Microwave heating in solid-phase peptide synthesis

Fragment Condensation of C-Terminal Pseudoproline Peptides without Racemization on the Solid Phase

(2011) Christian Heinlein et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

NMR solution structure of NBD94483-502 of the nucleotide-binding domain of the Plasmodium yoelii reticulocyte-binding protein Py235

(2011) Sandip Basak et al.   FEMS MICROBIOLOGY LETTERS

cis-Apa: A Practical Linker for the Microwave-Assisted Preparation of Cyclic Pseudopeptides via RCM Cyclative Cleavage

(2011) Alice Baron et al.   JOURNAL OF ORGANIC CHEMISTRY

Microwave-Assisted Solid-Phase Aza-peptide Synthesis: Aza Scan of a PKB/Akt Inhibitor Using Aza-arginine and Aza-proline Precursors

(2011) Noam S. Freeman et al.   JOURNAL OF ORGANIC CHEMISTRY

Single-Molecule Force Spectroscopy of β-Peptides That Display Well-Defined Three-Dimensional Chemical Patterns

(2011) Claribel Acevedo-Vélez et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rapid De-O-Glycosylation Concomitant with Peptide Labeling Using Microwave Radiation and an Alkyl Amine Base

(2010) Stephanie Maniatis et al.   ANALYTICAL CHEMISTRY

Synthesis of Peptide−Protein Conjugates UsingN-Succinimidyl Carbamate Chemistry

(2010) Reda Mhidia et al.   BIOCONJUGATE CHEMISTRY

Synthesis and Splice-Redirecting Activity of Branched, Arginine-Rich Peptide Dendrimer Conjugates of Peptide Nucleic Acid Oligonucleotides

(2010) Amer F. Saleh et al.   BIOCONJUGATE CHEMISTRY

Conjugates of a Novel 7-Substituted Camptothecin with RGD-Peptides as αvβ3Integrin Ligands: An Approach to Tumor-Targeted Therapy

(2010) Alma Dal Pozzo et al.   BIOCONJUGATE CHEMISTRY

Surface Modification and Polysaccharide Deposition on BisGMA/TEGDMA Thermoset

(2010) Andrea Travan et al.   BIOMACROMOLECULES

Rational Design of Responsive Self-Assembling Peptides from Native Protein Sequences†

(2010) Hongzhou Huang et al.   BIOMACROMOLECULES

Antibacterial Activities of Short Designer Peptides: a Link between Propensity for Nanostructuring and Capacity for Membrane Destabilization

(2010) Cuixia Chen et al.   BIOMACROMOLECULES

Synthesis and structure–activity relationship studies of peptidomimetic PKB/Akt inhibitors: The significance of backbone interactions

(2010) Yftah Tal-Gan et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Anhydrotetracycline–peptide conjugates as representatives for ligand-based transactivating systems

(2010) Susanne Lochner et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Microwave assisted SPPS of amylin and its toxicity of the pure product to RIN-5F cells

(2010) Karen Muthusamy et al.   BIOPOLYMERS

Toward the total chemical synthesis of the cancer protein NY-ESO-1

(2010) Paul W. R. Harris et al.   BIOPOLYMERS

Semi-automated microwave-assisted SPPS: Optimization of protocols and synthesis of difficult sequences

(2010) Søren L. Pedersen et al.   BIOPOLYMERS

Synthesis of Peptide Amides on Safety-catch Resin with Microwave Irradiation

(2010)   BULLETIN OF THE KOREAN CHEMICAL SOCIETY

Chemical synthesis of homogeneous glycopeptides and glycoproteins

(2010) Yasuhiro Kajihara et al.   CHEMICAL RECORD

Twisted Nanotubes Formed from Ultrashort Amphiphilic Peptide I3K and Their Templating for the Fabrication of Silica Nanotubes

(2010) Hai Xu et al.   CHEMISTRY OF MATERIALS

Growth Habit Modification of Ice Crystals Using Antifreeze Glycoprotein (AFGP) Analogues

(2010) Raoul Peltier et al.   CRYSTAL GROWTH & DESIGN

Bioinorganic Chemistry of Parkinson’s Disease: Structural Determinants for the Copper-Mediated Amyloid Formation of Alpha-Synuclein

(2010) Andrés Binolfi et al.   INORGANIC CHEMISTRY

Solid-Phase Synthesis and NMR Structural Studies of the Marine Antibacterial Cyclic Tetrapeptide: Cyclo[GSPE]

(2010) Huichang Annie Lim et al.   International Journal of Peptide Research and Therapeutics

Solid Phase Synthesis of an Analogue of Insulin, A0:R glargine, That Exhibits Decreased Mitogenic Activity

(2010) Seon-Yeong Kwak et al.   International Journal of Peptide Research and Therapeutics

Use of SPR to Study the Interaction of G7-18NATE Peptide with the Grb7-SH2 Domain

(2010) Menachem J. Gunzburg et al.   International Journal of Peptide Research and Therapeutics

An Efficient Approach for the Total Synthesis of Cyclotides by Microwave Assisted Fmoc-SPPS

(2010) Sungkyu Park et al.   International Journal of Peptide Research and Therapeutics

Synthesis of “Difficult” Fluorescence Quenched Substrates of Granzyme C

(2010) Susan E. Northfield et al.   International Journal of Peptide Research and Therapeutics

Methods for Enhancing Ring Closing Metathesis Yield in Peptides: Synthesis of a Dicarba Human Growth Hormone Fragment

(2010) Bianca J. van Lierop et al.   International Journal of Peptide Research and Therapeutics

Direct Solid-Phase Synthesis of the β-Amyloid (1−42) Peptide Using Controlled Microwave Heating

(2010) Bernadett Bacsa et al.   JOURNAL OF ORGANIC CHEMISTRY

Novel Pyridinium Dyes That Enable Investigations of Peptoids at the Single-Molecule Level

(2010) Birgit Rudat et al.   JOURNAL OF PHYSICAL CHEMISTRY B

Molecular Recognition at the Membrane−Water Interface: Controlling Integral Peptide Helices by Off-Membrane Nucleobase Pairing

(2010) Philipp Erik Schneggenburger et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Bridged β3-Peptide Inhibitors of p53-hDM2 Complexation: Correlation between Affinity and Cell Permeability

(2010) Arjel D. Bautista et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of MUC1 Neoglycopeptides using efficient microwave-enhanced chaotrope-assisted click chemistry

(2010) Dong Jun Lee et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Efficient Microwave-Assisted Synthesis of Human Islet Amyloid Polypeptide Designed to Facilitate the Specific Incorporation of Labeled Amino Acids

(2010) Peter Marek et al.   ORGANIC LETTERS

Understanding microwave heating effects in single mode type cavities—theory and experiment

(2010) John Robinson et al.   PHYSICAL CHEMISTRY CHEMICAL PHYSICS

Hot or not—the influence of elevated temperature and microwave irradiation on the solid phase synthesis of an affibody

(2010) Felix Nissen et al.   TETRAHEDRON LETTERS

Synthesis and antifreeze activity of fish antifreeze glycoproteins and their analogues

(2010) Raoul Peltier et al.   Chemical Science

Synthesis of a 68Ga-Labeled Peptoid−Peptide Hybrid for Imaging of Neurotensin Receptor Expression in Vivo

(2010) Simone Maschauer et al.   ACS Medicinal Chemistry Letters

Antifreeze glycopeptide analogues: microwave-enhanced synthesis and functional studies

(2009) Carolin Heggemann et al.   AMINO ACIDS

One-bead, one-compound peptide library sequencing via high-pressure ammonia cleavage coupled to nanomanipulation/nanoelectrospray ionization mass spectrometry

(2009) Jennifer M. Brown et al.   ANALYTICAL BIOCHEMISTRY

Fmoc Solid-Phase Synthesis of C-Terminal Peptide Thioesters by Formation of a Backbone Pyroglutamyl Imide Moiety

(2009) A. Pernille Tofteng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Tumor-Associated MUC1 Tandem-Repeat Glycopeptide Microarrays to Evaluate Serum- and Monoclonal-Antibody Specificity

(2009) Ulrika Westerlind et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Functional Neoglycopeptides: Synthesis and Characterization of a New Class of MUC1 Glycoprotein Models Having Core 2-BasedO-Glycan and Complex-TypeN-Glycan Chains

(2009) Takahiko Matsushita et al.   BIOCHEMISTRY

Release of Liposomal Contents by Cell-Secreted Matrix Metalloproteinase-9

(2009) Jayati Banerjee et al.   BIOCONJUGATE CHEMISTRY

Use of a Temporary “Solubilizing” Peptide Tag for the Fmoc Solid-Phase Synthesis of Human Insulin Glargine via Use of Regioselective Disulfide Bond Formation

(2009) Mohammed Akhter Hossain et al.   BIOCONJUGATE CHEMISTRY

Effect of Peptide Sequence on Surface Properties and Self-Assembly of an Amphiphilic pH-Responsive Peptide

(2009) Jeanne N. Shera et al.   BIOMACROMOLECULES

Peptide inhibitors of HIV-1 integrase: From mechanistic studies to improved lead compounds

(2009) Michal Maes et al.   BIOORGANIC & MEDICINAL CHEMISTRY

β-Peptides with improved affinity for hDM2 and hDMX

(2009) Elizabeth A. Harker et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Identification of a β3-peptide HIV fusion inhibitor with improved potency in live cells

(2009) Arjel D. Bautista et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

VCD spectroscopic properties of the β-hairpin forming miniprotein CLN025 in various solvents

(2009) Marcus P. D. Hatfield et al.   BIOPOLYMERS

Regioselective formation of interlocked dicarba bridges in naturally occurring cyclic peptide toxins using olefin metathesis

(2009) Andrea J. Robinson et al.   CHEMICAL COMMUNICATIONS

COMU: A Safer and More Effective Replacement for Benzotriazole-Based Uronium Coupling Reagents

(2009) Ayman El-Faham et al.   CHEMISTRY-A EUROPEAN JOURNAL

Oxyma: An Efficient Additive for Peptide Synthesis to Replace the Benzotriazole-Based HOBt and HOAt with a Lower Risk of Explosion[1]

(2009) Ramon Subirós-Funosas et al.   CHEMISTRY-A EUROPEAN JOURNAL

Solid phase synthesis of fatty acid modified glucagon-like peptide-1 (7-36) amide under thermal and controlled microwave irradiation

(2009) Shuai Jian Ni et al.   CHINESE CHEMICAL LETTERS

Identification and Suppression of β-Elimination Byproducts Arising from the Use of Fmoc-Ser(PO3Bzl,H)-OH in Peptide Synthesis

(2009) Troy J. Attard et al.   International Journal of Peptide Research and Therapeutics

Computational Design of Highly Selective Antimicrobial Peptides

(2009) Davor Juretić et al.   Journal of Chemical Information and Modeling

Discovery of Small Peptides Derived from Embryonic Lethal Abnormal Vision Proteins Structure Showing RNA-Stabilizing Properties

(2009) Daniela Rossi et al.   JOURNAL OF MEDICINAL CHEMISTRY

Benzotriazole-Assisted Solid-Phase Assembly of Leu-Enkephalin, Amyloid β segment 34−42, and other “Difficult” Peptide Sequences

(2009) Alan R. Katritzky et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis and Characterization of Nitroaromatic Peptoids: Fine Tuning Peptoid Secondary Structure through Monomer Position and Functionality

(2009) Sarah A. Fowler et al.   JOURNAL OF ORGANIC CHEMISTRY

Microwave-assisted solid-phase peptide synthesis at 60 °C: alternative conditions with low enantiomerization

(2009) Carina Loffredo et al.   JOURNAL OF PEPTIDE SCIENCE

Microwave-assisted TFA cleavage of peptides from Merrifield resin

(2009) Alicja Kluczyk et al.   JOURNAL OF PEPTIDE SCIENCE

New Strategies for the Design of Folded Peptoids Revealed by a Survey of Noncovalent Interactions in Model Systems

(2009) Benjamin C. Gorske et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Pleomorphic Copper Coordination by Alzheimer’s Disease Amyloid-β Peptide

(2009) Simon C. Drew et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

An Essential Epitope of Anti-MUC1 Monoclonal Antibody KL-6 Revealed by Focused Glycopeptide Library

(2009) Naoki Ohyabu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A Preliminary Survey of the Peptoid Folding Landscape

(2009) Glenn L. Butterfoss et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Peptides Grafted from Solids for the Control of Interfacial Properties

(2009) Wade K. J. Mosse et al.   LANGMUIR

Microwave-assisted synthesis of triple-helical, collagen-mimetic lipopeptides

(2009) Jayati Banerjee et al.   Nature Protocols

Regulation by phosphorylation of the relative affinities of the N-terminal transactivation domains of p53 for p300 domains and Mdm2

(2009) D P Teufel et al.   ONCOGENE

Solid phase synthesis and structural analysis of novel A-chain dicarba analogs of human relaxin-3 (INSL7) that exhibit full biological activity

(2009) Mohammed Akhter Hossain et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Development of a new microwave-assisted cleavable backbone amide linker (BAL): a comparative study

(2009) Stijn Claerhout et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis of Fish Antifreeze Neoglycopeptides Using Microwave-Assisted “Click Chemistry”

(2009) Nicole Miller et al.   ORGANIC LETTERS

Microwave irradiation and COMU: a potent combination for solid-phase peptide synthesis

(2009) Ramon Subiros-Funosas et al.   TETRAHEDRON LETTERS

N-Methylation of Peptides: A New Perspective in Medicinal Chemistry

(2008) Jayanta Chatterjee et al.   ACCOUNTS OF CHEMICAL RESEARCH

Solid-Phase Synthesis of Europium-Labeled Human INSL3 as a Novel Probe for the Study of Ligand−Receptor Interactions

(2008) Fazel Shabanpoor et al.   BIOCONJUGATE CHEMISTRY

A peptoid antagonist of VEGF Receptor 2 recognizes a ‘hotspot’ in the extracellular domain distinct from the hormone-binding site

(2008) D. Gomika Udugamasooriya et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Microwave-assisted solid phase synthesis, PEGylation, and biological activity studies of glucagon-like peptide-1(7–36) amide

(2008) Yushi Chi et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Search for α-helical propensity in the receptor-bound conformation of glucagon-like peptide-1

(2008) Eunice N. Murage et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Novel insights into GPCR—Peptide interactions: Mutations in extracellular loop 1, ligand backbone methylations and molecular modeling of neurotensin receptor 1

(2008) Steffen Härterich et al.   BIOORGANIC & MEDICINAL CHEMISTRY

High-throughput evaluation of relative cell permeability between peptoids and peptides

(2008) Niclas C. Tan et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis, penetrability and intracellular targeting of fluorescein-tagged peptoids and peptide–peptoid hybrids

(2008) Asier Unciti-Broceta et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Ferrocenyl glycopeptides as electrochemical probes to detect autoantibodies in multiple sclerosis patients' sera

(2008) Feliciana Real-Fernández et al.   BIOPOLYMERS

Enhanced microwave-assisted method for on-bead disulfide bond formation: Synthesis of α-conotoxin MII

(2008) Athanassios S. Galanis et al.   BIOPOLYMERS

Total Synthesis of desB30 Insulin Analogues by Biomimetic Folding of Single-Chain Precursors

(2008) A. Pernille Tofteng et al.   CHEMBIOCHEM

Glycoprotein Synthesis: An Update

(2008) David P. Gamblin et al.   CHEMICAL REVIEWS

Microwave-assisted Solid Phase Peptide Synthesis on High Loaded Resins

(2008) Stéphanie Coantic et al.   International Journal of Peptide Research and Therapeutics

The Synthesis of Phosphopeptides Using Microwave-assisted Solid Phase Peptide Synthesis

(2008) Paul W. R. Harris et al.   International Journal of Peptide Research and Therapeutics

Exploration of Structure−Activity Relationships among Foldamer Ligands for a Specific Protein Binding Site via Parallel and Split-and-Mix Library Synthesis

(2008) Justin K. Murray et al.   JOURNAL OF COMBINATORIAL CHEMISTRY

Synthesis of a Positional Scanning Library of Pentamers ofN-Alkylglycines Assisted by Microwave Activation and Validation via the Identification of Trypsin Inhibitors

(2008) Joaquim Messeguer et al.   JOURNAL OF COMBINATORIAL CHEMISTRY

Designed Glycopeptides with Different β-Turn Types as Synthetic Probes for the Detection of Autoantibodies as Biomarkers of Multiple Sclerosis

(2008) Alfonso Carotenuto et al.   JOURNAL OF MEDICINAL CHEMISTRY

Identification of Potent, Selective, and Metabolically Stable Peptide Antagonists to the Calcitonin Gene-Related Peptide (CGRP) Receptor

(2008) Les P. Miranda et al.   JOURNAL OF MEDICINAL CHEMISTRY

Solid-Phase Synthesis of Difficult Peptide Sequences at Elevated Temperatures: A Critical Comparison of Microwave and Conventional Heating Technologies

(2008) Bernadett Bacsa et al.   JOURNAL OF ORGANIC CHEMISTRY

Peptide-Based SAMs that Resist the Adsorption of Proteins

(2008) Rolf Chelmowski et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Toward β-Amino Acid Proteins:  Design, Synthesis, and Characterization of a Fifteen Kilodalton β-Peptide Tetramer

(2008) E. James Petersson et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Adsorption of a Statherin Peptide Fragment on the Surface of Nanocrystallites of Hydroxyapatite

(2008) Peng-Huan Chen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Mechanistic Studies of the Triggered Release of Liposomal Contents by Matrix Metalloproteinase-9

(2008) Adekunle I. Elegbede et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Hydrophobic-Region-Induced Transitions in Self-Assembled Peptide Nanostructures†

(2008) Hai Xu et al.   LANGMUIR

Microwave-Assisted Solid Phase Synthesis of GLP-1-Analogues

(2008) Yushi Chi et al.   LETTERS IN ORGANIC CHEMISTRY

Distinctive Circular Dichroism Signature for 14-Helix-Bundle Formation by β-Peptides

(2008) William C. Pomerantz et al.   ORGANIC LETTERS

Scope and limitations of the designer proline-rich antibacterial peptide dimer, A3-APO, alone or in synergy with conventional antibiotics

(2008) Marco Cassone et al.   PEPTIDES

Microwave-assisted orthogonal synthesis of PNA–peptide conjugates

(2008) Nina Svensen et al.   TETRAHEDRON LETTERS

Nonthermal Microwave Effects Revisited:  On the Importance of Internal Temperature Monitoring and Agitation in Microwave Chemistry

(2007) M. Antonia Herrero et al.   JOURNAL OF ORGANIC CHEMISTRY

Microwave-assisted Boc-solid phase peptide synthesis of cyclic cysteine-rich peptides

(2007) Maša Čemažar et al.   JOURNAL OF PEPTIDE SCIENCE

Application of microwave method to the solid phase synthesis of pseudopeptides containing ester bond

(2007) Bishnu Prasad Joshi et al.   TETRAHEDRON LETTERS

Peptoid dendrimers—microwave-assisted solid-phase synthesis and transfection agent evaluation

(2007) Juan J. Diaz-Mochon et al.   TETRAHEDRON LETTERS