Extending the Scope of the Aza-Fischer Synthesis of 4- and 6-Azaindoles

Synthesis of 2,5-Disubstituted 6-Azaindoles from Substituted Aziridines via Intramolecular Cyclization

(2012) Hogyu Lee et al.   ORGANIC LETTERS

Synthesis and antimycobacterial activities of non-purine analogs of 6-aryl-9-benzylpurines: Imidazopyridines, pyrrolopyridines, benzimidazoles, and indoles

(2011) Abhijit Datta Khoje et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Design and synthesis of 1-(2-alkanamidoethyl)-6-methoxy-7-azaindole derivatives as potent melatonin agonists

(2011) Matthieu Jeanty et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Discovery and optimization of indoles and 7-azaindoles as Rho kinase (ROCK) inhibitors (part-I)

(2011) Sarwat Chowdhury et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

A facile, water mediated, microwave-assisted synthesis of 4,6-diaryl-2,3,3a,4-tetrahydro-1H-pyrido[3,2,1-jk]carbazoles by a domino Fischer indole reaction–intramolecular cyclization sequence

(2011) Selvam Chitra et al.   GREEN CHEMISTRY

One-pot-one-step, microwave-assisted Fischer indole synthesis

(2011) Evelyn Cuevas Creencia et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Two-Step Route to Indoles and Analogues from Haloarenes: A Variation on the Fischer Indole Synthesis

(2011) Martyn Inman et al.   JOURNAL OF ORGANIC CHEMISTRY

Blue-luminescent 5-(3-indolyl)oxazoles via microwave-assisted three-component coupling–cycloisomerization–Fischer indole synthesis

(2011) Oliver Grotkopp et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

A direct copper-catalyzed route to pyrrolo-fused heterocycles from boronic acids

(2011) Ramsay E. Beveridge et al.   TETRAHEDRON LETTERS

Synthesis and biological evaluation of 2,3-bis(het)aryl-4-azaindole derivatives as protein kinase inhibitors

(2011) Frédéric Pin et al.   MedChemComm

Microwave-accelerated Dimroth rearrangement for the synthesis of 4-anilino-6-nitroquinazolines. Application to an efficient synthesis of a microtubule destabilizing agent

(2010) Alicia Foucourt et al.   TETRAHEDRON

Strategies for Innovation in Multicomponent Reaction Design

(2009) Bruce Ganem   ACCOUNTS OF CHEMICAL RESEARCH

New insights into homopiperazine-based 5-HT1A/5-HT7R ligands: synthesis and biological evaluation

(2009) Eduard Badarau et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Discovery of Novel Antileishmanial Agents in an Attempt to Synthesize Pentamidine−Aplysinopsin Hybrid Molecule

(2009) Sharad Porwal et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of 4- and 6-Azaindoles via the Fischer Reaction

(2009) Matthieu Jeanty et al.   ORGANIC LETTERS

Synthesis of 5,7-Dichloro-6-azaindoles and Functionalization via a Highly Selective Lithium-Chlorine Exchange

(2009) Nicolas Lachance et al.   SYNTHESIS-STUTTGART

Highly functionalized 7-azaindoles as selective PPARγ modulators

(2008) Sheryl D. Debenham et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis of C3-Substituted 4-Azaindoles: An Easy Access to 4-Azamelatonin and Protected 4-Azatryptophan

(2008) Matthieu Jeanty et al.   JOURNAL OF ORGANIC CHEMISTRY