标题
The antibacterial activity of fluoroquinolone derivatives: An update (2018–2021)
作者
关键词
Fluoroquinolone, Antibacterial, Multidrug-resistant bacteria, Structure-activity relationship, Drug resistance
出版物
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Volume 224, Issue -, Pages 113741
出版商
Elsevier BV
发表日期
2021-08-02
DOI
10.1016/j.ejmech.2021.113741
参考文献
相关参考文献
注意：仅列出部分参考文献，下载原文获取全部文献信息。- Antibiotic resistance and drug modification: Synthesis, characterization and bioactivity of newly modified potent ciprofloxacin derivatives
- (2021) Abdulhakeem Alsughayer et al. BIOORGANIC CHEMISTRY
- Synthesis, antitumor, antibacterial and urease inhibitory evaluation of new piperazinyl N-4 carbamoyl functionalized ciprofloxacin derivatives
- (2021) Mohamed A. A. Abdel-Aal et al. Pharmacological Reports
- In Vitro and In Vivo Antibacterial Activities of a Novel Quinolone Compound, OPS-2071, Against Clostridioides difficile
- (2021) Daisuke Oka et al. ANTIMICROBIAL AGENTS AND CHEMOTHERAPY
- Novel Mannich bases of ciprofloxacin with improved physicochemical properties, antibacterial, anticancer activities and caspase-3 mediated apoptosis
- (2021) Islam M. Abdel-Rahman et al. BIOORGANIC CHEMISTRY
- Recent Innovations in Bacterial Infection Detection and Treatment
- (2021) Carly Deusenbery et al. ACS Infectious Diseases
- Design, Synthesis, and Antibacterial Screening of Some Novel Heteroaryl-Based Ciprofloxacin Derivatives as DNA Gyrase and Topoisomerase IV Inhibitors
- (2021) Lamya H. Al-Wahaibi et al. Pharmaceuticals
- Enhancing the Activity of Drugs by Conjugation to Organometallic Fragments
- (2020) Prinessa Chellan et al. CHEMISTRY-A EUROPEAN JOURNAL
- Design, synthesis and structure-activity relationships of novel 15-membered macrolides: Quinolone/quinoline-containing sidechains tethered to the C-6 position of azithromycin acylides
- (2020) Bing-Zhi Fan et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Fluoroquinolone Metalloantibiotics: A Promising Approach against Methicillin-Resistant Staphylococcus aureus
- (2020) Mariana Ferreira et al. International Journal of Environmental Research and Public Health
- Conjugates of Ciprofloxacin and Levofloxacin with Cell-Penetrating Peptide Exhibit Antifungal Activity and Mammalian Cytotoxicity
- (2020) Natalia Ptaszyńska et al. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES
- Synthesis of Bioactive Complex Small Molecule–Ciprofloxacin Conjugates and Evaluation of Their Antibacterial Activity
- (2020) Rahul Upadhyay et al. ACS Combinatorial Science
- Synthesis, characterization, antimicrobial activity, 3D‐QSAR, DFT, and molecular docking of some ciprofloxacin derivatives and their copper(II) complexes
- (2020) Tarek E. Khalil et al. APPLIED ORGANOMETALLIC CHEMISTRY
- Synthesis and antimicrobial evaluation of new nitric oxide‐donating fluoroquinolone/oxime hybrids
- (2020) Hossameldin A. Aziz et al. ARCHIV DER PHARMAZIE
- Novel C-7 carbon substituted fourth generation fluoroquinolones targeting N. Gonorrhoeae infections
- (2020) Ralph Kirk et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Design, synthesis and antimicrobial evaluation of novel glycosylated-fluoroquinolones derivatives
- (2020) Aya A.M. Mohammed et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Multidrug-Resistant Bacteria in the Community
- (2020) David van Duin et al. INFECTIOUS DISEASE CLINICS OF NORTH AMERICA
- Spectral, structural, biological and molecular docking studies of a new mixed-valence V(IV)/V(V) ofloxacin complex
- (2020) Mina Alikhani et al. JOURNAL OF MOLECULAR STRUCTURE
- Novel N-4-Piperazinyl Ciprofloxacin-Ester Hybrids: Synthesis, Biological Evaluation, and Molecular Docking Studies
- (2020) A. Shahbazi et al. RUSSIAN JOURNAL OF GENERAL CHEMISTRY
- Design, synthesis, molecular docking study, and antibacterial evaluation of some new fluoroquinolone analogues bearing a quinazolinone moiety
- (2020) Maryam Norouzbahari et al. DARU-Journal of Pharmaceutical Sciences
- Design, Synthesis and Pharmacological Evaluation of Some C3 Heterocyclic-Substituted Ciprofloxacin Derivatives as Chimeric Antitubercular Agents
- (2020) Nakka Niveditha et al. CHEMICAL & PHARMACEUTICAL BULLETIN
- Roles of long noncoding RNAs in bacterial infection
- (2020) Yating Wen et al. LIFE SCIENCES
- Discovery of Novel 7-[(1R,5S)-1-Amino-5-fluoro-3-azabicyclo[3.3.0]octan-3-yl]-6-fluoro-1-[(1R,2S)-2-fluorocyclopropane]-8-(methoxy or methyl)quinolones
- (2019) Satoshi Komoriya et al. CHEMICAL & PHARMACEUTICAL BULLETIN
- Biological investigations and spectroscopic studies of new Moxifloxacin/Glycine-Metal complexes
- (2019) Hazem Salaheldin Elshafie et al. CHEMISTRY & BIODIVERSITY
- DESIGN, SYNTHESIS, MOLECULAR DOCKING, AND ANTIBACTERIAL ACTIVITY EVALUATION OF SOME NOVEL NORFLOXACIN ANALOGUES
- (2019) SMARANDA ONIGA FARMACIA
- Synthesis, characterization and biological evaluation of Co(III) complexes with quinolone drugs
- (2019) Máté Kozsup et al. JOURNAL OF INORGANIC BIOCHEMISTRY
- Synthesis, characterization and biological activity of Zn coordination compounds with the quinolone gatifloxacin
- (2019) Chrisoula Kakoulidou et al. POLYHEDRON
- Design, synthesis and anti-bacterial studies of piperazine derivatives against drug resistant bacteria
- (2019) Saba Tahir et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- New fluoroquinolones compounds with endo -nortropine derivatives at C-7 position show antibacterial activity against fluoroquinolone-resistant strains of Staphylococcus aureus
- (2019) Ramkrushna Ashok Salunke et al. Chemical Biology & Drug Design
- Metal Complexes As Promising Agents For Biomedical Applications
- (2019) Natalia V. Loginova et al. CURRENT MEDICINAL CHEMISTRY
- Design and synthesis of aminothiazolyl norfloxacin analogues as potential antimicrobial agents and their biological evaluation
- (2019) Liang-Liang Wang et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Polymeric bisphosphonate derivative of ciprofloxacin – synthesis, structural analysis and antibacterial activity of the prospective conjugate
- (2019) Marcin Sobczak et al. International Journal of Polymeric Materials and Polymeric Biomaterials
- Fluoroquinolones structural and medicinal developments (2013–2018): Where are we now?
- (2019) Ghadeer A.R.Y. Suaifan et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Design, synthesis and molecular docking of new N-4-piperazinyl ciprofloxacin-triazole hybrids with potential antimicrobial activity
- (2019) Hamada H.H. Mohammed et al. BIOORGANIC CHEMISTRY
- Design, synthesis and molecular modeling studies on novel moxifloxacin derivatives as potential antibacterial and antituberculosis agents
- (2019) Aslı Türe et al. BIOORGANIC CHEMISTRY
- Repurposed Antimicrobial Combination Therapy: Tobramycin-Ciprofloxacin Hybrid Augments Activity of the Anticancer Drug Mitomycin C Against Multidrug-Resistant Gram-Negative Bacteria
- (2019) Ronald Domalaon et al. Frontiers in Microbiology
- Design and synthesis of new norfloxacin-1,3,4-oxadiazole hybrids as antibacterial agents against methicillin-resistant Staphylococcus aureus (MRSA)
- (2019) Yong Guo et al. EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES
- Synthesis, molecular docking, antimicrobial evaluation, and DNA cleavage assay of new thiadiazole/oxadiazole ciprofloxacin derivatives
- (2019) Hamada H. H. Mohammed et al. MONATSHEFTE FUR CHEMIE
- Design, synthesis and antibacterial activity evaluation of moxifloxacin-amide-1,2,3-triazole-isatin hybrids
- (2019) Feng Gao et al. BIOORGANIC CHEMISTRY
- Novel 7-substituted Fluoroquinolone Citrate Conjugates as Powerful Antibacterial and Anticancer Agents: Synthesis and Molecular Docking Studies
- (2019) Tejeswara R. Allaka et al. CURRENT ORGANIC CHEMISTRY
- A new exploration towards aminothiazolquinolone oximes as potentially multi-targeting antibacterial agents: Design, synthesis and evaluation acting on microbes, DNA, HSA and topoisomerase IV
- (2019) Liang-Liang Wang et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis and biological evaluation of hybrid quinolone-based quaternary ammonium antibacterial agents
- (2019) Joanna Fedorowicz et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Design, Synthesis and Biological Evaluation of New Piperazin-4-yl-(acetyl-thiazolidine-2,4-dione) Norfloxacin Analogues as Antimicrobial Agents
- (2019) Marc et al. MOLECULES
- Dual Escherichia coli DNA Gyrase A and B Inhibitors with Antibacterial Activity
- (2019) Benedetta Fois et al. ChemMedChem
- Anticancer and antimicrobial effects of novel ciprofloxacin fatty acids conjugates
- (2019) Alicja Chrzanowska et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Theoretical molecular predictions and antimicrobial activities of newly synthesized molecular hybrids of norfloxacin and ciprofloxacin
- (2019) Gurmeet Kaur et al. JOURNAL OF HETEROCYCLIC CHEMISTRY
- A new calcium(II) complex of marbofloxacin showing much lower acute toxicity with retained antibacterial activity
- (2019) Yan-Jie Xie et al. JOURNAL OF INORGANIC BIOCHEMISTRY
- Crystal structure and antibacterial activity of polyoxometalate cobalt-ciprofloxacin complex
- (2019) Guang-Zhi Shen et al. JOURNAL OF MOLECULAR STRUCTURE
- Introduction of the antibacterial drugs norfloxacin and Ciprofloxacin into a polyoxometalate structure: Synthesis, characterization, and antibacterial activity
- (2019) Yu-Long Zou et al. JOURNAL OF MOLECULAR STRUCTURE
- New triorganotin(IV) complexes of quinolone antibacterial drug sparfloxacin: Synthesis, structural characterization, DFT studies and biological activity
- (2018) Rachana Joshi et al. APPLIED ORGANOMETALLIC CHEMISTRY
- In silico study of Moxifloxacin derivatives with possible antibacterial activity against a resistant form of DNA gyrase from Porphyromonas gingivalis
- (2018) Cristian Rocha-Roa et al. ARCHIVES OF ORAL BIOLOGY
- Discovery of a Novel Fluoroquinolone Antibiotic Candidate WFQ-228 with Potent Antimicrobial Activity and the Potential to Overcome Major Drug Resistance
- (2018) Tatsuya Hirano et al. CHEMICAL & PHARMACEUTICAL BULLETIN
- Design, Synthesis and Antibacterial Evaluation of 1-[(1R, 2S)-2-Fluorocyclopropyl]ciprofloxacin-1,2,4-triazole-5(4H )-thione Hybrids
- (2018) Yang Gao et al. CHEMISTRY & BIODIVERSITY
- Biology-Oriented Drug Synthesis (BIODS) Approach towards Synthesis of Ciprofloxacin-Dithiocarbamate Hybrids and Their Antibacterial Potential both in vitro and in silico
- (2018) Ensieh Nasli Esfahani et al. CHEMISTRY & BIODIVERSITY
- Discovery of Benzimidazole-Quinolone Hybrids as New Cleaving Agents toward Drug-Resistant Pseudomonas aeruginosa DNA
- (2018) Ya-Nan Wang et al. ChemMedChem
- Ciprofloxacin-metal complexes –stability and toxicity tests in the presence of humic substances
- (2018) Agnieszka Cuprys et al. CHEMOSPHERE
- Novel ciprofloxacin hybrids using biology oriented drug synthesis (BIODS) approach: Anticancer activity, effects on cell cycle profile, caspase-3 mediated apoptosis, topoisomerase II inhibition, and antibacterial activity
- (2018) Asmaa E. Kassab et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Design, synthesis and antimicrobial evaluation of propylene-tethered ciprofloxacin-isatin hybrids
- (2018) Ruo Wang et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis, antibacterial properties and 2D-QSAR studies of quinolone-triazole conjugates
- (2018) Hassan M. Faidallah et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Design, Synthesis, and Biological Evaluation of Novel 8-Methoxyquinolones Bearing Fused Pyrrolidinyl Moieties at the C-7 Position with Potent Antibacterial Activity Against Respiratory Pathogens
- (2018) Takashi Odagiri et al. HETEROCYCLES
- Design, Synthesis, and In Vitro Antibacterial Activities of Propylene-tethered Gatifloxacin-isatin Hybrids
- (2018) Hua Guo JOURNAL OF HETEROCYCLIC CHEMISTRY
- 4-Quinolone Derivatives and Their Activities Against Gram-negative Pathogens
- (2018) Dan Jiang JOURNAL OF HETEROCYCLIC CHEMISTRY
- Synthesis, spectroscopic, thermal, biological, morphological and molecular docking studies of the different quinolone drugs and their cobalt(II) complexes
- (2018) Foziah A. Al-Saif et al. JOURNAL OF MOLECULAR LIQUIDS
- Combined experimental and theoretical studies on the diorganotin(IV) complexes of sparfloxacin: Synthesis, spectroscopic and DFT studies, and biological activity
- (2018) Rachana Joshi et al. JOURNAL OF MOLECULAR STRUCTURE
- Chemical and biological evaluation of moxifloxacin-benzimidazole mixed ligands complexes: Anti-cancer and anti-oxidant activities
- (2018) Heba M. Refaat et al. JOURNAL OF MOLECULAR STRUCTURE
- Esterase-Catalyzed Siderophore Hydrolysis Activates an Enterobactin–Ciprofloxacin Conjugate and Confers Targeted Antibacterial Activity
- (2018) Wilma Neumann et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Enhanced Antibacterial Activity of Endo-nortropine Substituted (C-7) Fluoroquinolones Against V. cholerae, S. aureus and B. subtilis
- (2018) Ramkrushna Ashok Salunke et al. Letters in Drug Design & Discovery
- Synthesis, Spectroscopic, and Biological Studies of Mixed Ligand Complexes of Gemifloxacin and Glycine with Zn(II), Sn(II), and Ce(III)
- (2018) Shimaa Sakr et al. MOLECULES
- The role of vaccines in preventing bacterial antimicrobial resistance
- (2018) Kathrin U Jansen et al. NATURE MEDICINE
- Recent updates of fluoroquinolones as antibacterial agents
- (2018) Hend A. A. Ezelarab et al. ARCHIV DER PHARMAZIE
- Quinolone derivatives and their activities against methicillin-resistant Staphylococcus aureus (MRSA)
- (2018) Chuan Gao et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Recent developments of quinolone-based derivatives and their activities against Escherichia coli
- (2018) Feng Gao et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Interaction of triorganotin(IV) moiety with quinolone antibacterial drug ciprofloxacin: Synthesis, spectroscopic investigation, electronic structure calculation, and biological evaluation
- (2018) Rachana Joshi et al. HETEROATOM CHEMISTRY
- Design, Synthesis, and Antibacterial Evaluation of Propylene-tethered 8-Methoxyl Ciprofloxacin-isatin Hybrids
- (2018) Hua Guo JOURNAL OF HETEROCYCLIC CHEMISTRY
- Design, Synthesis, and Biological Evaluation of Novel 7-[(3aS,7aS)-3a-Aminohexahydropyrano[3,4-c]pyrrol-2(3H)-yl]-8-methoxyquinolines with Potent Antibacterial Activity against Respiratory Pathogens
- (2018) Takashi Odagiri et al. JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis and Antibacterial/Antitubercular/Antioxidant Activities of Compounds Containing Fluoroquinolone Ring Linked to a 4-thiazolidinone Moiety
- (2018) Tejeswara Rao Allaka et al. Letters in Drug Design & Discovery
- New model of metalloantibiotic: synthesis, structure and biological activity of a zinc(ii) mononuclear complex carrying two enrofloxacin and sulfadiazine antibiotics
- (2018) Amina Boughougal et al. NEW JOURNAL OF CHEMISTRY
- Synthesis, Antimicrobial Activity and QSAR Studies of Some New Sparfloxacin Derivatives
- (2018) Ayush Kumar et al. PHARMACEUTICAL CHEMISTRY JOURNAL
- New ciprofloxacin–dithiocarbamate–benzyl hybrids: design, synthesis, antibacterial evaluation, and molecular modeling studies
- (2018) Ensieh Nasli Esfahani et al. RESEARCH ON CHEMICAL INTERMEDIATES
- New N -4 piperazinyl derivatives of norfloxacin: design, synthesis, and correlation of calculated physicochemical parameters with antibacterial activity
- (2018) Gamal El-Din ABUO-RAHMA et al. TURKISH JOURNAL OF CHEMISTRY
- Synthesis and antimicrobial activity evaluation of new norfloxacine-azole hybrids
- (2018) Serpil Demirci et al. HETEROCYCLIC COMMUNICATIONS
- N-substituted piperazinyl sarafloxacin derivatives: synthesis and in vitro antibacterial evaluation
- (2018) Ali Asadipour et al. DARU-Journal of Pharmaceutical Sciences
- In vitro activities of a new fluoroquinolone derivative highly active against Chlamydia trachomatis
- (2018) Thi Huyen Vu et al. BIOORGANIC CHEMISTRY
- 4-Quinolone hybrids and their antibacterial activities
- (2017) Yuan-Qiang Hu et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis of novel tetrazole containing hybrid ciprofloxacin and pipemidic acid analogues and preliminary biological evaluation of their antibacterial and antiproliferative activity
- (2017) Kommula Dileep et al. MOLECULAR DIVERSITY
- Photodynamic antimicrobial chemotherapy with cationic phthalocyanines against Escherichia coli planktonic and biofilm cultures
- (2017) Min Li et al. RSC Advances
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