期刊
BIOORGANIC & MEDICINAL CHEMISTRY
卷 17, 期 22, 页码 7802-7815出版社
PERGAMON-ELSEVIER SCIENCE LTD
DOI: 10.1016/j.bmc.2009.09.023
关键词
Monoamine reuptake inhibitors; Norepinephrine reuptake inhibitors; NRI; 5-HT2A receptor antagonists; 4-Aminoethyl-3-(phenylsulfonyl)-1H-indoles
The discovery of a series of 4-aminoethyl-3-(phenylsulfonyl)-1H-indoles, dual acting norepinephrine reuptake inhibitors (NRIs) and 5-HT2A receptor antagonists, is described. The synthesis and structure-activity relationship (SAR) of this novel series of compounds is also presented. (C) 2009 Elsevier Ltd. All rights reserved.
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