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Discovery of 1-(2,4-Dichlorophenyl)-4-ethyl-5-(5-(2-(4-(trifluoromethyl)phenyl)ethynyl)thiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide as a Potential Peripheral Cannabinoid-1 Receptor Inverse Agonist

CHEMMEDCHEM (2010)

Journal

CHEMMEDCHEM

Volume 5, Issue 9, Pages 1439-1443

Publisher

WILEY-V C H VERLAG GMBH

DOI: 10.1002/cmdc.201000246

Keywords

blood-brain barrier; brain-to-plasma ratio; cannabinoid-1 receptor; central nervous system; diet-induced obesity

Funding

National Health Research Institutes
National Science Council of the Republic of China [NSC 96-2323-B-400-001]

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Discovery of 1-(2,4-Dichlorophenyl)-4-ethyl-5-(5-(2-(4-(trifluoromethyl)phenyl)ethynyl)thiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide as a Potential Peripheral Cannabinoid-1 Receptor Inverse Agonist

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CHEMMEDCHEM

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WILEY-V C H VERLAG GMBH

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Discovery of 1-(2,4-Dichlorophenyl)-4-ethyl-5-(5-(2-(4-(trifluoromethyl)phenyl)ethynyl)thiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide as a Potential Peripheral Cannabinoid-1 Receptor Inverse Agonist

Journal

CHEMMEDCHEM

Publisher

WILEY-V C H VERLAG GMBH

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Funding

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