Journal
GREEN CHEMISTRY
Volume 13, Issue 10, Pages 2723-2726Publisher
ROYAL SOC CHEMISTRY
DOI: 10.1039/c1gc15401j
Keywords
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Funding
- National Mega Project on Major Drug Development [2009ZX09301-014-1]
- NSFC [20872116, 91017005]
- State Key Laboratory of Phytochemistry and Plant Resources in West China [P2010-KF10]
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Metal-free direct amidation of peptidyl thiol esters with alpha-amino acid esters in the presence of bis(trimethylsilyl) acetamide (BSA) has been developed. This general method provides convenient access to N-protected peptides in good yields under mild conditions and demonstrates a high tolerance to functionality.
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