Development of Isoxazoline-Containing Peptidomimetics as Dual αvβ3 and α5β1 Integrin Ligands

Advances in Imaging

(2011) Klaudia U. Hunter et al.   CANCER JOURNAL

A Glimpse of the Future

(2011) Michelle Alonso-Basanta et al.   CANCER JOURNAL

Integrin αvβ3-targeted gold nanoshells augment tumor vasculature-specific imaging and therapy

(2011) Huan Xie et al.   International Journal of Nanomedicine

Integrin  5 1 facilitates cancer cell invasion through enhanced contractile forces

(2011) C. T. Mierke et al.   JOURNAL OF CELL SCIENCE

PET of  v 3-Integrin and  v 5-Integrin Expression with 18F-Fluciclatide for Assessment of Response to Targeted Therapy: Ready for Prime Time?

(2011) A. J. Beer et al.   JOURNAL OF NUCLEAR MEDICINE

The tail of integrin activation

(2011) Nicholas J. Anthis et al.   TRENDS IN BIOCHEMICAL SCIENCES

Inhibition of HIV-1 Replication by Isoxazolidine and Isoxazole Sulfonamides

(2010) Belinda Loh et al.   Chemical Biology & Drug Design

Total Syntheses of Tubulysins

(2010) Taku Shibue et al.   CHEMISTRY-A EUROPEAN JOURNAL

Small Molecule Antagonists of Integrin Receptors

(2010) A. Perdih et al.   CURRENT MEDICINAL CHEMISTRY

Click-Chemistry-Derived Triazole Ligands of Arginine−Glycine−Aspartate (RGD) Integrins with a Broad Capacity To Inhibit Adhesion of Melanoma Cells and Both in Vitro and in Vivo Angiogenesis

(2010) Andrea Trabocchi et al.   JOURNAL OF MEDICINAL CHEMISTRY

Unknown

(2010) Miguel Lopez-Lazaro   MOLECULAR MEDICINE

Towards novel paradigms for cancer therapy

(2010) V Pavet et al.   ONCOGENE

Ligands for Mapping αvβ3-Integrin Expression in Vivo

(2009) Margret Schottelius et al.   ACCOUNTS OF CHEMICAL RESEARCH

Mapping the ligand-binding pocket of integrin α5β1 using a gain-of-function approach

(2009) A. Paul Mould et al.   BIOCHEMICAL JOURNAL

Integrins

(2009) Malgorzata Barczyk et al.   CELL AND TISSUE RESEARCH

Cyclic RGD-Containing Functionalized Azabicycloalkane Peptides as Potent Integrin Antagonists for Tumor Targeting

(2009) Leonardo Manzoni et al.   ChemMedChem

 5 1-Integrin controls ebolavirus entry by regulating endosomal cathepsins

(2009) K. L. Schornberg et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

A convenient synthesis of functionalized isoxazolines and related 5-hydroxyisoxazolidine-4-carboxylates

(2009) Fides Benfatti et al.   TETRAHEDRON

Investigations on synthesis of indole based constrained mimetic scaffolds through 1,3-dipolar cycloadditions of the C-(3-indolyl)-N-phenylnitrone with a variety of olefinic and allenic dipolarophiles under microwave irradiation

(2009) Surinderjit Singh Bhella et al.   TETRAHEDRON

Expanding the repertoire of small molecule transcriptional activation domains

(2008) Ryan J. Casey et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Rational Design of Highly Active and Selective Ligands for the α5β1 Integrin Receptor

(2008) Dominik Heckmann et al.   CHEMBIOCHEM

ANTI-ADHESION Evolves To a Promising Therapeutic Concept in Oncology

(2008) R. Schmidmaier et al.   CURRENT MEDICINAL CHEMISTRY

Synthesis of Ethyl 5-Hydroxyisoxazolidine-4-carboxylates via Michael Addition/Intramolecular Hemiketalisation

(2008) Fides Benfatti et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Integrin-associated proteins as potential therapeutic targets

(2008) Joseph M. Cantor et al.   IMMUNOLOGICAL REVIEWS

Multi-target-Directed Ligands To Combat Neurodegenerative Diseases

(2008) Andrea Cavalli et al.   JOURNAL OF MEDICINAL CHEMISTRY

Transcriptional activation of human mu-opioid receptor gene by insulin-like growth factor-I in neuronal cells is modulated by the transcription factor REST

(2008) Andrea Bedini et al.   JOURNAL OF NEUROCHEMISTRY

Molecular imaging in drug development

(2008) Jürgen K. Willmann et al.   NATURE REVIEWS DRUG DISCOVERY

Lewis Acid Induced Highly Regioselective Synthesis of a New Class of Substituted Isoxazolidines

(2008) Fides Benfatti et al.   SYNLETT

Diastereoselective synthesis of d-xylo-isoxazolidinyl nucleosides

(2008) Eva Hýrošová et al.   TETRAHEDRON