A New Benzotriazole-Mediated Stereoflexible Gateway to Hetero-2,5-diketopiperazines

Structure, Bioactivity and Synthesis of Natural Products with Hexahydropyrrolo[2,3-b]indole

(2011) Pau Ruiz-Sanchis et al.   CHEMISTRY-A EUROPEAN JOURNAL

Nocardioazines: A Novel Bridged Diketopiperazine Scaffold from a Marine-Derived Bacterium Inhibits P-Glycoprotein

(2011) Ritesh Raju et al.   ORGANIC LETTERS

Asymmetic Organocatalytic 1,3-Dipolar Cycloaddition of Azomethine Ylide to Methyl 2-(2-Nitrophenyl)acrylate for the Synthesis of Diastereoisomers of Spirotryprostatin A

(2011) Mou-Nuo Cheng et al.   ORGANIC LETTERS

A scaleable formal total synthesis of dehydrogliotoxin

(2011) Travis C. McMahon et al.   TETRAHEDRON LETTERS

Total Synthesis of Tryprostatins A and B

(2010) Takayuki Yamakawa et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Design, synthesis, and structure–activity relationship study of bicyclic piperazine analogs of indole-3-carboxamides as novel cannabinoid CB1 receptor agonists

(2010) Elizabeth M. Moir et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Stereoselective ring contraction of 2,5-diketopiperazines: An innovative approach to the synthesis of promising bioactive 5-membered scaffolds

(2010) Thibault Coursindel et al.   BIOORGANIC CHEMISTRY

Bifunctional 2,5-Diketopiperazines as Rigid Three-Dimensional Scaffolds in Receptors and Peptidomimetics

(2010) Ana Sofia M. Ressurreição et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

An Efficient and General Method for the Stereodivergent Syntheses of Tadalafil-Like Tetracyclic Compounds

(2010) Sen Xiao et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Macrocyclization of Linear Peptides Enabled by Amphoteric Molecules

(2010) Ryan Hili et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Concise total synthesis and structural revision of (+)-pestalazine B

(2010) Carlos Pérez-Balado et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Annulated Diketopiperazines from Dipeptides or Schöllkopf Reagents via Tandem Cyclization−Intramolecular N-Arylation

(2010) Hwan Jung Lim et al.   ORGANIC LETTERS

An efficient green synthesis of proline-based cyclic dipeptides under water-mediated catalyst-free conditions

(2010) Habeebullah Thajudeen et al.   TETRAHEDRON LETTERS

First total synthesis and stereochemical revision of okaramine M

(2010) Toshimasa Iizuka et al.   TETRAHEDRON LETTERS

A straightforward synthesis and partial hydrolysis of cysteine-derived 2,5-diketopiperazines

(2010) Daniela Iannotta et al.   TETRAHEDRON LETTERS

New and Unexpected Insights into the Modulation of LuxR-Type Quorum Sensing by Cyclic Dipeptides

(2009) Jennifer Campbell et al.   ACS Chemical Biology

Synthesis of Proline-Based Diketopiperazine Scaffolds

(2009) N. Deppermann et al.   JOURNAL OF ORGANIC CHEMISTRY

Regioselective and sequential reactivity of activated 2,5-diketopiperazines

(2009) Daniel Farran et al.   JOURNAL OF PEPTIDE SCIENCE

The thaxtomin phytotoxins: Sources, synthesis, biosynthesis, biotransformation and biological activity

(2009) Russell R. King et al.   PHYTOCHEMISTRY

Chiral Acylation with N-(Protected α-Aminoacyl)benzotriazoles for Advantageous Syntheses of Peptides and Peptide Conjugates

(2009) Alan Katritzky et al.   SYNLETT

Novel and facile solution-phase synthesis of 2,5-diketopiperazines and O-glycosylated analogs

(2009) Vanessa L. Campo et al.   TETRAHEDRON

Concise Total Synthesis of (+)-WIN 64821 and (−)-Ditryptophenaline

(2008) Mohammad Movassaghi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis and structure–activity relationship studies on tryprostatin A, an inhibitor of breast cancer resistance protein

(2008) Hiteshkumar D. Jain et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Microwave-Assisted Stereoselective One-Pot Synthesis of Symmetrical and Unsymmetrical 2,5-Diketopiperazines from Unprotected Amino Acids

(2008) Manuel Jainta et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

The Total Synthesis of Roquefortine C and a Rationale for the Thermodynamic Stability of Isoroquefortine C over Roquefortine C

(2008) Ning Shangguan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Transannular rearrangement of activated 2,5-diketopiperazines: a key route to original scaffolds

(2008) Daniel Farran et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Studies towards complex bridged alkaloids: regio- and stereocontrolled enolate chemistry of 2,5-diketopiperazines

(2008) Mark Pichowicz et al.   TETRAHEDRON

[15N]-Isotopic labeling: a suitable tool to study the reactivity of bis lactams

(2007) Thibault Coursindel et al.   TETRAHEDRON LETTERS