Bivalent Enzyme Inhibitors Discovered Using Dynamic Covalent Chemistry

Dynamic Combinatorial Mass Spectrometry Leads to Inhibitors of a 2-Oxoglutarate-Dependent Nucleic Acid Demethylase

(2012) Esther C. Y. Woon et al.   JOURNAL OF MEDICINAL CHEMISTRY

Dynamic Hydrogels with an Environmental Adaptive Self-Healing Ability and Dual Responsive Sol–Gel Transitions

(2012) Guohua Deng et al.   ACS Macro Letters

4-Aminophenylalanine as a Biocompatible Nucleophilic Catalyst for Hydrazone Ligations at Low Temperature and Neutral pH

(2011) Adam R. Blanden et al.   BIOCONJUGATE CHEMISTRY

From static to dynamic: escaping kinetic traps in hydrazone-based dynamic combinatorial libraries

(2011) Sophie R. Beeren et al.   CHEMICAL COMMUNICATIONS

Ternary resin-bound dynamic combinatorial chemistry

(2011) Anna V. Gromova et al.   CHEMICAL COMMUNICATIONS

Potent and Selective Inhibitors of GlutathioneS-Transferase Omega 1 That Impair Cancer Drug Resistance

(2011) Katsunori Tsuboi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Discovery of Linear Receptors for Multiple Dihydrogen Phosphate Ions Using Dynamic Combinatorial Chemistry

(2011) Sophie R. Beeren et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Ferrocene-amino acid macrocycles as hydrazone-based receptors for anions

(2011) Sophie R. Beeren et al.   Chemical Science

Isozyme-Specific Fluorescent Inhibitor of GlutathioneS-Transferase Omega 1

(2010) Junghyun Son et al.   ACS Chemical Biology

Nucleophilic catalysis of acylhydrazone equilibration for protein-directed dynamic covalent chemistry

(2010) Venugopal T. Bhat et al.   Nature Chemistry

Dynamic combinatorial chemistry with hydrazones: cholate-based building blocks and libraries

(2010) Mark G. Simpson et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Dynamic combinatorial chemistry with hydrazones: libraries incorporating heterocyclic and steroidal motifs

(2010) Mark G. Simpson et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Rational Design of an Organometallic Glutathione Transferase Inhibitor

(2009) Wee Han Ang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Structural Basis for the Binding of the Anticancer Compound 6-(7-Nitro-2,1,3-Benzoxadiazol-4-Ylthio)Hexanol to Human Glutathione S-Transferases

(2009) L. Federici et al.   CANCER RESEARCH

Overcoming the Drug Resistance in Breast Cancer Cells by Rational Design of Efficient GlutathioneS-Transferase Inhibitors

(2009) Wen-Shan Li et al.   ORGANIC LETTERS

Inhibition of human glutathioneS-transferases by curcumin and analogues

(2009) R. Appiah-Opong et al.   XENOBIOTICA

Dynamic Combinatorial Mass Spectrometry Leads to Metallo-β-lactamase Inhibitors

(2008) Benoît M. R. Liénard et al.   JOURNAL OF MEDICINAL CHEMISTRY

Exploring the Relation between Amplification and Binding in Dynamic Combinatorial Libraries of Macrocyclic Synthetic Receptors in Water

(2007) Peter T. Corbett et al.   CHEMISTRY-A EUROPEAN JOURNAL