Efficient Synthesis of 1,2,3-Triazoles by Copper-Mediated CN and NN Bond Formation Starting FromN-Tosylhydrazones and Amines

Ligand-enabled cross-coupling of C(sp3)–H bonds with arylboron reagents via Pd(II)/Pd(0) catalysis

(2014) Kelvin S. L. Chan et al.   Nature Chemistry

Copper-Mediated Synthesis of 1,2,3-Triazoles fromN-Tosylhydrazones and Anilines

(2013) Zhengkai Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Click Chemistry for Drug Development and Diverse Chemical–Biology Applications

(2013) Prakasam Thirumurugan et al.   CHEMICAL REVIEWS

Clicking 3′-Azidothymidine into Novel Potent Inhibitors of Human Immunodeficiency Virus

(2013) Venkata Ramana Sirivolu et al.   JOURNAL OF MEDICINAL CHEMISTRY

Pd(II)-Catalyzed ortho- or meta-C–H Olefination of Phenol Derivatives

(2013) Hui-Xiong Dai et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Cross-Coupling of Remote meta-C–H Bonds Directed by a U-Shaped Template

(2013) Li Wan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Hybrid Bombesin Analogues: Combining an Agonist and an Antagonist in Defined Distances for Optimized Tumor Targeting

(2013) Carsten Kroll et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

RhIII/CuII-Cocatalyzed Synthesis of 1H-Indazoles through C–H Amidation and N–N Bond Formation

(2013) Da-Gang Yu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Ligand-Accelerated ortho-C–H Alkylation of Arylcarboxylic Acids using Alkyl Boron Reagents

(2013) Peter S. Thuy-Boun et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of 2α-Heteroarylalkyl Active Vitamin D3 with Therapeutic Effect on Enhancing Bone Mineral Density in Vivo

(2013) Miki Matsuo et al.   ACS Medicinal Chemistry Letters

Traceless Tosylhydrazone-Based Triazole Formation: A Metal-Free Alternative to Strain-Promoted Azide-Alkyne Cycloaddition

(2012) Sander S. van Berkel et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of Symmetrical and Unsymmetrical N,N′-Diaryl Guanidines via Copper/N-Methylglycine-Catalyzed Arylation of Guanidine Nitrate

(2012) Hui Xing et al.   JOURNAL OF ORGANIC CHEMISTRY

Carboxylate-Assisted Transition-Metal-Catalyzed C−H Bond Functionalizations: Mechanism and Scope

(2011) Lutz Ackermann   CHEMICAL REVIEWS

Organocatalytic Synthesis of 1,2,3-Triazoles from Unactivated Ketones and Arylazides

(2011) Mokhtaria Belkheira et al.   CHEMISTRY-A EUROPEAN JOURNAL

Organocatalytic Enamide-Azide Cycloaddition Reactions: Regiospecific Synthesis of 1,4,5-Trisubstituted-1,2,3-Triazoles

(2011) Lee Jin Tu Danence et al.   CHEMISTRY-A EUROPEAN JOURNAL

Non-Peptide Macrocyclic Histone Deacetylase Inhibitors Derived from Tricyclic Ketolide Skeleton

(2010) Sandra C. Mwakwari et al.   JOURNAL OF MEDICINAL CHEMISTRY

Copper-Catalyzed Azide-Alkyne Cycloaddition: Regioselective Synthesis of 1,4,5-Trisubstituted 1,2,3-Triazoles

(2009) Christian Spiteri et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper(I)-Catalyzed Cycloaddition of Organic Azides and 1-Iodoalkynes

(2009) Jason E. Hein et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

1,1′-Disubstituted Ferrocenes as Molecular Hinges in Mono- and Bivalent Dopamine Receptor Ligands

(2009) Daniela Huber et al.   JOURNAL OF MEDICINAL CHEMISTRY

Amino acid-promoted Ullmann-type coupling reactions and their applications in organic synthesis

(2009) Qian Cai et al.   PURE AND APPLIED CHEMISTRY

Copper/Amino Acid Catalyzed Cross-Couplings of Aryl and Vinyl Halides with Nucleophiles†

(2008) Dawei Ma et al.   ACCOUNTS OF CHEMICAL RESEARCH

Cu-Catalyzed Azide−Alkyne Cycloaddition

(2008) Morten Meldal et al.   CHEMICAL REVIEWS

Amino Acid-Catalyzed Cascade [3+2]-Cycloaddition/Hydrolysis Reactions Based on the Push-Pull Dienamine Platform: Synthesis of Highly FunctionalizedNH-1,2,3-Triazoles

(2008) Dhevalapally B. Ramachary et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis of 1-Amino-1H-indole-3-carboxylates by Copper(I)-Catalyzed Intramolecular Amination of Aryl Bromides

(2008) Ferdinand Melkonyan et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

A One-Pot Coupling/Hydrolysis/Condensation Process to Pyrrolo[1,2-a]quinoxaline

(2008) Qiliang Yuan et al.   JOURNAL OF ORGANIC CHEMISTRY

Ruthenium-Catalyzed Azide−Alkyne Cycloaddition: Scope and Mechanism

(2008) Brant C. Boren et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Elaboration of 2-(Trifluoromethyl)indoles via a Cascade Coupling/Condensation/Deacylation Process

(2008) Yu Chen et al.   ORGANIC LETTERS