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Title
Inhibitors of cathepsin K: a patent review (2004 – 2010)
Authors
Keywords
-
Journal
EXPERT OPINION ON THERAPEUTIC PATENTS
Volume 21, Issue 10, Pages 1611-1629
Publisher
Informa Healthcare
Online
2011-09-17
DOI
10.1517/13543776.2011.616283
References
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Related references
Note: Only part of the references are listed.- Safety and efficacy of the cathepsin K inhibitor ONO-5334 in postmenopausal osteoporosis: The OCEAN study
- (2011) Richard Eastell et al. JOURNAL OF BONE AND MINERAL RESEARCH
- Conformational flexibility and allosteric regulation of cathepsin K
- (2010) Marko Novinec et al. BIOCHEMICAL JOURNAL
- Optimisation of 2-cyano-pyrimidine inhibitors of cathepsin K: Improving selectivity over hERG
- (2010) Zoran Rankovic et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Orally Bioavailable Cathepsin K Inhibitors with Pyrrolopyrimidine Scaffold
- (2010) Naoki Teno et al. CURRENT TOPICS IN MEDICINAL CHEMISTRY
- Development of Nitrile-Based Peptidic Inhibitors of Cysteine Cathepsins
- (2010) Maxim Frizler et al. CURRENT TOPICS IN MEDICINAL CHEMISTRY
- Cathepsin K inhibitors prevent bone loss in estrogen-deficient rabbits
- (2010) Brenda L Pennypacker et al. JOURNAL OF BONE AND MINERAL RESEARCH
- Odanacatib in the treatment of postmenopausal women with low bone mineral density: Three-year continued therapy and resolution of effect
- (2010) John A Eisman et al. JOURNAL OF BONE AND MINERAL RESEARCH
- The discovery of MK-0674, an orally bioavailable cathepsin K inhibitor
- (2009) Elise Isabel et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Pharmacological Promiscuity: Dependence on Compound Properties and Target Specificity in a Set of Recent Roche Compounds
- (2009) Jens-Uwe Peters et al. ChemMedChem
- Cathepsin K inhibitors for osteoporosis and potential off-target effects
- (2009) Dieter Brömme et al. EXPERT OPINION ON INVESTIGATIONAL DRUGS
- Covalent Modifiers: An Orthogonal Approach to Drug Design
- (2009) Michele H. Potashman et al. JOURNAL OF MEDICINAL CHEMISTRY
- Deficiency and Inhibition of Cathepsin K Reduce Body Weight Gain and Increase Glucose Metabolism in Mice
- (2008) Min Yang et al. ARTERIOSCLEROSIS THROMBOSIS AND VASCULAR BIOLOGY
- The discovery of odanacatib (MK-0822), a selective inhibitor of cathepsin K
- (2008) Jacques Yves Gauthier et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Investigation of ketone warheads as alternatives to the nitrile for preparation of potent and selective cathepsin K inhibitors
- (2008) Michael J. Boyd et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Cysteine cathepsin S as an immunomodulatory target: present and future trends
- (2008) Suman Gupta et al. EXPERT OPINION ON THERAPEUTIC TARGETS
- Discovery of Orally Bioavailable Cathepsin S Inhibitors for the Reversal of Neuropathic Pain
- (2008) Osamu Irie et al. JOURNAL OF MEDICINAL CHEMISTRY
- Identification of a Nonbasic, Nitrile-Containing Cathepsin K Inhibitor (MK-1256) that is Efficacious in a Monkey Model of Osteoporosis
- (2008) Jöel Robichaud et al. JOURNAL OF MEDICINAL CHEMISTRY
- Beyond Picomolar Affinities: Quantitative Aspects of Noncovalent and Covalent Binding of Drugs to Proteins
- (2008) Adam J. T. Smith et al. JOURNAL OF MEDICINAL CHEMISTRY
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