Elucidation of the Structure-Activity Relationships of Apelin: Influence of Unnatural Amino Acids on Binding, Signaling, and Plasma Stability

Discovery of a Competitive Apelin Receptor (APJ) Antagonist

(2011) N. J. Maximilian Macaluso et al.   ChemMedChem

Communication: The electrostatic polarization is essential to differentiate the helical propensity in polyalanine mutants

(2011) Caiyi Wei et al.   JOURNAL OF CHEMICAL PHYSICS

Apelin and APJ regulation in adipose tissue and skeletal muscle of type 2 diabetic mice and humans

(2010) Cédric Dray et al.   AMERICAN JOURNAL OF PHYSIOLOGY-ENDOCRINOLOGY AND METABOLISM

Apelin Attenuates Hyperoxic Lung and Heart Injury in Neonatal Rats

(2010) Yvonne P. de Visser et al.   AMERICAN JOURNAL OF RESPIRATORY AND CRITICAL CARE MEDICINE

Participation de l’apéline à la régulation de l’équilibre hydrique, de l’homéostasie glucidique et des fonctions cardiovasculaires

(2010) L. Bodineau et al.   ANNALES D ENDOCRINOLOGIE

The fate of the internalized apelin receptor is determined by different isoforms of apelin mediating differential interaction with β-arrestin

(2010) Dennis K. Lee et al.   BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS

Exploring the ‘RPRL’ Motif of Apelin-13 through Molecular Simulation and Biological Evaluation of Cyclic Peptide Analogues

(2010) N. J. Maximilian Macaluso et al.   ChemMedChem

Apelin Decreases Lipolysis via Gq, Gi, and AMPK-Dependent Mechanisms

(2010) Patrick Yue et al.   ENDOCRINOLOGY

By Interacting with the C-terminal Phe of Apelin, Phe255and Trp259in Helix VI of the Apelin Receptor Are Critical for Internalization

(2010) Xavier Iturrioz et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Myocardial Apelin Production is Reduced in Humans With Left Ventricular Systolic Dysfunction

(2010) Badrinathan Chandrasekaran et al.   JOURNAL OF CARDIAC FAILURE

Apelin Expression in Human Non-small Cell Lung Cancer: Role in Angiogenesis and Prognosis

(2010) Judit Berta et al.   Journal of Thoracic Oncology

International Union of Basic and Clinical Pharmacology. LXXIV. Apelin Receptor Nomenclature, Distribution, Pharmacology, and Function

(2010) S. L. Pitkin et al.   PHARMACOLOGICAL REVIEWS

Structural Insight into G-Protein Coupled Receptor Binding by Apelin†

(2009) David N. Langelaan et al.   BIOCHEMISTRY

Identification and pharmacological properties of E339-3D6, the first nonpeptidic apelin receptor agonist

(2009) Xavier Iturrioz et al.   FASEB JOURNAL

Supraspinal administration of apelin-13 induces antinociception via the opioid receptor in mice

(2009) Ning Xu et al.   PEPTIDES

Apelin protects heart against ischemia/reperfusion injury in rat

(2009) Xiang Jun Zeng et al.   PEPTIDES

The apelin–APJ system in heart failure

(2008) Alan G. Japp et al.   BIOCHEMICAL PHARMACOLOGY

Apelin Stimulates Glucose Utilization in Normal and Obese Insulin-Resistant Mice

(2008) Cédric Dray et al.   Cell Metabolism

Vascular Effects of Apelin In Vivo in Man

(2008) Alan G. Japp et al.   JOURNAL OF THE AMERICAN COLLEGE OF CARDIOLOGY