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CFTR Inhibitors for Treating Diarrheal Disease

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Non-Systemic Drugs: A Critical Review

(2012) Dominique Charmot   CURRENT PHARMACEUTICAL DESIGN

Recent advances and new perspectives in targeting CFTR for therapy of cystic fibrosis and enterotoxin-induced secretory diarrheas

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Potent, Metabolically Stable Benzopyrimido-pyrrolo-oxazine-dione (BPO) CFTR Inhibitors for Polycystic Kidney Disease

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Evidence for intestinal chloride secretion

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Nanomolar Potency Pyrimido-pyrrolo-quinoxalinedione CFTR Inhibitor Reduces Cyst Size in a Polycystic Kidney Disease Model

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Crofelemer, an Antisecretory Antidiarrheal Proanthocyanidin Oligomer Extracted from Croton lechleri, Targets Two Distinct Intestinal Chloride Channels

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Nanomolar CFTR Inhibition by Pore-Occluding Divalent Polyethylene Glycol-Malonic Acid Hydrazides

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Small-Molecule CFTR Inhibitors Slow Cyst Growth in Polycystic Kidney Disease

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