Enantioselective Organocatalytic One-Pot Amination/aza-Michael/Aldol Condensation Reaction Sequence: Synthesis of 3-Pyrrolines with a Quaternary Stereocenter

Organocatalytic Enantioselective Synthesis of Pyrazolidines, Pyrazolines and Pyrazolidinones

(2012) Maitane Fernández et al.   ADVANCED SYNTHESIS & CATALYSIS

Cinchona Alkaloid-Catalyzed Enantioselective Amination of α,β-Unsaturated Ketones: An Asymmetric Approach to Δ2-Pyrazolines

(2011) Nathaniel R. Campbell et al.   ADVANCED SYNTHESIS & CATALYSIS

Versatile Enantioselective [3+2] Cyclization between Imines and Allenoates Catalyzed by Dipeptide-Based Phosphines

(2011) Xiaoyu Han et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The Marriage of Organocatalysis with Metal Catalysis: Access to Multisubstituted Chiral 2,5-Dihydropyrroles by Cascade Iminium/Enamine-Metal Cooperative Catalysis

(2011) Wangsheng Sun et al.   CHEMISTRY-A EUROPEAN JOURNAL

Total Synthesis of Chloptosin: A Dimeric Cyclohexapeptide

(2011) Alexander J. Oelke et al.   CHEMISTRY-A EUROPEAN JOURNAL

Organocatalyzed Aziridination of α-Branched Enals: Enantioselective Synthesis of Aziridines with a Quaternary Stereo­center

(2011) Alaric Desmarchelier et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Grandilodines A−C, Biologically Active Indole Alkaloids fromKopsia grandifolia

(2011) Wai-Sum Yap et al.   JOURNAL OF NATURAL PRODUCTS

Stereoselective Organocatalytic One-Pot α,α-Bifunctionalization of Acetaldehyde by a Tandem Mannich Reaction/Electrophilic Amination

(2011) Vincent Coeffard et al.   ORGANIC LETTERS

Lewis Acid-catalyzed [3 + 2]Cyclo-addition of Alkynes withN-Tosyl-aziridines via Carbon–Carbon Bond Cleavage: Synthesis of Highly Substituted 3-Pyrrolines

(2011) Lei Li et al.   ORGANIC LETTERS

Primary amine catalyzed electrophilic amination of α,α-disubstituted aldehydes

(2011) Alaric Desmarchelier et al.   TETRAHEDRON LETTERS

Enantioselective Phase-Transfer Catalysis: Synthesis of Pyrazolines

(2010) Olivier Mahé et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Total Synthesis of Chloptosin

(2010) Alexander J. Oelke et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Diversity Through a Branched Reaction Pathway: Generation of Multicyclic Scaffolds and Identification of Antimigratory Agents

(2010) Zhiming Wang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Concise Formal Synthesis of (−)-Salinosporamide A (Marizomib) Using a Regio- and Stereoselective Epoxidation and Reductive Oxirane Ring-Opening Strategy

(2010) Taotao Ling et al.   JOURNAL OF ORGANIC CHEMISTRY

Asymmetric Synthesis of Sphinganine and Clavaminol H

(2010) Ramzi Ait-Youcef et al.   JOURNAL OF ORGANIC CHEMISTRY

Asymmetric organocatalytic Michael–α-amination sequence for the construction of a quaternary stereocenter

(2010) Alaric Desmarchelier et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Creative approaches towards the synthesis of 2,5-dihydro- furans, thiophenes, and pyrroles. One method does not fit all!

(2009) Matthew Brichacek et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Kinesin Spindle Protein (KSP) Inhibitors. 9. Discovery of (2S)-4-(2,5-Difluorophenyl)-N-[(3R,4S)-3-fluoro-1-methylpiperidin-4-yl]-2-(hydroxymethyl)-N-methyl-2-phenyl-2,5-dihydro-1H-pyrrole-1-carboxamide (MK-0731) for the Treatment of Taxane-Refractory Cancer

(2008) Christopher D. Cox et al.   JOURNAL OF MEDICINAL CHEMISTRY

Cooperative, Highly Enantioselective Phosphinothiourea Catalysis of Imine−Allene [3 + 2] Cycloadditions

(2008) Yuan-Qing Fang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY