et al.   JOURNAL OF MEDICINAL CHEMISTRY

Substituent Effects on Aryltrifluoroborate Solvolysis in Water: Implications for Suzuki−Miyaura Coupling and the Design of Stable18F-Labeled Aryltrifluoroborates for Use in PET Imaging

(2008) Richard Ting et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of masked haloareneboronic acids via iridium-catalyzed aromatic C–H borylation with 1,8-naphthalenediaminatoborane (danBH)

(2008) Noriyuki Iwadate et al.   JOURNAL OF ORGANOMETALLIC CHEMISTRY

Site-Specific18F-Labeling of the Protein Hormone Leptin Using a General Two-Step Ligation Procedure

(2008) Robert R. Flavell et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Toward [18F]-Labeled Aryltrifluoroborate Radiotracers: In Vivo Positron Emission Tomography Imaging of Stable Aryltrifluoroborate Clearance in Mice

(2008) Richard Ting et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Direct Site-Specific Radiolabeling of an Affibody Protein with 4-[18F]Fluorobenzaldehyde via Oxime Chemistry

(2008) Mohammad Namavari et al.   MOLECULAR IMAGING AND BIOLOGY

Differentially Protected Benzenediboronic Acids:  Divalent Cross-Coupling Modules for the Efficient Synthesis of Boron-Substituted Oligoarenes

(2008) Hiroyoshi Noguchi et al.   ORGANIC LETTERS

Potassium Organotrifluoroborates:  New Perspectives in Organic Synthesis

(2007) Sylvain Darses et al.   CHEMICAL REVIEWS