Syntheses of 1 H ‐Indoles, Quinolines, and 6‐Membered Aromatic N ‐Heterocycle‐Fused Scaffolds via Palladium(II)‐Catalyzed Aerobic Dehydrogenation under Alkoxide‐Free Conditions

Manganese(III) Acetate Catalyzed Aerobic Dehydrogenation of Tertiary Indolines, Tetrahydroquinolines and an N ‐Unsubstituted Indoline

(2021) Xiaokang Niu et al.   ADVANCED SYNTHESIS & CATALYSIS

DMSO/t-BuONa/O2-Mediated Aerobic Dehydrogenation of Saturated N-Heterocycles

(2020) Ruchun Yang et al.   JOURNAL OF ORGANIC CHEMISTRY

Role of Indole Scaffolds as Pharmacophores in the Development of Anti-Lung Cancer Agents

(2020) Jyothi Dhuguru et al.   MOLECULES

Aerobic Dehydrogenation of N‐Heterocycles with Grubbs Catalyst: Its Application to Assisted‐Tandem Catalysis to Construct N‐Containing Fused Heteroarenes

(2020) Daichi Kawauchi et al.   CHEMISTRY-A EUROPEAN JOURNAL

Nickel-Catalyzed Dehydrogenation of N-Heterocycles Using Molecular Oxygen

(2020) Sourajit Bera et al.   ORGANIC LETTERS

A Novel Approach to N ‐Tf 2‐Aryl‐2,3‐Dihydroquinolin‐ 4(1 H )‐ones via a Ligand‐Free Pd(II)‐Catalyzed Oxidative Aza‐Michael Cyclization

(2020) Young Min Kim et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Replacement of Stoichiometric DDQ with a Low Potential o-Quinone Catalyst Enabling Aerobic Dehydrogenation of Tertiary Indolines in Pharmaceutical Intermediates

(2019) Bao Li et al.   ORGANIC LETTERS

Potassium tert ‐Butoxide‐Promoted Acceptorless Dehydrogenation of N‐Heterocycles

(2019) Tingting Liu et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of Flavanones via Palladium(II)-Catalyzed One-Pot β-Arylation of Chromanones with Arylboronic Acids

(2019) Hyung-Seok Yoo et al.   JOURNAL OF ORGANIC CHEMISTRY

Visible-Light-Mediated Photocatalytic Aerobic Dehydrogenation of N-heterocycles by Surface-Grafted TiO2 and 4-amino-TEMPO

(2019) Narmina O. Balayeva et al.   ACS Catalysis

Metal-Free Dehydrogenation of N-Heterocycles by Ternary h -BCN Nanosheets with Visible Light

(2018) Meifang Zheng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Double Dehydrogenation of Primary Amines to Nitriles by a Ruthenium Complex Featuring Pyrazole Functionality

(2018) Indranil Dutta et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Acceptorless Dehydrogenation of N-Heterocycles and Secondary Alcohols by Ru(II)-NNC Complexes Bearing a Pyrazoyl-indolyl-pyridine Ligand

(2018) Qingfu Wang et al.   ORGANOMETALLICS

Aerobic oxidative dehydrogenation of N -heterocycles catalyzed by cobalt porphyrin

(2018) Weiyou Zhou et al.   TETRAHEDRON LETTERS

Synthesis of Enones and Enals via Dehydrogenation of Saturated Ketones and Aldehydes

(2018) Gao-Fei Pan et al.   ADVANCED SYNTHESIS & CATALYSIS

Picomole-Scale Real-Time Photoreaction Screening: Discovery of the Visible-Light-Promoted Dehydrogenation of Tetrahydroquinolines under Ambient Conditions

(2016) Suming Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Indoles — A promising scaffold for drug development

(2016) T.V. Sravanthi et al.   EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES

KOtBu: A Privileged Reagent for Electron Transfer Reactions?

(2016) Joshua P. Barham et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A versatile approach to flavones via a one-pot Pd(ii)-catalyzed dehydrogenation/oxidative boron-Heck coupling sequence of chromanones

(2016) Jun Lee et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Metal catalyzed defunctionalization reactions

(2016) Atanu Modak et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Cu-Catalyzed Aerobic Oxidation of Di-tert-butyl Hydrazodicarboxylate to Di-tert-butyl Azodicarboxylate and Its Application on Dehydrogenation of 1,2,3,4-Tetrahydroquinolines under Mild Conditions

(2016) Dahyeon Jung et al.   ORGANIC LETTERS

Palladium-Catalyzed Wacker-Type Oxidation of N-Boc Indoles under Mild Conditions

(2016) Xiao-Yu Zhou et al.   SYNLETT

Palladium-Catalyzed Aerobic Dehydrogenation of Cyclic Hydrocarbons for the Synthesis of Substituted Aromatics and Other Unsaturated Products

(2016) Andrei V. Iosub et al.   ACS Catalysis

External-Ligand-Free Aerobic Oxidation ofN-andC-Containing Cyclic Systems under Pd-Catalyzed Conditions

(2016) Yue Wang et al.   Asian Journal of Organic Chemistry

Rhodium(III)-Catalyzed Selective CH Cyanation of Indolines and Indoles with an Easily Accessible Cyano Source

(2015) Neeraj Kumar Mishra et al.   ADVANCED SYNTHESIS & CATALYSIS

Quinone-Catalyzed Selective Oxidation of Organic Molecules

(2015) Alison E. Wendlandt et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Aerobic Dehydrogenation of Nitrogen Heterocycles Using Heterogeneous Cobalt Oxide Supported on Nitrogen-Doped Carbon

(2015) Andrei V. Iosub et al.   ORGANIC LETTERS

Decarboxylative acylation of indolines with α-keto acids under palladium catalysis: a facile strategy for the synthesis of 7-substituted indoles

(2014) Minyoung Kim et al.   CHEMICAL COMMUNICATIONS

Rings in Drugs

(2014) Richard D. Taylor et al.   JOURNAL OF MEDICINAL CHEMISTRY

A Molecular Iron Catalyst for the Acceptorless Dehydrogenation and Hydrogenation of N-Heterocycles

(2014) Sumit Chakraborty et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper(II)-Catalyzed Three-Component Cascade Annulation of Diaryliodoniums, Nitriles, and Alkynes: A Regioselective Synthesis of Multiply Substituted Quinolines

(2013) Yong Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Acceptorless Dehydrogenation of Nitrogen Heterocycles with a Versatile Iridium Catalyst

(2013) Jianjun Wu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Oxidative Palladium(II)-Catalyzed Dehydrogenative CH/CH Cross-Coupling of 2,3-Substituted Indolines with Arenes at the C7 Position

(2013) Lin-Yu Jiao et al.   CHEMISTRY-A EUROPEAN JOURNAL

Bioinspired Aerobic Oxidation of Secondary Amines and Nitrogen Heterocycles with a Bifunctional Quinone Catalyst

(2013) Alison E. Wendlandt et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Oxidative Palladium(II)-Catalyzed C-7 Alkenylation of Indolines

(2013) Lin-Yu Jiao et al.   ORGANIC LETTERS

Aerobic Synthesis of Substituted Quinoline from Aldehyde and Aniline: Copper-Catalyzed Intermolecular C–H Active and C–C Formative Cyclization

(2013) Rulong Yan et al.   ORGANIC LETTERS

Rhodium(III)-Catalyzed Direct Regioselective Synthesis of 7-Substituted Indoles

(2013) Zengqiang Song et al.   ORGANIC LETTERS

Applications of Acceptorless Dehydrogenation and Related Transformations in Chemical Synthesis

(2013) C. Gunanathan et al.   SCIENCE

Cu(I)/TEMPO-catalyzed aerobic oxidative synthesis of imines directly from primary and secondary amines under ambient and neat conditions

(2013) Bo Huang et al.   TETRAHEDRON LETTERS

Iron-Promoted Tandem Reaction of Anilines with Styrene Oxides via C–C Cleavage for the Synthesis of Quinolines

(2012) Yicheng Zhang et al.   ORGANIC LETTERS

Indole synthesis – something old, something new

(2012) Martyn Inman et al.   Chemical Science

Update 1 of: Synthesis and Functionalization of Indoles Through Palladium-Catalyzed Reactions

(2011) Sandro Cacchi et al.   CHEMICAL REVIEWS

On the “Reverse Gear”Mechanism of the Reversible Dehydrogenation/Hydrogenation of a Nitrogen Heterocycle Catalyzed by a Cp*Ir Complex: A Computational Study

(2011) Haixia Li et al.   ORGANOMETALLICS

Indole synthesis: a review and proposed classification

(2011) Douglass F. Taber et al.   TETRAHEDRON

Total Synthesis of Dictyodendrin A and B

(2010) Kentaro Okano et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Marine Indole Alkaloids: Potential New Drug Leads for the Control of Depression and Anxiety

(2010) Anna J. Kochanowska-Karamyan et al.   CHEMICAL REVIEWS

Luminescence and reactivity of 7-azaindole derivatives and complexes

(2010) Shu-Bin Zhao et al.   CHEMICAL SOCIETY REVIEWS

Total Synthesis of Dictyodendrins A-E

(2010) Hidetoshi Tokuyama et al.   Chemistry-An Asian Journal

Dehydrogenation as a Substrate-Activating Strategy in Homogeneous Transition-Metal Catalysis

(2009) Graham E. Dobereiner et al.   CHEMICAL REVIEWS

Transition-Metal-Free Indirect Friedländer Synthesis of Quinolines from Alcohols†

(2008) Ricardo Martínez et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium catalyzed-dehalogenation of aryl chlorides and bromides using phosphite ligands

(2008) Jeongju Moon et al.   JOURNAL OF ORGANOMETALLIC CHEMISTRY