Application of BRET to monitor ligand binding to GPCRs

Bioluminescent sensor proteins for point-of-care therapeutic drug monitoring

(2014) Rudolf Griss et al.   Nature Chemical Biology

Fluorescent ligands to investigate GPCR binding properties and oligomerization

(2013) Martin Cottet et al.   BIOCHEMICAL SOCIETY TRANSACTIONS

The evolving small-molecule fluorescent-conjugate toolbox for Class A GPCRs

(2013) Andrea J Vernall et al.   BRITISH JOURNAL OF PHARMACOLOGY

Conversion of a non-selective adenosine receptor antagonist into A3-selective high affinity fluorescent probes using peptide-based linkers

(2013) Andrea J. Vernall et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Engineered Luciferase Reporter from a Deep Sea Shrimp Utilizing a Novel Imidazopyrazinone Substrate

(2012) Mary P. Hall et al.   ACS Chemical Biology

Effect of enhanced Renilla luciferase and fluorescent protein variants on the Förster distance of Bioluminescence resonance energy transfer (BRET)

(2012) Helen Dacres et al.   BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS

Fragment Screening at Adenosine-A3 Receptors in Living Cells Using a Fluorescence-Based Binding Assay

(2012) Leigh A. Stoddart et al.   CHEMISTRY & BIOLOGY

Highly Potent and Selective Fluorescent Antagonists of the Human Adenosine A3 Receptor Based on the 1,2,4-Triazolo[4,3-a]quinoxalin-1-one Scaffold

(2012) Andrea J. Vernall et al.   JOURNAL OF MEDICINAL CHEMISTRY

Molecular determinants of A2AR-D2R allosterism: role of the intracellular loop 3 of the D2R

(2012) Víctor Fernández-Dueñas et al.   JOURNAL OF NEUROCHEMISTRY

Single-molecule analysis of fluorescently labeled G-protein-coupled receptors reveals complexes with distinct dynamics and organization

(2012) D. Calebiro et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Allosteric interactions across native adenosine-A3 receptor homodimers: quantification using single-cell ligand-binding kinetics

(2011) Lauren T. May et al.   FASEB JOURNAL

Influence of fluorophore and linker composition on the pharmacology of fluorescent adenosine A1 receptor ligands

(2010) Jillian G Baker et al.   BRITISH JOURNAL OF PHARMACOLOGY