Benzocyclobutane, Benzocycloheptane and Heptene Derivatives as Melatonin Agonists and Antagonists

New melatonin (MT1/MT2) ligands: Design and synthesis of (8,9-dihydro-7H-furo[3,2-f]chromen-1-yl) derivatives

(2014) Elodie Landagaray et al.   BIOORGANIC & MEDICINAL CHEMISTRY

A Molecular and Chemical Perspective in Defining Melatonin Receptor Subtype Selectivity

(2013) King Chan et al.   INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES

MT1 and MT2 Melatonin Receptors: Ligands, Models, Oligomers, and Therapeutic Potential

(2013) Darius. P. Zlotos et al.   JOURNAL OF MEDICINAL CHEMISTRY

Investigational Selective Melatoninergic Ligands for Receptor Subtype MT2

(2013) Ning Wan et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

Upcoming market catalysts in Q4 2013

(2013) Stacey Fong   NATURE REVIEWS DRUG DISCOVERY

Design, synthesis, and pharmacological effects of structurally simple ligands for MT1 and MT2 melatonin receptors

(2010) Alessia Carocci et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis of substituted N-[3-(3-methoxyphenyl)propyl] amides as highly potent MT2-selective melatonin ligands

(2010) Yueqing Hu et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

International Union of Basic and Clinical Pharmacology. LXXV. Nomenclature, Classification, and Pharmacology of G Protein-Coupled Melatonin Receptors

(2010) M. L. Dubocovich et al.   PHARMACOLOGICAL REVIEWS

3-Methoxylphenylpropyl amides as novel receptor subtype-selective melatoninergic ligands: characterization of physicochemical and pharmacokinetic properties

(2010) Jing Zhu et al.   XENOBIOTICA

Discovery of TAK-875: A Potent, Selective, and Orally Bioavailable GPR40 Agonist

(2010) Nobuyuki Negoro et al.   ACS Medicinal Chemistry Letters

Melatonin Receptor Antagonist Luzindole: A Facile New Synthesis

(2008) Andrew Tsotinis et al.   LETTERS IN ORGANIC CHEMISTRY