Regio- and Enantioselective Synthesis of N-Substituted Pyrazoles by Rhodium-Catalyzed Asymmetric Addition to Allenes
Published 2015 View Full Article
- Home
- Publications
- Publication Search
- Publication Details
Title
Regio- and Enantioselective Synthesis of N-Substituted Pyrazoles by Rhodium-Catalyzed Asymmetric Addition to Allenes
Authors
Keywords
-
Journal
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
Volume 54, Issue 24, Pages 7149-7153
Publisher
Wiley
Online
2015-04-30
DOI
10.1002/anie.201501758
References
Ask authors/readers for more resources
Related references
Note: Only part of the references are listed.- Asymmetric Rhodium-Catalyzed Addition of Thiols to Allenes: Synthesis of Branched Allylic Thioethers and Sulfones
- (2015) Adrian B. Pritzius et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Rhodium-Catalyzed Chemo-, Regio-, and Enantioselective Addition of 2-Pyridones to Terminal Allenes
- (2014) Changkun Li et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Unlocking theN2 Selectivity of Benzotriazoles: Regiodivergent and Highly Selective Coupling of Benzotriazoles with Allenes
- (2014) Kun Xu et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Atom-Economic, Regiodivergent, and Stereoselective Coupling of Imidazole Derivatives with Terminal Allenes
- (2014) Kun Xu et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Combined Experimental and Computational Investigations of Rhodium-Catalysed CH Functionalisation of Pyrazoles with Alkenes
- (2014) Andrés G. Algarra et al. CHEMISTRY-A EUROPEAN JOURNAL
- Cu-Promoted Sydnone Cycloadditions of Alkynes: Scope and Mechanism Studies
- (2014) Júlia Comas-Barceló et al. CHEMISTRY-A EUROPEAN JOURNAL
- Rhodium-Catalyzed Chemo- and Regioselective Decarboxylative Addition of β-Ketoacids to Allenes: Efficient Construction of Tertiary and Quaternary Carbon Centers
- (2014) Changkun Li et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Synthesis of Polysubstituted Pyrazoles by a Platinum-Catalyzed Sigmatropic Rearrangement/Cyclization Cascade
- (2014) Jia-Jie Wen et al. ORGANIC LETTERS
- Single cell imaging of Bruton's Tyrosine Kinase using an irreversible inhibitor
- (2014) Anna Turetsky et al. Scientific Reports
- The design and synthesis of a potent glucagon receptor antagonist with favorable physicochemical and pharmacokinetic properties as a candidate for the treatment of type 2 diabetes mellitus
- (2013) Angel Guzman-Perez et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Synthesis of 4-Fluoromethylsydnones and their Participation in Alkyne Cycloaddition Reactions
- (2013) Robert S. Foster et al. JOURNAL OF ORGANIC CHEMISTRY
- Targeting BTK with Ibrutinib in Relapsed Chronic Lymphocytic Leukemia
- (2013) John C. Byrd et al. NEW ENGLAND JOURNAL OF MEDICINE
- Asymmetric Intramolecular Hydroamination of Allenes using Mononuclear Gold Catalysts
- (2013) Christophe Michon et al. ORGANOMETALLICS
- Organocatalytic asymmetric aza-Michael addition of pyrazole to chalcone
- (2013) Pengfei Li et al. TETRAHEDRON-ASYMMETRY
- Rhodium-catalyzed hydroformylation of alkynes employing a self-assembling ligand system
- (2013) Vladislav Agabekov et al. Chemical Science
- Enantioselective Rhodium-Catalyzed Synthesis of Branched Allylic Amines by Intermolecular Hydroamination of Terminal Allenes
- (2012) Michael L. Cooke et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Gold(I)-Catalyzed Stereoconvergent, Intermolecular Enantioselective Hydroamination of Allenes
- (2012) Kristina L. Butler et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Mechanistic Insights into a Supramolecular Self-Assembling Catalyst System: Evidence for Hydrogen Bonding during Rhodium-Catalyzed Hydroformylation
- (2012) Urs Gellrich et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- The More Gold-The More Enantioselective: Cyclohydroaminations of γ-Allenyl Sulfonamides with Mono-, Bis-, and Trisphospholane Gold(I) Catalysts
- (2012) Lara-Isabel Rodríguez et al. CHEMISTRY-A EUROPEAN JOURNAL
- Oxidative Trifluoromethylthiolations of Aryl Boronic Acids Using a Copper/O2-Based Protocol
- (2012) Cheng-Pan Zhang et al. Chemistry-An Asian Journal
- Discovery of a Novel Glucagon Receptor Antagonist N-[(4-{(1S)-1-[3-(3, 5-Dichlorophenyl)-5-(6-methoxynaphthalen-2-yl)-1H-pyrazol-1-yl]ethyl}phenyl)carbonyl]-β-alanine (MK-0893) for the Treatment of Type II Diabetes
- (2012) Yusheng Xiong et al. JOURNAL OF MEDICINAL CHEMISTRY
- Covalent Inhibitors of Interleukin-2 Inducible T Cell Kinase (Itk) with Nanomolar Potency in a Whole-Blood Assay
- (2012) Christoph W. Zapf et al. JOURNAL OF MEDICINAL CHEMISTRY
- Heterodimeric JAK–STAT activation as a mechanism of persistence to JAK2 inhibitor therapy
- (2012) Priya Koppikar et al. NATURE
- Ruxolitinib
- (2012) Ruben A. Mesa et al. NATURE REVIEWS DRUG DISCOVERY
- A Double-Blind, Placebo-Controlled Trial of Ruxolitinib for Myelofibrosis
- (2012) Srdan Verstovsek et al. NEW ENGLAND JOURNAL OF MEDICINE
- Stereoselective synthesis of novel pyrazole derivatives using tert-butansulfonamide as a chiral auxiliary
- (2012) Chang Min Park et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Redox-Neutral Atom-Economic Rhodium-Catalyzed Coupling of Terminal Alkynes with Carboxylic Acids Toward Branched Allylic Esters
- (2011) Alexandre Lumbroso et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Enantioselective Synthesis of Branched Allylic Esters via Rhodium-Catalyzed Coupling of Allenes with Carboxylic Acids
- (2011) Philipp Koschker et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Asymmetric additions to dienes catalysed by a dithiophosphoric acid
- (2011) Nathan D. Shapiro et al. NATURE
- Iridium-catalysed direct C–C coupling of methanol and allenes
- (2011) Joseph Moran et al. Nature Chemistry
- Atom economic macrolactonization and lactonization viaredox-neutral rhodium-catalyzed coupling of terminal alkynes with carboxylic acids
- (2011) Alexandre Lumbroso et al. Chemical Science
- The interplay of hydrogen bonds and halogen bonds in the structure of NH-pyrazoles bearing C-aryl and C-halogen substituents
- (2010) M. Ángeles García et al. INORGANICA CHIMICA ACTA
- Scope and Mechanism of Allylic C−H Amination of Terminal Alkenes by the Palladium/PhI(OPiv)2Catalyst System: Insights into the Effect of Naphthoquinone
- (2010) Guoyin Yin et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Rhodium-catalyzed asymmetric hydroalkoxylation and hydrosulfenylation of diphenylphosphinylallenes
- (2009) Takahiro Kawamoto et al. CHEMICAL COMMUNICATIONS
- Enantioselective Synthesis of Janus Kinase Inhibitor INCB018424 via an Organocatalytic Aza-Michael Reaction
- (2009) Qiyan Lin et al. ORGANIC LETTERS
- Enantioselective Synthesis of β-(3-Hydroxypyrazol-1-yl) Ketones Using an Organocatalyzed Michael Addition Reaction
- (2009) Sanjib Gogoi et al. ORGANIC LETTERS
- A Highly Enantioselective Allylic Amination Reaction Using a Commercially Available Chiral Rhodium Catalyst: Resolution of Racemic Allylic Carbonates
- (2009) Derek C. Vrieze et al. ORGANIC LETTERS
- A Versatile Catalyst System for Suzuki−Miyaura Cross-Coupling Reactions of C(sp2)-Tosylates and Mesylates
- (2009) Brijesh Bhayana et al. ORGANIC LETTERS
- Synthesis of derivatives of pyrazole with chiral substituents at the nitrogen atom
- (2008) A. V. Kurkin et al. Chemistry of Heterocyclic Compounds
- Iridium-Catalyzed Hydrocarboxylation of 1,1-Dimethylallene: Byproduct-Free Reverse Prenylation of Carboxylic Acids
- (2008) In Su Kim et al. ORGANIC LETTERS
- A molecular balance to measure the strength of N–H⋯π hydrogen bonds based on the tautomeric equilibria of C-benzylphenyl substituted NH-pyrazoles
- (2008) Pilar Cornago et al. TETRAHEDRON
- A practical, two-step synthesis of 1-alkyl-4-aminopyrazoles
- (2008) Anna A. Zabierek et al. TETRAHEDRON LETTERS
- Metal-Catalyzed Enantioselective Allylation in Asymmetric Synthesis
- (2007) Zhan Lu et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
Discover Peeref hubs
Discuss science. Find collaborators. Network.
Join a conversationFind the ideal target journal for your manuscript
Explore over 38,000 international journals covering a vast array of academic fields.
Search