Access to N-cyanosulfoximines by transition metal-free iminations of sulfoxides

Sulfoximines from a Medicinal Chemist's Perspective: Physicochemical and in vitro Parameters Relevant for Drug Discovery

(2017) Marcus Frings et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of Sulfoximidoyl-Containing Hypervalent Iodine(III) Reagents and Their Use in Transition-Metal-Free Sulfoximidations of Alkynes

(2016) Han Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Transfer of Electrophilic NH Using Convenient Sources of Ammonia: Direct Synthesis of NH Sulfoximines from Sulfoxides

(2016) Marina Zenzola et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Iron-Catalyzed Amination of Sulfides and Sulfoxides with Azides in Photochemical Continuous Flow Synthesis

(2016) Hélène Lebel et al.   ACS Catalysis

Abstract 2828: Rapid identification of potent and highly selective, oral PTEFb Inhibitor BAY 1143572 with first in class potential

(2015) Ulrich TJ Luecking et al.   CANCER RESEARCH

Sulfur imidations: access to sulfimides and sulfoximines

(2015) Vincent Bizet et al.   CHEMICAL SOCIETY REVIEWS

Sulfur Imidations by Light-Induced Ruthenium-Catalyzed Nitrene Transfer Reactions

(2015) Vincent Bizet et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Sulfoximine Carbamates by Rhodium-Catalyzed Nitrene Transfer of Carbamates to Sulfoxides

(2015) Marina Zenzola et al.   JOURNAL OF ORGANIC CHEMISTRY

Development of a Continuous Flow Sulfoxide Imidation Protocol Using Azide Sources under Superacidic Conditions

(2015) Bernhard Gutmann et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Development of a Scalable Process for the Crop Protection Agent Isoclast

(2015) Kim E. Arndt et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Study of Sustainability and Scalability in the Cp*Rh(III)-Catalyzed Direct C–H Amidation with 1,4,2-Dioxazol-5-ones

(2015) Yoonsu Park et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Light-Induced Ruthenium-Catalyzed Nitrene Transfer Reactions: A Photochemical Approach towards N-Acyl Sulfimides and Sulfoximines

(2014) Vincent Bizet et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Rhodium-catalyzed direct synthesis of unprotected NH-sulfoximines from sulfoxides

(2014) Jinmin Miao et al.   CHEMICAL COMMUNICATIONS

Fluorinated sulfoximines: syntheses, properties and applications

(2014) Vincent Bizet et al.   CHEMICAL SOCIETY REVIEWS

Fluorinated Sulfoximines: Preparation, Reactions and Applications

(2014) Xiao Shen et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

General synthetic strategies towards N-alkyl sulfoximine building blocks for medicinal chemistry and the use of dimethylsulfoximine as a versatile precursor

(2014) Frederick W. Goldberg et al.   TETRAHEDRON

Sulfoximines: A Neglected Opportunity in Medicinal Chemistry

(2013) Ulrich Lücking   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantioselective Nitrene Transfer to Sulfides Catalyzed by a Chiral Iron Complex

(2013) Jun Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The Lab Oddity Prevails: Discovery of Pan-CDK Inhibitor (R)-S-Cyclopropyl-S-(4-{[4-{[(1R,2R)-2-hydroxy-1-methylpropyl]oxy}-5-(trifluoromethyl)pyrimidin-2-yl]amino}phenyl)sulfoximide (BAY 1000394) for the Treatment of Cancer

(2013) Ulrich Lücking et al.   ChemMedChem

Synthesis of Sulfondiimines byN-Chlorosuccinimide-Mediated Oxidative Imination of Sulfiliminium Salts

(2012) Mathieu Candy et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

N-Cyano Sulfoximines: COX Inhibition, Anticancer Activity, Cellular Toxicity, and Mutagenicity

(2012) Seong Jun Park et al.   ChemMedChem

BAY 1000394, a Novel Cyclin-Dependent Kinase Inhibitor, with Potent Antitumor Activity in Mono- and in Combination Treatment upon Oral Application

(2012) G. Siemeister et al.   MOLECULAR CANCER THERAPEUTICS

Bioactive sulfoximines: Syntheses and properties of Vioxx® analogs

(2011) Seong Jun Park et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Novel nicotinic action of the sulfoximine insecticide sulfoxaflor

(2011) Gerald B. Watson et al.   INSECT BIOCHEMISTRY AND MOLECULAR BIOLOGY

Discovery and Characterization of Sulfoxaflor, a Novel Insecticide Targeting Sap-Feeding Pests

(2010) Yuanming Zhu et al.   JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY

Biological characterization of sulfoxaflor, a novel insecticide

(2010) Jonathan M Babcock et al.   PEST MANAGEMENT SCIENCE

Sulfoximine-substituted trifluoromethylpyrimidine analogs as inhibitors of proline-rich tyrosine kinase 2 (PYK2) show reduced hERG activity

(2009) Daniel P. Walker et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Iron(II) Triflate as an Efficient Catalyst for the Imination of Sulfoxides

(2009) Olga García Mancheño et al.   ORGANIC LETTERS

Preparation, Use, and Safety ofO-Mesitylenesulfonylhydroxylamine

(2009) Javier Mendiola et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Synthesis of aryl benzyl NH-sulfoximines

(2009) Nicola Barry et al.   TETRAHEDRON

Stereoselective Rhodium-Catalyzed Imination of Sulfides

(2008) Florence Collet et al.   ORGANIC LETTERS