Enantioselective synthesis of bio-relevant 3,5-diaryl pyrazolines

Organocatalytic Enantioselective Synthesis of Pyrazolidines, Pyrazolines and Pyrazolidinones

(2012) Maitane Fernández et al.   ADVANCED SYNTHESIS & CATALYSIS

Cinchona Alkaloid-Catalyzed Enantioselective Amination of α,β-Unsaturated Ketones: An Asymmetric Approach to Δ2-Pyrazolines

(2011) Nathaniel R. Campbell et al.   ADVANCED SYNTHESIS & CATALYSIS

Pyrazoline based MAO inhibitors: Synthesis, biological evaluation and SAR studies

(2011) Monika Jagrat et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Intramolecular CH Oxidative N-Allylation of C-Homoallylhydrazones to 5-Vinyl-2-pyrazolines Catalyzed by the [Pd(OAc)2]/BIMINAP System

(2011) Thanh-Tung Dang et al.   ChemCatChem

Determination of the absolute configuration of 1,3,5-triphenyl-4,5-dihydropyrazole enantiomers by a combination of VCD, ECD measurements, and theoretical calculations

(2011) Nicolas Vanthuyne et al.   TETRAHEDRON-ASYMMETRY

Enantioselective Phase-Transfer Catalysis: Synthesis of Pyrazolines

(2010) Olivier Mahé et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Development of selective and reversible pyrazoline based MAO-A inhibitors: Synthesis, biological evaluation and docking studies

(2010) Muthukumar Karuppasamy et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and molecular modelling studies of prenylated pyrazolines as MAO-B inhibitors

(2010) Rossella Fioravanti et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and evaluation of some new substituted benzothiazepine and benzoxazepine derivatives as anticonvulsant agents

(2010) Neha Garg et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and biological evaluation of N-substituted-3,5-diphenyl-2-pyrazoline derivatives as cyclooxygenase (COX-2) inhibitors

(2010) Rossella Fioravanti et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

A Catalytic Asymmetric 6 π Electrocyclization: Enantioselective Synthesis of 2-Pyrazolines

(2009) Steffen Müller et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Design, Synthesis, andIn-VivoPharmacological Screening ofN,3-(Substituted Diphenyl)-5-phenyl-1H-pyrazoline-1-carbothioamide Derivatives

(2009) Nadeem Siddiqui et al.   ARCHIV DER PHARMAZIE

Towards development of selective and reversible pyrazoline based MAO-inhibitors: Synthesis, biological evaluation and docking studies

(2009) Anasuya Sahoo et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Catalytic enantioselective 1,3-dipolar cycloadditions of alkyl diazoacetates with α,β-disubstituted acroleins

(2009) Lizhu Gao et al.   CHEMICAL COMMUNICATIONS

Cinchona-based phase-transfer catalysts for asymmetric synthesis

(2009) Sang-sup Jew et al.   CHEMICAL COMMUNICATIONS

Knowledge based identification of MAO-B selective inhibitors using pharmacophore and structure based virtual screening models

(2009) Kiran Boppana et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

TBD-organocatalysed synthesis of pyrazolines

(2009) Olivier Mahé et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

New pyrazoline bearing 4(3H)-quinazolinone inhibitors of monoamine oxidase: Synthesis, biological evaluation, and structural determinants of MAO-A and MAO-B selectivity

(2008) Nesrin Gökhan-Kelekçi et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Pyrazoline-based mycobactin analogues as MAO-inhibitors

(2008) Venkatesan Jayaprakash et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis, molecular modeling studies and selective inhibitory activity against MAO of N1-propanoyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives

(2008) Franco Chimenti et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of novel thiazolone-based compounds containing pyrazoline moiety and evaluation of their anticancer activity

(2008) Dmytro Havrylyuk et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

One-pot three-component synthesis of pyrazoles through a tandem coupling-cyclocondensation sequence

(2008) Hai-Ling Liu et al.   TETRAHEDRON LETTERS