Copper promoted N-alkylation of sulfoximines with alkylboronic acid under mild conditions
出版年份 2017 全文链接
标题
Copper promoted N-alkylation of sulfoximines with alkylboronic acid under mild conditions
作者
关键词
-
出版物
ORGANIC & BIOMOLECULAR CHEMISTRY
Volume 15, Issue 40, Pages 8493-8498
出版商
Royal Society of Chemistry (RSC)
发表日期
2017-09-20
DOI
10.1039/c7ob02234d
参考文献
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注意:仅列出部分参考文献,下载原文获取全部文献信息。- Sulfoximines from a Medicinal Chemist's Perspective: Physicochemical and in vitro Parameters Relevant for Drug Discovery
- (2017) Marcus Frings et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Therapeutic effects of methionine sulfoximine in multiple diseases include and extend beyond inhibition of glutamine synthetase
- (2017) William S. A. Brusilow et al. EXPERT OPINION ON THERAPEUTIC TARGETS
- Copper-catalyzed oxidative decarboxylative coupling of α-keto acids and sulfoximines
- (2017) Chaleena Pimpasri et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Access to N-cyanosulfoximines by transition metal-free iminations of sulfoxides
- (2017) C. A. Dannenberg et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Ruthenium(II)-Catalyzed C–H Oxygenations of Reusable Sulfoximine Benzamides
- (2017) Keshav Raghuvanshi et al. ORGANIC LETTERS
- Ruthenium-Catalyzed Hydroarylation and One-Pot Twofold Unsymmetrical C−H Functionalization of Arenes
- (2016) Koushik Ghosh et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Copper-catalyzed N-thioetherification of sulfoximines using disulfides
- (2016) Hui Zhu et al. CHEMICAL COMMUNICATIONS
- Copper-Catalyzed Amidation of Primary and Secondary Alkyl Boronic Esters
- (2016) Luis M. Mori-Quiroz et al. CHEMISTRY-A EUROPEAN JOURNAL
- The “Cyclopropyl Fragment” is a Versatile Player that Frequently Appears in Preclinical/Clinical Drug Molecules
- (2016) Tanaji T. Talele JOURNAL OF MEDICINAL CHEMISTRY
- Copper-catalyzed oxidative C(sp3)–H/N–H coupling of sulfoximines and amides with simple alkanes via a radical process
- (2015) Fan Teng et al. CHEMICAL COMMUNICATIONS
- Iron-Catalyzed Acylative Dealkylation ofN-Alkylsulfoximines
- (2015) Philip Lamers et al. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
- Aerobic Copper-Catalyzed O-Methylation with Methylboronic Acid
- (2015) Clare E. Jacobson et al. JOURNAL OF ORGANIC CHEMISTRY
- Copper-catalyzed N-methylation/ethylation of sulfoximines
- (2015) Fan Teng et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Silver-Mediated N-Trifluoromethylation of Sulfoximines
- (2015) Fan Teng et al. ORGANIC LETTERS
- Methionine and Buthionine Sulfoximines: Syntheses under Mild and Safe Imidation/Oxidation Conditions
- (2014) Laura Buglioni et al. ADVANCED SYNTHESIS & CATALYSIS
- N-Alkylations ofNH-Sulfoximines andNH-Sulfondiimines with Alkyl Halides Mediated by Potassium Hydroxide in Dimethyl Sulfoxide
- (2014) Christine M. M. Hendriks et al. ADVANCED SYNTHESIS & CATALYSIS
- A copper-mediated oxidative N-cyanation reaction
- (2014) Fan Teng et al. CHEMICAL COMMUNICATIONS
- Fluorinated sulfoximines: syntheses, properties and applications
- (2014) Vincent Bizet et al. CHEMICAL SOCIETY REVIEWS
- Hydroarylations of Heterobicyclic Alkenes through Rhodium-Catalyzed Directed CH Functionalizations of S-Aryl Sulfoximines
- (2014) Wanrong Dong et al. CHEMISTRY-A EUROPEAN JOURNAL
- General synthetic strategies towards N-alkyl sulfoximine building blocks for medicinal chemistry and the use of dimethylsulfoximine as a versatile precursor
- (2014) Frederick W. Goldberg et al. TETRAHEDRON
- Sulfoximines: A Neglected Opportunity in Medicinal Chemistry
- (2013) Ulrich Lücking ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Copper-Catalyzed Oxidative Cross-Coupling of Sulfoximines and Alkynes
- (2013) Long Wang et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Primary Alkylboronic Acids as Highly Active Catalysts for the Dehydrative Amide Condensation of α-Hydroxycarboxylic Acids
- (2013) Risa Yamashita et al. ORGANIC LETTERS
- Copper-Catalyzed N- and O-Alkylation of Amines and Phenols using Alkylborane Reagents
- (2013) Shunsuke Sueki et al. ORGANIC LETTERS
- Selective Formation of Secondary Amides via the Copper-Catalyzed Cross-Coupling of Alkylboronic Acids with Primary Amides
- (2013) Steven A. Rossi et al. ORGANIC LETTERS
- Synthesis of chiral sulfoximine-based thioureas and their application in asymmetric organocatalysis
- (2012) Marcus Frings et al. Beilstein Journal of Organic Chemistry
- N,N-Dimethyl-S-difluoromethyl-S-phenylsulfoximinium tetrafluoroborate: A versatile electrophilic difluoromethylating reagent
- (2011) G.K. Surya Prakash et al. JOURNAL OF FLUORINE CHEMISTRY
- Copper-promoted N-cyclopropylation of anilines and amines by cyclopropylboronic acid
- (2010) Sébastien Bénard et al. CHEMICAL COMMUNICATIONS
- Synthesis of Phosphanyl Sulfoximines Through Phospha-Michael Reaction of Alkenyl Sulfoximines and Their Evaluation as Chiral Bidentate 1,5-N,P Ligands for Palladium in Asymmetric Allylic Alkylation
- (2010) Fabien Lemasson et al. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
- Sulfoximine-substituted trifluoromethylpyrimidine analogs as inhibitors of proline-rich tyrosine kinase 2 (PYK2) show reduced hERG activity
- (2009) Daniel P. Walker et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Selective Monomethylation of Anilines by Cu(OAc)2-Promoted Cross-Coupling with MeB(OH)2
- (2009) Israel González et al. ORGANIC LETTERS
- Fluorinated Johnson Reagent for Transfer-Trifluoromethylation to Carbon Nucleophiles
- (2008) Shun Noritake et al. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
- N-Cyclopropylation of Indoles and Cyclic Amides with Copper(II) Reagent
- (2008) Takayuki Tsuritani et al. ORGANIC LETTERS
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