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The Inhibition by Levocetirizine and Fexofenadine of the Histamine-induced Wheal and Flare Response in Healthy Caucasian and Japanese Volunteers

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Safety considerations in the management of allergic diseases: focus on antihistamines

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Improving the prediction of the brain disposition for orally administered drugs using BDDCS

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Comparison of the sedating effects of levocetirizine and cetirizine: a randomized, double-blind, placebo-controlled trial

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Positron emission tomography evaluation of sedative properties of antihistamines

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Brain histamine H1 receptor occupancy of loratadine measured by positron emission topography: comparison of H1 receptor occupancy and proportional impairment ratio

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(2010) M. K. Church et al.   ALLERGY

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Transporter-Mediated Efflux Influences CNS Side Effects: ABCB1, from Antitarget to Target

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Dose dependency of brain histamine H1 receptor occupancy following oral administration of cetirizine hydrochloride measured using PET with [11C]doxepin

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Brain histamine H1receptor occupancy of orally administered antihistamines, bepotastine and diphenhydramine, measured by PET with11C-doxepin

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Non-Interventional Study Comparing Treatment Satisfaction in Patients Treated with Antihistamines

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Physicochemical, Pharmacological and Pharmacokinetic Properties of the Zwitterionic Antihistamines Cetirizine and Levocetirizine

(2008) Chen Chen   CURRENT MEDICINAL CHEMISTRY

Sedation and antihistamines: an update. Review of inter-drug differences using proportional impairment ratios

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Neuroimaging of histamine H1-receptor occupancy in human brain by positron emission tomography (PET): A comparative study of ebastine, a second-generation antihistamine, and (+)-chlorpheniramine, a classical antihistamine

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