Three‐Component Vicinal Sulfonamination of Alkynes toward 3‐Sulfonylindoles via the Insertion of Sulfur Dioxide

Copper-Catalyzed Regioselective 1,4-Selenosulfonylation of 1,3-Enynes to Access Cyanoalkylsulfonylated Allenes

(2021) Fu-Sheng He et al.   ORGANIC LETTERS

Photoredox‐Catalyzed Functionalization of Alkenes with Thiourea Dioxide: Construction of Alkyl Sulfones or Sulfonamides

(2020) Yuewen Li et al.   CHINESE JOURNAL OF CHEMISTRY

Sequential C–S and S–N Coupling Approach to Sulfonamides

(2020) Kai Chen et al.   ORGANIC LETTERS

Sodium Dithionite‐Mediated Decarboxylative Sulfonylation: Facile Access to Tertiary Sulfones

(2020) Yaping Li et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Sulfonylation from sodium dithionite or thiourea dioxide

(2020) Fu-Sheng He et al.   CHINESE CHEMICAL LETTERS

Site-Selective C–H Functionalization–Sulfination Sequence to Access Aryl Sulfonamides

(2020) Eva Maria Alvarez et al.   ORGANIC LETTERS

Sulfonylation of Aryl/Alkyl Halides with Sulfur Dioxide under Photoinduced Conditions

(2020) Yuewen Li et al.   CHEMISTRY LETTERS

Metal‐Free Synthesis of ( E )‐Vinyl Sulfones via An Insertion of Sulfur Dioxide/1,5‐Hydrogen Atom Transfer Sequence

(2020) Fu‐Sheng He et al.   ADVANCED SYNTHESIS & CATALYSIS

New Dimensions in Rongalite Chemistry: The Land of Opportunities in Organic Synthesis and Material Sciences

(2020) Rashid Ali   ChemistrySelect

Synthesis of 3-(Methylsulfonyl)benzo[b]thiophenes from Methyl(2-alkynylphenyl)sulfanes and Sodium Metabisulfite via a Radical Relay Strategy

(2019) Xinxing Gong et al.   ORGANIC LETTERS

Metal‐Free Synthesis of Thiosulfonates via Insertion of Sulfur Dioxide

(2019) Guoqing Li et al.   ADVANCED SYNTHESIS & CATALYSIS

Direct C( sp 2 )‐H Arylsulfonylation of Enamides via Iridium(III)‐Catalyzed Insertion of Sulfur Dioxide with Aryldiazonium Tetrafluoroborates

(2019) Tong‐Hao Zhu et al.   ADVANCED SYNTHESIS & CATALYSIS

Photoredox-Catalyzed Sulfonylation of O-Acyl Oximes via Iminyl Radicals with the Insertion of Sulfur Dioxide

(2019) Jun Zhang et al.   ORGANIC LETTERS

TFA promoted multi-component reaction of aryldiazonium with sodium metabisulphite and thiols: Construction of thiosulfonate under transition-metal free conditions

(2019) Cheng-Mi Huang et al.   CHINESE CHEMICAL LETTERS

Radicals and Sulfur Dioxide: A Versatile Combination for the Construction of Sulfonyl-Containing Molecules

(2018) Kamil Hofman et al.   CHEMISTRY-A EUROPEAN JOURNAL

Visible-light mediated 3-component synthesis of sulfonylated coumarins from sulfur dioxide

(2018) Zhengkai Chen et al.   GREEN CHEMISTRY

Eosin Y photoredox catalyzed net redox neutral reaction for regiospecific annulation to 3-sulfonylindoles via anion oxidation of sodium sulfinate salts

(2018) Rajendra S. Rohokale et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Photo-Driven Synthesis of C6-Polyfunctionalized Phenanthridines from Three-Component Reactions of Isocyanides, Alkynes, and Sulfinic Acids by Electron Donor–Acceptor Complex

(2018) Yang Li et al.   ORGANIC LETTERS

Insertion of sulfur dioxide via a radical process: an efficient route to sulfonyl compounds

(2018) Guanyinsheng Qiu et al.   Organic Chemistry Frontiers

Recent advances in the sulfonylation of alkenes with the insertion of sulfur dioxide via radical reactions

(2018) Guanyinsheng Qiu et al.   CHEMICAL COMMUNICATIONS

Modern approaches for SO2 insertion in heterocyclic synthesis (microreview)

(2018) Krista Suta et al.   Chemistry of Heterocyclic Compounds

Copper-Catalyzed Synthesis of Activated Sulfonate Esters from Boronic Acids, DABSO, and Pentafluorophenol

(2018) Vincent Vedovato et al.   ORGANIC LETTERS

Catalyst-Free Sulfonylation of (Hetero)aryl Iodides with Sodium Dithionite

(2018) Yuewen Li et al.   ADVANCED SYNTHESIS & CATALYSIS

Indole-fused azepines and analogues as anticancer lead molecules: Privileged findings and future directions

(2017) Ashok K. Singh et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Copper-catalyzed S-methylation of sulfonyl hydrazides with TBHP for the synthesis of methyl sulfones in water

(2017) Yu Yang et al.   GREEN CHEMISTRY

Mushroom-Derived Indole Alkaloids

(2017) Joshua A. Homer et al.   JOURNAL OF NATURAL PRODUCTS

Synthesis of Sulfonylated Lactones via Ag-Catalyzed Cascade Sulfonylation/Cyclization of 1,6-Enynes with Sodium Sulfinates

(2017) Wanqing Wu et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Arylsulfonylation and Cyclizative Carbonation of N-(Arylsulfonyl)acrylamides Involving Desulfonative Arrangement toward Sulfonated Oxindoles

(2017) Hepan Wang et al.   ORGANIC LETTERS

Electrooxidative Tandem Cyclization of Activated Alkynes with Sulfinic Acids To Access Sulfonated Indenones

(2017) Jiangwei Wen et al.   ORGANIC LETTERS

Indole diterpenoid natural products as the inspiration for new synthetic methods and strategies

(2017) Michael A. Corsello et al.   Chemical Science

Recent progress in organocatalytic asymmetric total syntheses of complex indole alkaloids

(2017) Jin Song et al.   National Science Review

Reductive insertion of sulfur dioxide for the synthesis of trifluoromethyl thiolsulphonates through a one-pot reaction of aniline and trifluoromethanesulfanylamide

(2017) Jie Sheng et al.   Organic Chemistry Frontiers

Transition-metal-free oxidative reaction of hydrazines and potassium metabisulfite for preparation of sulfonohydrazides

(2017) Yang Wang et al.   Organic Chemistry Frontiers

Markovnikov-Selective Radical Addition of S-Nucleophiles to Terminal Alkynes through a Photoredox Process

(2016) Huamin Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Iron-catalyzed synthesis of arylsulfinates through radical coupling reaction

(2016) Weixi Zhang et al.   CHEMICAL COMMUNICATIONS

Visible-light initiated direct oxysulfonylation of alkenes with sulfinic acids leading to β-ketosulfones

(2016) Daoshan Yang et al.   GREEN CHEMISTRY

Bu4NI-Catalyzed Cross-Coupling between Sulfonyl Hydrazides and Diazo Compounds To Construct β-Carbonyl Sulfones Using Molecular Oxygen

(2016) Yaxiong Wang et al.   ORGANIC LETTERS

tert-Butyl Hydroperoxide (TBHP)-Initiated Vicinal Sulfonamination of Alkynes: A Radical Annulation toward 3-Sulfonylindoles

(2016) Fei Chen et al.   ORGANIC LETTERS

I2/TBHP Mediated C–N and C–H Bond Cleavage of Tertiary Amines toward Selective Synthesis of Sulfonamides and β-Arylsulfonyl Enamines: The Solvent Effect on Reaction

(2016) Junyi Lai et al.   ORGANIC LETTERS

Reaction of Alkyl Halides with Rongalite: One-Pot and Telescoped Syntheses of Aliphatic Sulfonamides, Sulfonyl Fluorides, and Unsymmetrical Sulfones

(2016) Andre Shavnya et al.   ORGANIC LETTERS

Palladium-Catalyzed Synthesis of (Hetero)Aryl Alkyl Sulfones from (Hetero)Aryl Boronic Acids, Unactivated Alkyl Halides, and Potassium Metabisulfite

(2015) Andre Shavnya et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Selective remote C–H sulfonylation of aminoquinolines with arylsulfonyl chlorides via copper catalysis

(2015) Hong-Wen Liang et al.   CHEMICAL COMMUNICATIONS

Copper-Catalyzed γ-Sulfonylation of α,β-Unsaturated Carbonyl Compounds by Means of Silyl Dienol Ethers

(2015) Xiaoguang Liu et al.   ORGANIC LETTERS

Catalytic Arylsulfonyl Radical Triggered 1,7-Enyne Bicyclizations

(2015) Yi-Long Zhu et al.   ORGANIC LETTERS

Base-Induced Radical Carboamination of Nonactivated Alkenes with Aryldiazonium Salts

(2015) Stephanie Kindt et al.   ORGANIC LETTERS

Catalytic arylsulfonyl radical-triggered 1,5-enyne-bicyclizations and hydrosulfonylation of α,β-conjugates

(2015) Zhen-Zhen Chen et al.   Chemical Science

Chemoselective Synthesis of Unsymmetrical Internal Alkynes or Vinyl SulfonesviaPalladium-Catalyzed Cross-Coupling Reaction of Sodium Sulfinates with Alkynes

(2014) Yanli Xu et al.   ADVANCED SYNTHESIS & CATALYSIS

Metal-Free Aminosulfonylation of Aryldiazonium Tetrafluoroborates with DABCO⋅(SO2)2and Hydrazines

(2014) Danqing Zheng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Selective sulfonylation and diazotization of indoles

(2014) Jiang-Kai Qiu et al.   CHEMICAL COMMUNICATIONS

Simple indole alkaloids and those with a non-rearranged monoterpenoid unit

(2013) Minoru Ishikura et al.   NATURAL PRODUCT REPORTS

Sulfonylation of Quinoline N-Oxides with Aryl Sulfonyl Chlorides via Copper-Catalyzed C–H Bonds Activation

(2013) Zhiyong Wu et al.   ORGANIC LETTERS

ZnO-mediated regioselective C-arylsulfonylation of indoles: a facile solvent-free synthesis of 2- and 3-sulfonylindoles and preliminary evaluation of their activity against drug-resistant mutant HIV-1 reverse transcriptases (RTs)

(2013) Graziella Tocco et al.   TETRAHEDRON LETTERS

A palladium-catalyzed reaction of aryl halides, potassium metabisulfite, and hydrazines

(2012) Shengqing Ye et al.   CHEMICAL COMMUNICATIONS

A palladium-catalyzed three-component coupling of arylboronic acids, sulfur dioxide and hydrazines

(2012) Shengqing Ye et al.   CHEMICAL COMMUNICATIONS

Indole Synthesis by Conjugate Addition of Anilines to Activated Acetylenes and an Unusual Ligand-Free Copper(II)-Mediated Intramolecular Cross-Coupling

(2012) Detian Gao et al.   CHEMISTRY-A EUROPEAN JOURNAL

A simple and efficient approach for the sulfonylation of indoles catalyzed by CuI

(2012) Matiur Rahman et al.   Journal of Sulfur Chemistry

Rongalite: A Useful Green Reagent in Organic Synthesis

(2011) Sambasivarao Kotha et al.   CHEMICAL REVIEWS

Rh2(II)-Catalyzed Nitro-Group Migration Reactions: Selective Synthesis of 3-Nitroindoles from β-Nitro Styryl Azides

(2011) Benjamin J. Stokes et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

DABCO-Bis(sulfur dioxide), DABSO, as a Convenient Source of Sulfur Dioxide for Organic Synthesis: Utility in Sulfonamide and Sulfamide Preparation

(2011) Holly Woolven et al.   ORGANIC LETTERS

3-(Arylsulfonyl)-1-(azacyclyl)-1H-indoles are 5-HT6 receptor modulators

(2010) Ronald C. Bernotas et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Dual acting norepinephrine reuptake inhibitors and 5-HT2A receptor antagonists: Identification, synthesis and activity of novel 4-aminoethyl-3-(phenylsulfonyl)-1H-indoles

(2009) Gavin D. Heffernan et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis of 3-Sulfenyl- and 3-Selenylindoles by the Pd/Cu-Catalyzed Coupling ofN,N-Dialkyl-2-iodoanilines and Terminal Alkynes, Followed byn-Bu4NI-Induced Electrophilic Cyclization

(2009) Yu Chen et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed C−H Bond Functionalization with Arylsulfonyl Chlorides

(2009) Xiaodan Zhao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY