Azide- and Alkyne-Derivatised α-Amino Acids

Letters

(2016)   CHEMICAL & ENGINEERING NEWS

Sensitivities of Some Imidazole-1-sulfonyl Azide Salts

(2012) Niko Fischer et al.   JOURNAL OF ORGANIC CHEMISTRY

Click Strategies for Single-Molecule Protein Fluorescence

(2012) Sigrid Milles et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

New β-Strand Templates Constrained by Huisgen Cycloaddition

(2012) Ashok D. Pehere et al.   ORGANIC LETTERS

Modular Assembly of Macrocyclic Organo-Peptide Hybrids Using Synthetic and Genetically Encoded Precursors

(2011) Jessica M. Smith et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Maintaining Biological Activity by Using Triazoles as Disufide Bond Mimetics

(2011) Kai Holland-Nell et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Access to Biomolecular Assemblies through One-Pot Triple Orthogonal Chemoselective Ligations

(2011) Mathieu Galibert et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis ofC-Linked Triazole-Containing AFGP Analogues and Their Ability to Inhibit Ice Recrystallization

(2011) Chantelle J. Capicciotti et al.   BIOCONJUGATE CHEMISTRY

Clickable Enzyme-Linked Immunosorbent Assay

(2011) Luiz A. Canalle et al.   BIOMACROMOLECULES

A readily synthesized cyclic pyrrolysine analogue for site-specific protein “click” labeling

(2011) Ziyang Hao et al.   CHEMICAL COMMUNICATIONS

Fluorophore-labeled, Peptide-based Glycoclusters: Synthesis, Binding Properties for Lectins, and Detection of Carbohydrate-Binding Proteins in Cells

(2011) Xizhe Tian et al.   Chemistry-An Asian Journal

Identification of pentacyclic triterpenes derivatives as potent inhibitors against glycogen phosphorylase based on 3D-QSAR studies

(2011) Zhongjie Liang et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

1,2,3-Triazoles in Peptidomimetic Chemistry

(2011) Daniel Sejer Pedersen et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Functionalization of Fe3O4 magnetic nanoparticles for organocatalytic Michael reactions

(2011) Paola Riente et al.   JOURNAL OF MATERIALS CHEMISTRY

Design of Triazole-Stapled BCL9 α-Helical Peptides to Target the β-Catenin/B-Cell CLL/lymphoma 9 (BCL9) Protein–Protein Interaction

(2011) Steven A. Kawamoto et al.   JOURNAL OF MEDICINAL CHEMISTRY

Stapling of a 310-Helix with Click Chemistry

(2011) Øyvind Jacobsen et al.   JOURNAL OF ORGANIC CHEMISTRY

An Efficient, Inexpensive, and Shelf-Stable Diazotransfer Reagent: Imidazole-1-sulfonyl Azide Hydrochloride

(2011) Ethan D. Goddard-Borger et al.   ORGANIC LETTERS

CuAAC Macrocyclization: High Intramolecular Selectivity through the Use of Copper–Tris(triazole) Ligand Complexes

(2011) Gagan Chouhan et al.   ORGANIC LETTERS

Amino Triazolo Diazepines (Ata) as Constrained Histidine Mimics

(2011) Koen Buysse et al.   ORGANIC LETTERS

Nonafluorobutanesulfonyl Azide: A Shelf-Stable Diazo Transfer Reagent for the Synthesis of Azides from Primary Amines

(2010) José Ramón Suárez et al.   ADVANCED SYNTHESIS & CATALYSIS

Azidohomoalanine: A Conformationally Sensitive IR Probe of Protein Folding, Protein Structure, and Electrostatics

(2010) Humeyra Taskent-Sezgin et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

1,2,3-Triazolyl amino acids as AMPA receptor ligands

(2010) N.J. Stanley et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Construction of 6-Triazole-Linked Mannopyranosyl Serine and Threonine as Novel Sugar Amino Acid Mimics

(2010) Qiong Deng et al.   BULLETIN OF THE KOREAN CHEMICAL SOCIETY

A simple quick route to fullerene amino acid derivatives

(2010) T. Amanda Strom et al.   CHEMICAL COMMUNICATIONS

End-stapled homo and hetero collagen triple helices: a click chemistry approach

(2010) Cillian Byrne et al.   CHEMICAL COMMUNICATIONS

In situ click chemistry: probing the binding landscapes of biological molecules

(2010) Sreeman K. Mamidyala et al.   CHEMICAL SOCIETY REVIEWS

Tricks with clicks: modification of peptidomimetic oligomers via copper-catalyzed azide-alkyne [3 + 2] cycloaddition

(2010) Justin M. Holub et al.   CHEMICAL SOCIETY REVIEWS

Click chemistry with DNA

(2010) Afaf H. El-Sagheer et al.   CHEMICAL SOCIETY REVIEWS

Cu-free click cycloaddition reactions in chemical biology

(2010) John C. Jewett et al.   CHEMICAL SOCIETY REVIEWS

Protein-Inorganic Array Construction: Design and Synthesis of the Building Blocks

(2010) Niculina D. Bogdan et al.   CHEMISTRY-A EUROPEAN JOURNAL

Efficient Access to New Chemical Space Through Flow-Construction of Druglike Macrocycles Through Copper-Surface-Catalyzed Azide-Alkyne Cycloaddition Reactions

(2010) Andrew R. Bogdan et al.   CHEMISTRY-A EUROPEAN JOURNAL

Click on silica: systematic immobilization of Co(ii) Schiff bases to the mesoporous silica via click reaction and their catalytic activity for aerobic oxidation of alcohols

(2010) Bharat S. Rana et al.   DALTON TRANSACTIONS

Solid-Phase Synthesis of Aza-Kahalalide F Analogues: (2R,3R)-2-Amino-3-azidobutanoic Acid as Precursor of the Aza-Threonine

(2010) Irene Izzo et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

2′-Linking of Lipids and Other Functions to Uridine through 1,2,3-Triazoles and Membrane Anchoring of the Amphiphilic Products

(2010) Oliver Kaczmarek et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Functional Characterization of the Cyclomarin/Cyclomarazine Prenyltransferase CymD Directs the Biosynthesis of Unnatural Cyclic Peptides⊥

(2010) Andrew W. Schultz et al.   JOURNAL OF NATURAL PRODUCTS

Synthesis ofC-Propargylic Esters of N-Protected Amino Acids and Peptides

(2010) Sean P. Bew et al.   JOURNAL OF ORGANIC CHEMISTRY

Benzotriazol-1-yl-sulfonyl Azide for Diazotransfer and Preparation of Azidoacylbenzotriazoles

(2010) Alan R. Katritzky et al.   JOURNAL OF ORGANIC CHEMISTRY

Photoinduced Addition of Glycosyl Thiols to Alkynyl Peptides: Use of Free-Radical Thiol−Yne Coupling for Post-Translational Double-Glycosylation of Peptides

(2010) Mauro Lo Conte et al.   JOURNAL OF ORGANIC CHEMISTRY

Bioorthogonal Chemical Reporters for Monitoring Protein Acetylation

(2010) Yu-Ying Yang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Universal Peptidomimetics

(2010) Eunhwa Ko et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Facile Synthesis of Glycopolypeptides by Combination of Ring-Opening Polymerization of an Alkyne-Substituted N-carboxyanhydride and Click “Glycosylation”

(2010) Chunsheng Xiao et al.   MACROMOLECULAR RAPID COMMUNICATIONS

A concise and scalable route to L-azidohomoalanine

(2010) Stefanie Roth et al.   Nature Protocols

Neoglycopeptides through direct functionalization of cysteine

(2010) Christine Vala et al.   TETRAHEDRON LETTERS

Bivalent Peptidomimetic Ligands of TrkC Are Biased Agonists and Selectively Induce Neuritogenesis or Potentiate Neurotrophin-3 Trophic Signals

(2009) Dianjun Chen et al.   ACS Chemical Biology

Development of Selective Bisubstrate-Based Inhibitors Against Protein Kinase C (PKC) Isozymes By Using Dynamic Peptide Microarrays

(2009) Alex J. Poot et al.   CHEMBIOCHEM

Activity-Based Probes for Monitoring Postproline Protease Activity

(2009) Eduard Sabidó et al.   CHEMBIOCHEM

A Click Approach to Structurally Diverse Conjugates Containing a Central Di-1,2,3-triazole Metal Chelate

(2009) Thomas L. Mindt et al.   ChemMedChem

Microwave-Assisted Intramolecular Huisgen Cycloaddition of Azido Alkynes Derived from α-Amino Acids

(2009) Evita Balducci et al.   JOURNAL OF ORGANIC CHEMISTRY

Genetic Encoding and Labeling of Aliphatic Azides and Alkynes in Recombinant Proteinsviaa Pyrrolysyl-tRNA Synthetase/tRNACUAPair and Click Chemistry

(2009) Duy P. Nguyen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of Fish Antifreeze Neoglycopeptides Using Microwave-Assisted “Click Chemistry”

(2009) Nicole Miller et al.   ORGANIC LETTERS

A One-Pot Approach to Neoglycopeptides using Orthogonal Native Chemical Ligation and Click Chemistry

(2009) Dong Jun Lee et al.   ORGANIC LETTERS

Synthesis of crosslinking amino acids by click chemistry

(2009) Chun Li et al.   TETRAHEDRON

“Click-to-Chelate”: In Vitro and In Vivo Comparison of a99mTc(CO)3-Labeled N(τ)-Histidine Folate Derivative with Its Isostructural, Clicked 1,2,3-Triazole Analogue

(2008) Thomas L. Mindt et al.   BIOCONJUGATE CHEMISTRY

Synthesis and evaluation of homodimeric GnRHR antagonists having a rigid bis-propargylated benzene core

(2008) Kimberly M. Bonger et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Application of Metal‐Free Triazole Formation in the Synthesis of Cyclic RGD–DTPA Conjugates

(2008) Sander S. van Berkel et al.   CHEMBIOCHEM

“Click‐to‐Chelate”: Design and Incorporation of Triazole‐Containing Metal‐Chelating Systems into Biomolecules of Diagnostic and Therapeutic Interest

(2008) Harriet Struthers et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthetic Receptors for the Differentiation of Phosphorylated Peptides with Nanomolar Affinities

(2008) Andreas Grauer et al.   CHEMISTRY-A EUROPEAN JOURNAL

Immobilization of Cobalt(II) Schiff Base Complexes on Polystyrene Resin and a Study of Their Catalytic Activity for the Aerobic Oxidation of Alcohols

(2008) Suman Jain et al.   ChemSusChem

Nα-Fmoc-Protected ω-Azido- and ω-Alkynyl-L-amino Acids as Building Blocks for the Synthesis of “Clickable” Peptides

(2008) Alexandra Le Chevalier Isaad et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Strategies for the Solid-Phase Diversification of Poly-l-proline-Type II Peptide Mimic Scaffolds and Peptide Scaffolds Through Guanidinylation

(2008) Stevenson Flemer et al.   JOURNAL OF ORGANIC CHEMISTRY

Preparation ofNG-Substitutedl-Arginine Analogues Suitable for Solid Phase Peptide Synthesis

(2008) Nathaniel I. Martin et al.   JOURNAL OF ORGANIC CHEMISTRY

β-Azidoalanine as an IR Probe: Application to Amyloid Aβ(16-22) Aggregation

(2008) Kwang-Im Oh et al.   JOURNAL OF PHYSICAL CHEMISTRY B