Application of bioluminescence resonance energy transfer to quantitate cell-surface expression of membrane proteins

Functional Rescue of Inactivating Mutations of the Human Neurokinin 3 Receptor Using Pharmacological Chaperones

(2022) Ross C. Anderson et al.   INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES

FRET sensors reveal the retinal entry pathway in the G protein-coupled receptor rhodopsin

(2022) He Tian et al.   iScience

Coordination chemogenetics for activation of GPCR-type glutamate receptors in brain tissue

(2022) Kento Ojima et al.   Nature Communications

Differential Involvement of ACKR3 C-Tail in β-Arrestin Recruitment, Trafficking and Internalization

(2021) Aurélien Zarca et al.   Cells

Recurrent high-impact mutations at cognate structural positions in class A G protein-coupled receptors expressed in tumors

(2021) Eunna Huh et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Identification of novel GPCR partners of the central melanocortin signaling

(2021) Yunpeng Li et al.   Molecular Metabolism

Key phosphorylation sites in GPCR s orchestrate the contribution of β‐Arrestin 1 in ERK 1/2 activation

(2020) Mithu Baidya et al.   EMBO REPORTS

Molecular basis of β-arrestin coupling to formoterol-bound β1-adrenoceptor

(2020) Yang Lee et al.   NATURE

Distinct phosphorylation sites in a prototypical GPCR differently orchestrate β-arrestin interaction, trafficking, and signaling

(2020) Hemlata Dwivedi-Agnihotri et al.   Science Advances

Advances of CCR5 antagonists: From small molecules to macromolecules

(2020) Baowen Qi et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Multiplexed analysis of the secretin-like GPCR-RAMP interactome

(2019) Emily Lorenzen et al.   Science Advances

G protein subtype–specific signaling bias in a series of CCR5 chemokine analogs

(2018) Emily Lorenzen et al.   Science Signaling

Core engagement with β-arrestin is dispensable for agonist-induced vasopressin receptor endocytosis and ERK activation

(2017) Punita Kumari et al.   MOLECULAR BIOLOGY OF THE CELL

Trends in GPCR drug discovery: new agents, targets and indications

(2017) Alexander S. Hauser et al.   NATURE REVIEWS DRUG DISCOVERY

Recurrent activating mutations of G-protein-coupled receptor CYSLTR2 in uveal melanoma

(2016) Amanda R Moore et al.   NATURE GENETICS

Functional competence of a partially engaged GPCR–β-arrestin complex

(2016) Punita Kumari et al.   Nature Communications

NanoBRET—A Novel BRET Platform for the Analysis of Protein–Protein Interactions

(2015) Thomas Machleidt et al.   ACS Chemical Biology

Application of BRET to monitor ligand binding to GPCRs

(2015) Leigh A Stoddart et al.   NATURE METHODS

Engineered Luciferase Reporter from a Deep Sea Shrimp Utilizing a Novel Imidazopyrazinone Substrate

(2012) Mary P. Hall et al.   ACS Chemical Biology

HaloTag: A Novel Protein Labeling Technology for Cell Imaging and Protein Analysis

(2008) Georgyi V. Los et al.   ACS Chemical Biology