Bismuth compounds in medicinal chemistry

Recent advances in bioinorganic chemistry of bismuth

(2012) Hongyan Li et al.   CURRENT OPINION IN CHEMICAL BIOLOGY

Bismuth(III) Triflate-Based Catalytic Direct Opening of Oleanolic Hydroxy-γ-lactones to Afford 12-Oxo-28-carboxylic Acids

(2011) Jorge A. R. Salvador et al.   ADVANCED SYNTHESIS & CATALYSIS

Anti-CD45 pretargeted radioimmunotherapy using bismuth-213: high rates of complete remission and long-term survival in a mouse myeloid leukemia xenograft model

(2011) J. M. Pagel et al.   BLOOD

Alpha- versus Beta-Particle Radiopeptide Therapy in a Human Prostate Cancer Model (213Bi-DOTA-PESIN and 213Bi-AMBA versus177Lu-DOTA-PESIN)

(2011) D. Wild et al.   CANCER RESEARCH

Total synthesis of a 20-deoxybryostatin

(2011) Anthony P. Green et al.   CHEMICAL COMMUNICATIONS

Applications of bismuth(iii) compounds in organic synthesis

(2011) Jason M. Bothwell et al.   CHEMICAL SOCIETY REVIEWS

Analysis of patient survival in a Phase I trial of systemic targeted α-therapy for metastatic melanoma

(2011) Barry J Allen et al.   Immunotherapy

Synthesis, structural characterization, andin vitroantimicrobial properties of salicylate and pyrazoline complexes of bismuth(III)

(2011) Jeeven S. Solanki et al.   JOURNAL OF COORDINATION CHEMISTRY

Microwave-assisted synthesis, characterization, antimicrobial, and pesticidal activity of bismuth and antimony complexes with coumarin-based ligands

(2011) Latika Dawara et al.   JOURNAL OF COORDINATION CHEMISTRY

Tracking Bismuth Antiulcer Drug Uptake in Single Helicobacter pylori Cells

(2011) Cheuk-Nam Tsang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Helicobacter pylori eradication with a capsule containing bismuth subcitrate potassium, metronidazole, and tetracycline given with omeprazole versus clarithromycin-based triple therapy: a randomised, open-label, non-inferiority, phase 3 trial

(2011) Peter Malfertheiner et al.   LANCET

Bismuth(III) Reagents in Steroid and Terpene Chemistry

(2011) Jorge A. R. Salvador et al.   MOLECULES

Allobetulin and Its Derivatives: Synthesis and Biological Activity

(2011) Wim Dehaen et al.   MOLECULES

An overview of targeted alpha therapy

(2011) Young-Seung Kim et al.   TUMOR BIOLOGY

NO-releasing esters show carbonic anhydrase inhibitory action against human isoforms I and II

(2010) Deniz Ekinci et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis of new cis-fused tetrahydrochromeno[4,3-b]quinolines and their antiproliferative activity studies against MDA-MB-231 and MCF-7 breast cancer cell lines

(2010) K. Nagaiah et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Conventional and pretargeted radioimmunotherapy using bismuth-213 to target and treat non-Hodgkin lymphomas expressing CD20: a preclinical model toward optimal consolidation therapy to eradicate minimal residual disease

(2010) S. I. Park et al.   BLOOD

Improved efficacy of α-particle-targeted radiation therapy

(2010) Diane E. Milenic et al.   CANCER

Rapid assembly of gp120 oligosaccharide moieties via one-pot glycosidation–deprotection sequences

(2010) Antonello Pastore et al.   CARBOHYDRATE RESEARCH

Sequential Cytarabine and  -Particle Immunotherapy with Bismuth-213-Lintuzumab (HuM195) for Acute Myeloid Leukemia

(2010) T. L. Rosenblat et al.   CLINICAL CANCER RESEARCH

Tacrine Derivatives and Alzheimers Disease

(2010) V. Tumiatti et al.   CURRENT MEDICINAL CHEMISTRY

Bismuth(iii) complexes derived from non-steroidal anti-inflammatory drugs and their activity against Helicobacter pylori

(2010) Philip C. Andrews et al.   DALTON TRANSACTIONS

Structural and solution studies of phenylbismuth(III) sulfonate complexes and their activity against Helicobacter pylori

(2010) Philip C. Andrews et al.   DALTON TRANSACTIONS

Bismuth heterocycles based on a diphenyl sulfone scaffold: Synthesis and substituent effect on the antifungal activity against Saccharomyces cerevisiae

(2010) Toshihiro Murafuji et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

177Lu-immunotherapy of experimental peritoneal carcinomatosis shows comparable effectiveness to 213Bi-immunotherapy, but causes toxicity not observed with 213Bi

(2010) Christof Seidl et al.   EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING

Targeted alpha-radionuclide therapy of functionally critically located gliomas with 213Bi-DOTA-[Thi8,Met(O2)11]-substance P: a pilot trial

(2010) D. Cordier et al.   EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING

Attenuation of Pseudomonas aeruginosa virulence factors and biofilms by co-encapsulation of bismuth-ethanedithiol with tobramycin in liposomes

(2010) M. Alipour et al.   JOURNAL OF ANTIMICROBIAL CHEMOTHERAPY

Anti-Leishmanial activity of homo- and heteroleptic bismuth(III) carboxylates

(2010) Philip C. Andrews et al.   JOURNAL OF INORGANIC BIOCHEMISTRY

Bismuth subcarbonate nanoparticles fabricated by water-in-oil microemulsion-assisted hydrothermal process exhibit anti-Helicobacter pylori properties

(2010) Rong Chen et al.   MATERIALS RESEARCH BULLETIN

Green bismuth

(2010) Ram Mohan   Nature Chemistry

A Bismuth(III)-Catalyzed Friedel−Crafts Cyclization and Stereocontrolled Organocatalytic Approach to (−)-Platensimycin

(2010) Stanley T.-C. Eey et al.   ORGANIC LETTERS

A zinc-binding site by negative selection induces metallodrug susceptibility in an essential chaperonin

(2010) S. Cun et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Direct Catalytic Benzylation of Hydroxycoumarin - Efficient Synthesis of Warfarin Derivatives and Analogues

(2010) Magnus Rueping et al.   SYNLETT

Synthesis, Characterization, and Antimicrobial Evaluation of Sulfonamides ContainingN-Acyl Moieties Catalyzed by Bismuth(III) Salts Under Both Solvent and Solvent-Free Conditions

(2010) Hadi Adibi et al.   SYNTHETIC COMMUNICATIONS

Bismuth(III) Triflate: A Safe and Easily Handled Precursor for Triflic Acid: Application to the Esterification Reaction

(2010) Franciane Ho A Kwie et al.   SYNTHETIC COMMUNICATIONS

Efficient trans-diaxial hydroxylation of Δ5-steroids

(2010) João F.S. Carvalho et al.   TETRAHEDRON

Metalloantibiotics: Synthesis, characterization and antimicrobial evaluation of bismuth-fluoroquinolone complexes against Helicobacter pylori

(2009) Anwar Shaikh et al.   ACTA PHARMACEUTICA

In vitro inhibition of human erythrocyte glutathione reductase by some new organic nitrates

(2009) Murat Şentürk et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Recent Advances of Bismuth(III) Salts in Organic Chemistry: Application to the Synthesis of Heterocycles of Pharmaceutical Interest

(2009) Jorge Salvador et al.   CURRENT ORGANIC SYNTHESIS

Bismuth(iii) 5-sulfosalicylate complexes: structure, solubility and activity against Helicobacter pylori

(2009) Philip C. Andrews et al.   DALTON TRANSACTIONS

One-Pot Catalytic Glycosidation/Fmoc Removal - An Iterable Sequence for Straightforward Assembly of Oligosaccharides Related to HIV gp120

(2009) Antonello Pastore et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

The role of sulfamide derivatives in medicinal chemistry: a patent review (2006 – 2008)

(2009) Allen B Reitz et al.   EXPERT OPINION ON THERAPEUTIC PATENTS

Bismuth–thiol incorporation enhances biological activities of liposomal tobramycin against bacterial biofilm and quorum sensing molecules production by Pseudomonas aeruginosa

(2009) Majed Halwani et al.   INTERNATIONAL JOURNAL OF PHARMACEUTICS

Differential gene expression triggered by highly cytotoxic α-Emitter-immunoconjugates in gastric cancer cells

(2009) Christof Seidl et al.   INVESTIGATIONAL NEW DRUGS

Antioxidant Oligostilbenoids from the Stem Wood ofHopea hainanensis

(2009) Hui-Ming Ge et al.   JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY

Bismuth(III) Triflate-Catalyzed Direct Conversion of Corticosteroids into Highly Functionalized 17-Ketosteroids by Cleavage of theC17-Dihydroxyacetone Side Chain

(2009) Rui M. A. Pinto et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis, structure, and in vitro antiproliferative activity of cyclic hypervalent organobismuth(III) chlorides and their triphenylgermylpropionate derivatives

(2009) Xiao-Wen Zhang et al.   JOURNAL OF ORGANOMETALLIC CHEMISTRY

Heterocyclic Organobismuth(III) Compound Targets Tubulin to Induce G2/M Arrest in HeLa Cells

(2009) Katsuya Iuchi et al.   JOURNAL OF PHARMACOLOGICAL SCIENCES

Recent Advances of Bismuth(III) Salts in Organic Chemistry: Application to the Synthesis of Aliphatics, Alicyclics, Aromatics, Amino Acids and Peptides, Terpenes and Steroids of Pharmaceutical Interest

(2009) Jorge Salvador et al.   MINI-REVIEWS IN ORGANIC CHEMISTRY

A versatile approach to oligostilbenoid natural products – synthesis of permethylated analogues of viniferifuran, malibatol A, and shoreaphenol

(2009) Ikyon Kim et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Multicatalytic Synthesis of Complex Tetrahydrofurans Involving Bismuth(III) Triflate Catalyzed Intramolecular Hydroalkoxylation of Unactivated Olefins

(2009) Brendan D. Kelly et al.   ORGANIC LETTERS

Versatile method for the synthesis of 4-substituted 6-methyl-3-oxabicyclo[3.3.1]non-6-ene-1-methanol derivatives: Prins-type cyclization reaction catalyzed by hafnium triflate

(2009) Masayuki Nakamura et al.   TETRAHEDRON LETTERS

Heterocyclic organobismuth(III) induces apoptosis of human promyelocytic leukemic cells through activation of caspases and mitochondrial perturbation

(2008) Katsuya Iuchi et al.   BIOCHEMICAL PHARMACOLOGY

Synthesis and cytotoxicity of methyl-and methoxy-substituted metal 8-quinolinethiolates

(2008) E. Lukevics et al.   Chemistry of Heterocyclic Compounds

Recent Advances in Bismuth-Catalyzed Organic Synthesis

(2008) Ruimao Hua   CURRENT ORGANIC SYNTHESIS

Synthesis of the Mannopeptimycin Disaccharide and Its Conjugation with 4-Alkylidene-β-lactams

(2008) Matteo Adinolfi et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of New β-Hydroxy Nitrate Esters as Potential Glycomimetics or Vasodilators

(2008) Huseyin Cavdar et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Liposomal bismuth-ethanedithiol formulation enhances antimicrobial activity of tobramycin

(2008) Majed Halwani et al.   INTERNATIONAL JOURNAL OF PHARMACEUTICS

Synthesis, spectral study and antimicrobial activity of bismuth(III) 3(2′-hydroxyphenyl)-5-(4-substituted phenyl) pyrazolinates

(2008) Jeeven S. Solanki et al.   JOURNAL OF COORDINATION CHEMISTRY

In vitro antileukemia, antibacterial and antifungal activities of some 3d metal complexes: Chemical synthesis and structure – activity relationships

(2008) Aurelian Gulea et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Outstanding plasmodicidal properties within a small panel of metallic compounds: Hints for the development of new metal-based antimalarials

(2008) Chiara Gabbiani et al.   JOURNAL OF INORGANIC BIOCHEMISTRY

A Route to 1,4-Disubstituted Aromatics and Its Application to the Synthesis of the Antibiotic Culpin

(2008) Rajesh Sunasee et al.   JOURNAL OF ORGANIC CHEMISTRY

Sequential One-Pot Glycosidations Catalytically Promoted: Unprecedented Strategy in Oligosaccharide Synthesis for the Straightforward Assemblage of the Antitumor PI-88 Pentasaccharide

(2008) Silvia Valerio et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of 5-Arylidene Barbiturates: A Novel Class of DPPH Radical Scavengers

(2008) Khalid M. Khan et al.   Letters in Drug Design & Discovery

An Efficient Synthesis of 2,3-Diaryl-2-azabicyclooctanones Via BiCl3- Catalysed Three-Component aza Diels-Alder Reaction

(2008) Luis S. et al.   LETTERS IN ORGANIC CHEMISTRY

Bismuth triflate-catalyzed Wagner-Meerwein rearrangement in terpenes. Application to the synthesis of the 18α-oleanane core and A-neo-18α-oleanene compounds from lupanes

(2008) Jorge A. R. Salvador et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Bismuth Chloride Mediated Synthesis, Antimicrobial, and Anti-Inflammatory Activities of New 4-Aryl-2-Amino Thiazoles

(2008) T. Giridhar et al.   PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS

Targeting the carbohydrates on HIV-1: Interaction of oligomannose dendrons with human monoclonal antibody 2G12 and DC-SIGN

(2008) S.-K. Wang et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

How corticosteroids control inflammation: Quintiles Prize Lecture 2005

(2006) Peter J Barnes   BRITISH JOURNAL OF PHARMACOLOGY