Activity-Based Probes for the Study of Proteases: Recent Advances and Developments
Published 2012 View Full Article
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Title
Activity-Based Probes for the Study of Proteases: Recent Advances and Developments
Authors
Keywords
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Journal
ChemMedChem
Volume 7, Issue 7, Pages 1146-1159
Publisher
Wiley
Online
2012-03-19
DOI
10.1002/cmdc.201200057
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- Cleavable linkers in chemical biology
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- (2011) Laura E Edgington et al. CURRENT OPINION IN CHEMICAL BIOLOGY
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- A Substrate-Free Activity-Based Protein Profiling Screen for the Discovery of Selective PREPL Inhibitors
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- (2011) Katsunori Tsuboi et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- A Peptide Aldehyde Microarray for High-Throughput Profiling of Cellular Events
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- Multicolor, One- and Two-Photon Imaging of Enzymatic Activities in Live Cells with Fluorescently Quenched Activity-Based Probes (qABPs)
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- Academic cross-fertilization by public screening yields a remarkable class of protein phosphatase methylesterase-1 inhibitors
- (2011) D. A. Bachovchin et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- Chemical Probes of Surface Layer Biogenesis inClostridium difficile
- (2010) T. H. Tam Dang et al. ACS Chemical Biology
- A Cleavable Linker Based on the Levulinoyl Ester for Activity-Based Protein Profiling
- (2010) Paul P. Geurink et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
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- Two-Step Labeling of Endogenous Enzymatic Activities by Diels-Alder Ligation
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- Cu-free click cycloaddition reactions in chemical biology
- (2010) John C. Jewett et al. CHEMICAL SOCIETY REVIEWS
- Comparative Analysis of Cleavable Azobenzene-Based Affinity Tags for Bioorthogonal Chemical Proteomics
- (2010) Yu-Ying Yang et al. CHEMISTRY & BIOLOGY
- Cleavable Biotin Probes for Labeling of Biomolecules via Azide−Alkyne Cycloaddition
- (2010) Janek Szychowski et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Emerging principles in protease-based drug discovery
- (2010) Marcin Drag et al. NATURE REVIEWS DRUG DISCOVERY
- Fluorescence quenched quinone methide based activity probes – a cautionary tale
- (2010) Jonathan D. Sellars et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Superfamily-wide portrait of serine hydrolase inhibition achieved by library-versus-library screening
- (2010) D. A. Bachovchin et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
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- (2009) Ulrik Hillaert et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Syringolin A Selectively Labels the 20 S Proteasome in Murine EL4 and Wild-Type and Bortezomib-Adapted Leukaemic Cell Lines
- (2009) Jérôme Clerc et al. CHEMBIOCHEM
- Activity-Based Probes for Monitoring Postproline Protease Activity
- (2009) Eduard Sabidó et al. CHEMBIOCHEM
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- (2009) Adriaan W. Tuin et al. CHEMICAL RESEARCH IN TOXICOLOGY
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