4,5-Dihydro-1H-pyrazole: an indispensable scaffold

Synthesis, biological evaluation and molecular modeling study of pyrazole and pyrazoline derivatives as selective COX-2 inhibitors and anti-inflammatory agents. Part 2

(2012) Magda A.-A. El-Sayed et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and in vitro evaluation of novel tetrazole embedded 1,3,5-trisubstituted pyrazoline derivatives as Entamoeba histolytica growth inhibitors

(2012) Mohmmad Younus Wani et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and synergistic antifungal activities of a pyrazoline based ligand and its copper(II) and nickel(II) complexes with conventional antifungals

(2012) Imran Ali et al.   MICROBIAL PATHOGENESIS

Enantioselective synthesis of bio-relevant 3,5-diaryl pyrazolines

(2012) Olivier Mahé et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis, spectral studies and antimicrobial activities of some 2-naphthyl pyrazoline derivatives

(2012) S.P. Sakthinathan et al.   SPECTROCHIMICA ACTA PART A-MOLECULAR AND BIOMOLECULAR SPECTROSCOPY

Sc(OTf)3-catalyzed, solvent-free domino synthesis of functionalized pyrazoles under controlled microwave irradiation

(2012) Kumkum Kumari et al.   TETRAHEDRON LETTERS

N-(1,3-Diaryl-3-oxopropyl)amides as a new template for xanthine oxidase inhibitors

(2011) Kunal Nepali et al.   BIOORGANIC & MEDICINAL CHEMISTRY

A rational approach for the design and synthesis of 1-acetyl-3,5-diaryl-4,5-dihydro(1H)pyrazoles as a new class of potential non-purine xanthine oxidase inhibitors

(2011) Kunal Nepali et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis, molecular docking and evaluation of thiazolyl-pyrazoline derivatives as EGFR TK inhibitors and potential anticancer agents

(2011) Peng-Cheng Lv et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Graphical contents list

(2011)   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and biological evaluation of some new 2-pyrazolines bearing benzene sulfonamide moiety as potential anti-inflammatory and anti-cancer agents

(2011) Sameena Bano et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

One-pot synthesis of pyrazoline derivatised carbazoles as antitubercular, anticancer agents, their DNA cleavage and antioxidant activities

(2011) Tasneem Taj et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Xanthine oxidase inhibitors: a patent survey

(2011) Raj Kumar et al.   EXPERT OPINION ON THERAPEUTIC PATENTS

Synthesis of 1,3,5-trisubstituted pyrazoline nucleus containing compounds and screening for antimicrobial activity

(2011) Manish Agrawal et al.   MEDICINAL CHEMISTRY RESEARCH

A simple and efficient synthesis of pyrazoles in water

(2011) Jun Wen et al.   TETRAHEDRON

Suzuki–Miyaura reactions of N-protected tribromopyrazoles. Efficient and site-selective synthesis of 3,4,5-triaryl-pyrazoles, 3,5-diaryl-4-bromopyrazoles and 5-aryl-3,4-dibromopyrazoles

(2011) Rasheed Ahmad Khera et al.   TETRAHEDRON

Synthesis and in vitro antitumor activity of new 4,5-dihydropyrazole derivatives

(2010) Cenzo Congiu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis of novel α-pyranochalcones and pyrazoline derivatives as Plasmodium falciparum growth inhibitors

(2010) Gajanan Wanare et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Novel 1,3,5-triphenyl-2-pyrazolines as anti-infective agents

(2010) P.M. Sivakumar et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and molecular modelling studies of prenylated pyrazolines as MAO-B inhibitors

(2010) Rossella Fioravanti et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Design, synthesis, and structure–activity relationships of pyrazole derivatives as potential FabH inhibitors

(2010) Peng-Cheng Lv et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis, analgesic and anti-inflammatory activities of some novel pyrazolines derivatives

(2010) Ratnadeep S. Joshi et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and biological evaluation of N-substituted-3,5-diphenyl-2-pyrazoline derivatives as cyclooxygenase (COX-2) inhibitors

(2010) Rossella Fioravanti et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis, characterization and fluorescence studies of 3,5-diaryl substituted 2-pyrazolines

(2010) Geeta Joshi nee Pant et al.   SPECTROCHIMICA ACTA PART A-MOLECULAR AND BIOMOLECULAR SPECTROSCOPY

Studies on novel D-ring substituted steroidal pyrazolines as potential anticancer agents

(2010) Abid H. Banday et al.   STEROIDS

Regioselective synthesis of 1,3,5- and 1,3,4,5-substituted pyrazoles via acylation of N-Boc-N-substituted hydrazones

(2010) Alessandro Tinarelli et al.   TETRAHEDRON

Pyrazoline bearing benzimidazoles: Search for anticancer agent

(2009) Mohammad Shaharyar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and antimalarial evaluation of 1, 3, 5-trisubstituted pyrazolines

(2009) Badri Narayan Acharya et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Design, synthesis, and biological evaluation of 1-(4-sulfamylphenyl)-3-trifluoromethyl-5-indolyl pyrazolines as cyclooxygenase-2 (COX-2) and lipoxygenase (LOX) inhibitors

(2008) M.V. Ramana Reddy et al.   BIOORGANIC & MEDICINAL CHEMISTRY

New pyrazoline bearing 4(3H)-quinazolinone inhibitors of monoamine oxidase: Synthesis, biological evaluation, and structural determinants of MAO-A and MAO-B selectivity

(2008) Nesrin Gökhan-Kelekçi et al.   BIOORGANIC & MEDICINAL CHEMISTRY

The synthesis, structure and spectroscopic properties of novel oxazolone-, pyrazolone- and pyrazoline-containing heterocycle chromophores

(2008) Yi-Feng Sun et al.   DYES AND PIGMENTS

Synthesis, molecular modeling studies and selective inhibitory activity against MAO of N1-propanoyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives

(2008) Franco Chimenti et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and pharmacological evaluation of a novel series of 5-(substituted)aryl-3-(3-coumarinyl)-1-phenyl-2-pyrazolines as novel anti-inflammatory and analgesic agents

(2008) Suresh Khode et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and antimicrobial evaluation of 1-(benzofuran-2-yl)-4-nitro-3-arylbutan-1-ones and 3-(benzofuran-2-yl)-4,5-dihydro-5-aryl-1-[4-(aryl)-1,3-thiazol-2-yl]-1H-pyrazoles

(2008) Bakr F. Abdel-Wahab et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis, antitubercular activity and docking study of novel cyclic azole substituted diphenyl ether derivatives

(2008) Suvarna G. Kini et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of novel thiazolone-based compounds containing pyrazoline moiety and evaluation of their anticancer activity

(2008) Dmytro Havrylyuk et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Extraction and determination of 2-pyrazoline derivatives using liquid phase microextraction based on solidification of floating organic drop

(2008) Hamid Reza Sobhi et al.   JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS

Syntheses and evaluation of 3-(3-bromo phenyl)-5-phenyl-1-(thiazolo [4,5-b] quinoxaline-2-yl)-2-pyrazoline derivatives

(2007) Asha Budakoti et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Bis-pyrazolines: Synthesis, characterization and antiamoebic activity as inhibitors of growth of Entamoeba histolytica

(2007) Abdul R. Bhat et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY