C–H functionalization logic in total synthesis

Highly Selective Metalations of Pyridines and Related Heterocycles Using New Frustrated Lewis Pairs or tmp-Zinc and tmp-Magnesium Bases with BF3⋅OEt2

(2010) Milica Jaric et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Fluxible Monodisperse Quantum Dots with Efficient Luminescence

(2010) Qisong Feng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of the Leu–Trp Component of the Celogentin Family of Cyclic Peptides Through a C–H Activation–Cross-Coupling Strategy

(2010) Barbara T. Y. Li et al.   AUSTRALIAN JOURNAL OF CHEMISTRY

Palladium-Catalyzed Ligand-Directed C−H Functionalization Reactions

(2010) Thomas W. Lyons et al.   CHEMICAL REVIEWS

Functional Characterization of the Cyclomarin/Cyclomarazine Prenyltransferase CymD Directs the Biosynthesis of Unnatural Cyclic Peptides⊥

(2010) Andrew W. Schultz et al.   JOURNAL OF NATURAL PRODUCTS

Synthesis of Complex Allylic Esters via C−H Oxidation vs C−C Bond Formation

(2010) Nicolaas A. Vermeulen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total Synthesis of (+)-Complanadine A Using an Iridium-Catalyzed Pyridine C−H Functionalization

(2010) Daniel F. Fischer et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Direct C−H Arylation of Electron-Deficient Heterocycles with Arylboronic Acids

(2010) Ian B. Seiple et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total synthesis of eudesmane terpenes: cyclase phase

(2010) Ke Chen et al.   TETRAHEDRON

Total Synthesis of (+)-Haplophytine

(2009) K. C. Nicolaou et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Total Synthesis of Celogentin C

(2009) Bing Ma et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Total Synthesis of Palau’amine

(2009) Ian B. Seiple et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Strain Release in CH Bond Activation?

(2009) Ke Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Stereodivergent Synthesis of 17-α and 17-β-Aryl Steroids: Application and Biological Evaluation of D-Ring Cortistatin Analogues

(2009) Jun Shi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Direct, ChemoselectiveN-tert-Prenylation of Indoles by CH Functionalization

(2009) Michael R. Luzung et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of Cyclopamine Using a Biomimetic and Diastereoselective Approach

(2009) Athanassios Giannis et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Redox Economy in Organic Synthesis

(2009) Noah Z. Burns et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Carbene Insertion into C−H Bonds

(2009) Michael P. Doyle et al.   CHEMICAL REVIEWS

C−H Activation for the Construction of C−B Bonds

(2009) Ibraheem A. I. Mkhalid et al.   CHEMICAL REVIEWS

Transition metal-catalyzed C–H activation reactions: diastereoselectivity and enantioselectivity

(2009) Ramesh Giri et al.   CHEMICAL SOCIETY REVIEWS

The economies of synthesis

(2009) Timothy Newhouse et al.   CHEMICAL SOCIETY REVIEWS

Total Synthesis of (±)-Rhazinal Using Novel Palladium-Catalyzed Cyclizations

(2009) Alfred L. Bowie et al.   JOURNAL OF ORGANIC CHEMISTRY

Nickel-Catalyzed Reaction of Arylzinc Reagents with N-Aromatic Heterocycles: A Straightforward Approach to C−H Bond Arylation of Electron-Deficient Heteroaromatic Compounds

(2009) Mamoru Tobisu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total Synthesis of the Antimitotic Bicyclic Peptide Celogentin C

(2009) Bing Ma et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective Synthesis of (+)-Cephalostatin 1

(2009) Kevin C. Fortner et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total synthesis of eudesmane terpenes by site-selective C–H oxidations

(2009) Ke Chen et al.   NATURE

Total synthesis and study of 6-deoxyerythronolide B by late-stage C–H oxidation

(2009) Erik M. Stang et al.   Nature Chemistry

Protecting-group-free synthesis as an opportunity for invention

(2009) Ian S. Young et al.   Nature Chemistry

Total Synthesis of (+)-11,11'-Dideoxyverticillin A

(2009) J. Kim et al.   SCIENCE

Enantioselective Synthesis of (+)-Monobromophakellin and (+)-Phakellin: A Concise Phakellin Annulation Strategy Applicable to Palau'amine

(2008) Shaohui Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of Rhazinicine by a Metal-Catalyzed CH Bond Functionalization Strategy

(2008) Elizabeth M. Beck et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of 1,9-Dideoxy-pre-axinellamine

(2008) Junichiro Yamaguchi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Total Synthesis of (±)-Axinellamines A and B

(2008) Daniel P. O'Malley et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Synthesis of (−)-Incarvillateine Employing an Intramolecular Alkylation via Rh-Catalyzed Olefinic C−H Bond Activation

(2008) Andy S. Tsai et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total Syntheses of (±)-Massadine and Massadine Chloride

(2008) Shun Su et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of (+)-Cortistatin A

(2008) Ryan A. Shenvi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

1,3-Diol Synthesis via Controlled, Radical-Mediated C−H Functionalization

(2008) Ke Chen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantiospecific Total Synthesis of the Hapalindoles, Fischerindoles, and Welwitindolinonesviaa Redox Economic Approach

(2008) Jeremy M. Richter et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Intermolecular Enolate Heterocoupling: Scope, Mechanism, and Application

(2008) Michael P. DeMartino et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Catalytic C–H functionalization by metal carbenoid and nitrenoid insertion

(2008) Huw M. L. Davies et al.   NATURE